BRPI0912355A2 - Grupos de proteção de indolsulfonil para proteção dos grupamentos guanidino e amino - Google Patents

Grupos de proteção de indolsulfonil para proteção dos grupamentos guanidino e amino

Info

Publication number
BRPI0912355A2
BRPI0912355A2 BRPI0912355-5A BRPI0912355A BRPI0912355A2 BR PI0912355 A2 BRPI0912355 A2 BR PI0912355A2 BR PI0912355 A BRPI0912355 A BR PI0912355A BR PI0912355 A2 BRPI0912355 A2 BR PI0912355A2
Authority
BR
Brazil
Prior art keywords
indolsulfonyl
guanidine
protection
groups
amino groups
Prior art date
Application number
BRPI0912355-5A
Other languages
English (en)
Inventor
Matthieu Giraud
Fernando Albericio
Albert Isidro Llobet
Mercedes Alvarez Domingo
Original Assignee
Lonza Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lonza Ag filed Critical Lonza Ag
Publication of BRPI0912355A2 publication Critical patent/BRPI0912355A2/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BRPI0912355-5A 2008-05-05 2009-05-05 Grupos de proteção de indolsulfonil para proteção dos grupamentos guanidino e amino BRPI0912355A2 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP08008418 2008-05-05
US9570908P 2008-09-10 2008-09-10
PCT/EP2009/003210 WO2009135645A1 (en) 2008-05-05 2009-05-05 Indolesulfonyl protecting groups for protection of guanidino and amino groups

Publications (1)

Publication Number Publication Date
BRPI0912355A2 true BRPI0912355A2 (pt) 2015-07-28

Family

ID=39772857

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0912355-5A BRPI0912355A2 (pt) 2008-05-05 2009-05-05 Grupos de proteção de indolsulfonil para proteção dos grupamentos guanidino e amino

Country Status (17)

Country Link
US (1) US8431720B2 (pt)
EP (2) EP2420489B1 (pt)
JP (2) JP5567004B2 (pt)
KR (2) KR101521400B1 (pt)
CN (1) CN102026971B (pt)
AU (1) AU2009243730B2 (pt)
BR (1) BRPI0912355A2 (pt)
CA (1) CA2721644C (pt)
CO (1) CO6390068A2 (pt)
DK (1) DK2420489T3 (pt)
EA (1) EA022476B1 (pt)
ES (1) ES2477590T3 (pt)
HK (1) HK1154860A1 (pt)
IL (1) IL208930A (pt)
MX (1) MX2010012113A (pt)
WO (1) WO2009135645A1 (pt)
ZA (1) ZA201007614B (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103626996B (zh) * 2013-11-29 2016-04-27 沈阳药科大学 胍基化的含二硫键聚氨基胺类聚合物及其制备和应用
EP3305780A1 (en) 2016-10-05 2018-04-11 Lonza Ltd Method for the preparation of h-arg(mis)-oh
EP3523278A4 (en) * 2016-10-09 2020-07-15 Polypeptide Laboratories Holding (PPL) AB METHOD FOR PRODUCING H-ARG (MIS) -OH
EP3315490A1 (en) 2016-10-31 2018-05-02 Polypeptide Laboratories Holding (PPL) AB Method for the preparation of h-arg(mis)-oh

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10004572A1 (de) * 2000-02-02 2001-08-09 Boehringer Ingelheim Pharma Neue positive allosterische AMPA-Rezeptor Modulatoren (PAARM), Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
ATE340792T1 (de) 2002-02-01 2006-10-15 Hoffmann La Roche Substituierte indole als alpha-1 agonisten
CN100453537C (zh) * 2004-05-08 2009-01-21 上海依福瑞实业有限公司 一种双保护氨基酸的制备方法
US8585885B2 (en) * 2007-08-28 2013-11-19 Rohm And Haas Electronic Materials Llc Electrochemically deposited indium composites

Also Published As

Publication number Publication date
JP5567004B2 (ja) 2014-08-06
KR101493554B1 (ko) 2015-02-16
WO2009135645A1 (en) 2009-11-12
CA2721644A1 (en) 2009-11-12
US20110060125A1 (en) 2011-03-10
EP2420489B1 (en) 2014-04-23
EA022476B1 (ru) 2016-01-29
ES2477590T3 (es) 2014-07-17
EP2420489A1 (en) 2012-02-22
JP2014193872A (ja) 2014-10-09
IL208930A0 (en) 2011-01-31
CO6390068A2 (es) 2012-02-29
KR20110014167A (ko) 2011-02-10
AU2009243730A1 (en) 2009-11-12
EA201001738A1 (ru) 2011-06-30
CN102026971A (zh) 2011-04-20
CN102026971B (zh) 2014-10-29
HK1154860A1 (en) 2012-05-04
KR20140061548A (ko) 2014-05-21
JP2011519884A (ja) 2011-07-14
IL208930A (en) 2014-07-31
DK2420489T3 (da) 2014-07-21
CA2721644C (en) 2013-10-15
JP5985534B2 (ja) 2016-09-06
KR101521400B1 (ko) 2015-05-18
MX2010012113A (es) 2010-12-01
ZA201007614B (en) 2011-07-27
AU2009243730B2 (en) 2013-07-18
US8431720B2 (en) 2013-04-30
EP2280942A1 (en) 2011-02-09

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Legal Events

Date Code Title Description
B25A Requested transfer of rights approved

Owner name: POLYPEPTIDE LABORATORIES HOLDING (PPL) AB (SE)

B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 10A ANUIDADE.

B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2513 DE 06-03-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.