ZA200509698B - Target-oriented chemotherapy for treating tumors of the sexual organs - Google Patents

Target-oriented chemotherapy for treating tumors of the sexual organs Download PDF

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Publication number
ZA200509698B
ZA200509698B ZA200509698A ZA200509698A ZA200509698B ZA 200509698 B ZA200509698 B ZA 200509698B ZA 200509698 A ZA200509698 A ZA 200509698A ZA 200509698 A ZA200509698 A ZA 200509698A ZA 200509698 B ZA200509698 B ZA 200509698B
Authority
ZA
South Africa
Prior art keywords
estrogens
hydrogen
och
salts
independently
Prior art date
Application number
ZA200509698A
Other languages
English (en)
Inventor
Foerster Heinz
Original Assignee
Trin Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Trin Gmbh filed Critical Trin Gmbh
Publication of ZA200509698B publication Critical patent/ZA200509698B/en

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/50Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom condensed with carbocyclic rings or ring systems
    • C07D333/52Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes
    • C07D333/54Benzo[b]thiophenes; Hydrogenated benzo[b]thiophenes with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
    • C07D333/58Radicals substituted by nitrogen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A61K31/566Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol having an oxo group in position 17, e.g. estrone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26Androgens
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/24Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/28Antiandrogens
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C245/00Compounds containing chains of at least two nitrogen atoms with at least one nitrogen-to-nitrogen multiple bond
    • C07C245/22Compounds containing chains of at least two nitrogen atoms with at least one nitrogen-to-nitrogen multiple bond containing chains of three or more nitrogen atoms with one or more nitrogen-to-nitrogen double bonds
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C245/00Compounds containing chains of at least two nitrogen atoms with at least one nitrogen-to-nitrogen multiple bond
    • C07C245/22Compounds containing chains of at least two nitrogen atoms with at least one nitrogen-to-nitrogen multiple bond containing chains of three or more nitrogen atoms with one or more nitrogen-to-nitrogen double bonds
    • C07C245/24Chains of only three nitrogen atoms, e.g. diazoamines
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J1/00Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00Systems containing at least three condensed rings
    • C07C2603/02Ortho- or ortho- and peri-condensed systems
    • C07C2603/40Ortho- or ortho- and peri-condensed systems containing four condensed rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
ZA200509698A 2003-05-30 2004-05-18 Target-oriented chemotherapy for treating tumors of the sexual organs ZA200509698B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10324496A DE10324496A1 (de) 2003-05-30 2003-05-30 Targetorientierte Chemotherapie von Tumoren der Sexualorgane

Publications (1)

Publication Number Publication Date
ZA200509698B true ZA200509698B (en) 2007-03-28

Family

ID=33441483

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA200509698A ZA200509698B (en) 2003-05-30 2004-05-18 Target-oriented chemotherapy for treating tumors of the sexual organs

Country Status (12)

Country Link
US (1) US20070099876A1 (fr)
EP (1) EP1636249A1 (fr)
JP (1) JP2006526002A (fr)
KR (1) KR20060024784A (fr)
CN (1) CN1835964A (fr)
AU (1) AU2004242908A1 (fr)
CA (1) CA2531319A1 (fr)
DE (1) DE10324496A1 (fr)
IL (1) IL172298A0 (fr)
RU (1) RU2320669C2 (fr)
WO (1) WO2004106358A1 (fr)
ZA (1) ZA200509698B (fr)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1951043A2 (fr) * 2005-11-22 2008-08-06 SmithKline Beecham Corporation Composes chimiques
US8034797B2 (en) * 2007-07-04 2011-10-11 Trin Therapeutics Gmbh Triazene compounds for the treatment of cancer
US8338392B2 (en) * 2008-02-20 2012-12-25 The Wistar Institute MicroRNA modulators and method for identifying and using the same
JP2014515734A (ja) 2011-03-16 2014-07-03 クリエイティブ セラポーティクス ゲーエムベーハー 置換ジフェニル誘導体
WO2012130850A1 (fr) 2011-03-31 2012-10-04 Bayer Pharma Aktiengesellschaft Ciblage de tissu avec des dérivés diphényliques pontés oncocides pour le traitement sélectif de tumeurs des organes sexuels
EP2557075A1 (fr) 2011-08-09 2013-02-13 Trin Therapeutics GmbH Nouveaux alliages de triazène pour le traitement du cancer
EP3592757A2 (fr) * 2017-03-09 2020-01-15 ELITechGroup, Inc. Nitrodiaryléthènes utilisés en tant qu'extincteurs de fluorescence pour des sondes d'acide nucléique

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1016959A (en) * 1963-04-09 1966-01-12 Leo Ab Substituted steroid hormones

Also Published As

Publication number Publication date
AU2004242908A1 (en) 2004-12-09
EP1636249A1 (fr) 2006-03-22
CA2531319A1 (fr) 2004-12-09
DE10324496A1 (de) 2004-12-16
KR20060024784A (ko) 2006-03-17
WO2004106358A1 (fr) 2004-12-09
US20070099876A1 (en) 2007-05-03
JP2006526002A (ja) 2006-11-16
RU2320669C2 (ru) 2008-03-27
CN1835964A (zh) 2006-09-20
RU2005141057A (ru) 2006-06-10
IL172298A0 (en) 2006-04-10

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