ZA200603402B - Methods and compositions comprising thalidomide for treatment of fibromyalgia - Google Patents
Methods and compositions comprising thalidomide for treatment of fibromyalgia Download PDFInfo
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- ZA200603402B ZA200603402B ZA200603402A ZA200603402A ZA200603402B ZA 200603402 B ZA200603402 B ZA 200603402B ZA 200603402 A ZA200603402 A ZA 200603402A ZA 200603402 A ZA200603402 A ZA 200603402A ZA 200603402 B ZA200603402 B ZA 200603402B
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- South Africa
- Prior art keywords
- thalidomide
- fibromyalgia
- stereoisomer
- active agent
- solvate
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- 229960003147 reserpine Drugs 0.000 description 1
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- 229960000371 rofecoxib Drugs 0.000 description 1
- MDMGHDFNKNZPAU-UHFFFAOYSA-N roserpine Natural products C1C2CN3CCC(C4=CC=C(OC)C=C4N4)=C4C3CC2C(OC(C)=O)C(OC)C1OC(=O)C1=CC(OC)=C(OC)C(OC)=C1 MDMGHDFNKNZPAU-UHFFFAOYSA-N 0.000 description 1
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- 229960001918 tiagabine Drugs 0.000 description 1
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Classifications
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- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
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- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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- A—HUMAN NECESSITIES
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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- A—HUMAN NECESSITIES
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/553—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one oxygen as ring hetero atoms, e.g. loxapine, staurosporine
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/60—Salicylic acid; Derivatives thereof
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- A—HUMAN NECESSITIES
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- A61P19/00—Drugs for skeletal disorders
- A61P19/04—Drugs for skeletal disorders for non-specific disorders of the connective tissue
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- A—HUMAN NECESSITIES
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- A61P25/04—Centrally acting analgesics, e.g. opioids
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- A61P25/22—Anxiolytics
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Neurosurgery (AREA)
- Neurology (AREA)
- Pain & Pain Management (AREA)
- Molecular Biology (AREA)
- Psychiatry (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US51454803P | 2003-10-24 | 2003-10-24 |
Publications (1)
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| ZA200603402B true ZA200603402B (en) | 2007-09-26 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| ZA200603402A ZA200603402B (en) | 2003-10-24 | 2004-10-22 | Methods and compositions comprising thalidomide for treatment of fibromyalgia |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20050119194A1 (fr) |
| EP (1) | EP1680132A4 (fr) |
| JP (1) | JP2007509170A (fr) |
| KR (1) | KR20060123183A (fr) |
| CN (1) | CN1897956A (fr) |
| AU (1) | AU2004283716A1 (fr) |
| BR (1) | BRPI0415651A (fr) |
| CA (1) | CA2543312A1 (fr) |
| IL (1) | IL175098A0 (fr) |
| MX (1) | MXPA06004382A (fr) |
| NZ (1) | NZ547127A (fr) |
| WO (1) | WO2005039497A2 (fr) |
| ZA (1) | ZA200603402B (fr) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20050100529A1 (en) * | 2003-11-06 | 2005-05-12 | Zeldis Jerome B. | Methods of using and compositions comprising immunomodulatory compounds for the treatment and management of asbestos-related diseases and disorders |
| WO2006105670A1 (fr) * | 2005-04-08 | 2006-10-12 | Neuromed Pharmaceuticals Ltd. | Thérapie de combinaison qui comprend un agent bloquant les canaux calciques de type n pour le soulagement de la douleur |
| US20070233211A1 (en) * | 2006-04-04 | 2007-10-04 | Galer Bradley S | Methods and compositions for treating non-neuropathic pain |
| WO2008085927A2 (fr) * | 2007-01-05 | 2008-07-17 | Combinatorx, Incorporated | Procédés, compositions et kits destinés au traitement de la douleur |
| RU2464023C2 (ru) * | 2008-05-16 | 2012-10-20 | АКСИС, Инс | Лекарственное средство для лечения фибромиалгии |
| UA106384C2 (ru) * | 2009-07-27 | 2014-08-26 | БИАЛ-ПОРТЕЛА энд КА., С.А. | ПРИМЕНЕНИЕ ПРОИЗВОДНЫХ 5H-ДИБЕНЗ/б,ф/АЗЕПИН-5-КАРБОКСАМИДА ДЛЯ ЛЕЧЕНИЯ ФИБРОМИАЛГИИ |
| JPWO2011071136A1 (ja) * | 2009-12-11 | 2013-04-22 | アステラス製薬株式会社 | 線維筋痛症治療剤 |
| US8461171B2 (en) * | 2010-02-09 | 2013-06-11 | QRxPharma Ltd. | Hybrid opioid compounds and compositions |
| JP5699030B2 (ja) * | 2010-07-05 | 2015-04-08 | Ａｘｉｓ株式会社 | エタネルセプトを含む線維筋痛症の治療剤 |
| US20130203742A1 (en) | 2012-02-06 | 2013-08-08 | William L. Pridgen | Valaciclovir and meloxicam combination therapy for functional somatic syndromes |
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| US5434170A (en) * | 1993-12-23 | 1995-07-18 | Andrulis Pharmaceuticals Corp. | Method for treating neurocognitive disorders |
| US5643915A (en) * | 1995-06-06 | 1997-07-01 | Andrulis Pharmaceuticals Corp. | Treatment of ischemia/reperfusion injury with thalidomide alone or in combination with other therapies |
| US5731325A (en) * | 1995-06-06 | 1998-03-24 | Andrulis Pharmaceuticals Corp. | Treatment of melanomas with thalidomide alone or in combination with other anti-melanoma agents |
| US20020006403A1 (en) * | 1999-12-14 | 2002-01-17 | Xue-Zhong Yu | CD28-specific antibody compositions for use in methods of immunosuppression |
| US20040038874A1 (en) * | 2002-08-22 | 2004-02-26 | Osemwota Omoigui | Method of treatment of persistent pain |
| US20040087642A1 (en) * | 2002-10-24 | 2004-05-06 | Zeldis Jerome B. | Methods of using and compositions comprising a JNK inhibitor for the treatment, prevention, management and/or modification of pain |
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2004
- 2004-10-22 WO PCT/US2004/035180 patent/WO2005039497A2/fr active Application Filing
- 2004-10-22 ZA ZA200603402A patent/ZA200603402B/en unknown
- 2004-10-22 BR BRPI0415651-0A patent/BRPI0415651A/pt not_active IP Right Cessation
- 2004-10-22 KR KR1020067009996A patent/KR20060123183A/ko not_active Application Discontinuation
- 2004-10-22 US US10/972,311 patent/US20050119194A1/en not_active Abandoned
- 2004-10-22 EP EP04796214A patent/EP1680132A4/fr not_active Withdrawn
- 2004-10-22 NZ NZ547127A patent/NZ547127A/en unknown
- 2004-10-22 MX MXPA06004382A patent/MXPA06004382A/es not_active Application Discontinuation
- 2004-10-22 AU AU2004283716A patent/AU2004283716A1/en not_active Abandoned
- 2004-10-22 JP JP2006536857A patent/JP2007509170A/ja not_active Withdrawn
- 2004-10-22 CA CA002543312A patent/CA2543312A1/fr not_active Abandoned
- 2004-10-22 CN CNA2004800381703A patent/CN1897956A/zh active Pending
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2006
- 2006-04-23 IL IL175098A patent/IL175098A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2005039497A3 (fr) | 2005-10-20 |
| CN1897956A (zh) | 2007-01-17 |
| NZ547127A (en) | 2008-06-30 |
| IL175098A0 (en) | 2008-04-13 |
| CA2543312A1 (fr) | 2005-05-06 |
| MXPA06004382A (es) | 2006-07-06 |
| EP1680132A2 (fr) | 2006-07-19 |
| EP1680132A4 (fr) | 2009-01-14 |
| BRPI0415651A (pt) | 2006-12-19 |
| JP2007509170A (ja) | 2007-04-12 |
| KR20060123183A (ko) | 2006-12-01 |
| WO2005039497A2 (fr) | 2005-05-06 |
| US20050119194A1 (en) | 2005-06-02 |
| AU2004283716A1 (en) | 2005-05-06 |
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