ZA200403486B - Directly compressible formulations of azithromycin - Google Patents
Directly compressible formulations of azithromycin Download PDFInfo
- Publication number
- ZA200403486B ZA200403486B ZA200403486A ZA200403486A ZA200403486B ZA 200403486 B ZA200403486 B ZA 200403486B ZA 200403486 A ZA200403486 A ZA 200403486A ZA 200403486 A ZA200403486 A ZA 200403486A ZA 200403486 B ZA200403486 B ZA 200403486B
- Authority
- ZA
- South Africa
- Prior art keywords
- azithromycin
- tablet
- dry blend
- less
- tablets
- Prior art date
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- A61K9/00—Medicinal preparations characterised by special physical form
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Molecular Biology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US34348001P | 2001-12-21 | 2001-12-21 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200403486B true ZA200403486B (en) | 2006-05-31 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200403486A ZA200403486B (en) | 2001-12-21 | 2004-05-07 | Directly compressible formulations of azithromycin |
Country Status (20)
| Country | Link |
|---|---|
| US (4) | US20030165563A1 (zh) |
| EP (1) | EP1455758A1 (zh) |
| JP (1) | JP2005513099A (zh) |
| KR (1) | KR100632339B1 (zh) |
| CN (1) | CN1668282A (zh) |
| AR (1) | AR037930A1 (zh) |
| AU (1) | AU2002348884A1 (zh) |
| BR (1) | BR0215193A (zh) |
| CA (1) | CA2469246A1 (zh) |
| IL (1) | IL161996A0 (zh) |
| MX (1) | MXPA04005105A (zh) |
| NO (1) | NO20043110L (zh) |
| NZ (1) | NZ532707A (zh) |
| PA (1) | PA8562201A1 (zh) |
| PE (1) | PE20030591A1 (zh) |
| PL (1) | PL371259A1 (zh) |
| RU (1) | RU2277914C2 (zh) |
| TW (1) | TW200301138A (zh) |
| WO (1) | WO2003053416A1 (zh) |
| ZA (1) | ZA200403486B (zh) |
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| HRP20020614A2 (en) * | 2002-07-22 | 2004-06-30 | PLIVA-ISTRAŽIVAČKI INSTITUT d.o.o. | Rhombic pseudopolymorph of 9-deoxo-9a-aza-9a-methyl-9a-homoerythromycin a |
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| US20100048498A1 (en) * | 2004-12-21 | 2010-02-25 | Johnson Barbara A | Stable non-dihydrate azithromycin oral suspensions |
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| US20080045548A1 (en) * | 2006-08-21 | 2008-02-21 | Astrazeneca Ab | Pharmaceutical Compositions |
| TWI482772B (zh) * | 2006-08-21 | 2015-05-01 | Astrazeneca Ab | 適合口服且包含三唑并[4,5-d]嘧啶衍生物之組合物 |
| US20100179110A1 (en) * | 2006-12-20 | 2010-07-15 | Mostafa Akbarieh | Composition Containing a Bisphosphonic Acid in Combination with Vitamin D |
| CN101772304B (zh) * | 2007-07-31 | 2014-07-09 | 卡吉尔公司 | 直接可压缩的右旋糖 |
| WO2009059605A1 (en) * | 2007-11-08 | 2009-05-14 | University Of Copenhagen | Small scale solid state screening |
| BRPI0822359A2 (pt) * | 2008-03-18 | 2015-07-14 | Aleksander Vladimirovich Dikovskiy | Composição farmacêutica de antibióticos e prebióticos para prevenir e tratar disbiose durante terapia antibacteriana |
| CN101998859B (zh) * | 2008-03-18 | 2014-03-05 | 亚历山大·弗拉基米罗维奇·季科夫斯基 | 用于预防与抗生素肠道给药相关的生态失调的药物组合物 |
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| AR083417A1 (es) * | 2010-10-14 | 2013-02-21 | Novartis Ag | Composiciones farmaceuticas que contienen un dgat1 inhibidor |
| WO2013088274A1 (en) | 2011-12-14 | 2013-06-20 | Wockhardt Limited | Anhydrous amorphous azithromycin composition free of azithromycin dihydrate |
| KR20150092385A (ko) | 2014-02-03 | 2015-08-13 | 씨제이헬스케어 주식회사 | 솔리페나신을 포함하는 안정한 제제 및 이의 제조방법 |
| US20150242978A1 (en) | 2014-02-24 | 2015-08-27 | Mindojo Ltd. | Content development and moderation flow for e-learning datagraph structures |
| US20160145548A1 (en) * | 2014-11-20 | 2016-05-26 | The Procter & Gamble Company | Cleaning composition refill for an automatic dishwasher dispensing device |
| CN105193753A (zh) * | 2015-10-30 | 2015-12-30 | 成都通德药业有限公司 | 一种阿奇霉素分散片的制备方法 |
| CN110633487B (zh) * | 2019-07-03 | 2023-03-14 | 北京中医药大学 | 直接压片的片剂处方的设计方法 |
| CN111467362B (zh) * | 2020-05-09 | 2021-07-06 | 北京四环制药有限公司 | 一种阿奇霉素药用组合物及其制备方法和其应用 |
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| AU2001214115A1 (en) | 2000-08-01 | 2002-02-13 | Habil F. Khorakiwala | Process for the preparation of anhydrous azithromycin |
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| EA007618B1 (ru) * | 2001-05-22 | 2006-12-29 | Пфайзер Продактс Инк. | Кристаллический полуторогидрат азитромицина, содержащая его фармацевтическая композиция и способ лечения на его основе |
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| CN1668282A (zh) * | 2001-12-21 | 2005-09-14 | 辉瑞产品公司 | 可直接压制的阿齐霉素配方 |
| CN1606433A (zh) * | 2001-12-21 | 2005-04-13 | 辉瑞产品公司 | 阿齐霉素湿法制粒法 |
| WO2003063838A1 (en) * | 2002-02-01 | 2003-08-07 | Pfizer Products Inc. | Dry granulated formulations of azithromycin |
-
2002
- 2002-12-09 CN CNA028257553A patent/CN1668282A/zh active Pending
- 2002-12-09 MX MXPA04005105A patent/MXPA04005105A/es not_active Application Discontinuation
- 2002-12-09 PL PL02371259A patent/PL371259A1/xx not_active Application Discontinuation
- 2002-12-09 EP EP02781616A patent/EP1455758A1/en not_active Ceased
- 2002-12-09 RU RU2004118709/15A patent/RU2277914C2/ru not_active IP Right Cessation
- 2002-12-09 BR BR0215193-6A patent/BR0215193A/pt not_active IP Right Cessation
- 2002-12-09 WO PCT/IB2002/005222 patent/WO2003053416A1/en not_active Application Discontinuation
- 2002-12-09 IL IL16199602A patent/IL161996A0/xx unknown
- 2002-12-09 AU AU2002348884A patent/AU2002348884A1/en not_active Abandoned
- 2002-12-09 JP JP2003554175A patent/JP2005513099A/ja not_active Withdrawn
- 2002-12-09 CA CA002469246A patent/CA2469246A1/en not_active Abandoned
- 2002-12-09 KR KR1020047009446A patent/KR100632339B1/ko not_active IP Right Cessation
- 2002-12-09 NZ NZ532707A patent/NZ532707A/en unknown
- 2002-12-13 PE PE2002001219A patent/PE20030591A1/es not_active Application Discontinuation
- 2002-12-19 AR ARP020105016A patent/AR037930A1/es unknown
- 2002-12-20 US US10/327,459 patent/US20030165563A1/en not_active Abandoned
- 2002-12-20 TW TW091136916A patent/TW200301138A/zh unknown
- 2002-12-20 PA PA20028562201A patent/PA8562201A1/es unknown
-
2004
- 2004-05-07 ZA ZA200403486A patent/ZA200403486B/en unknown
- 2004-07-20 NO NO20043110A patent/NO20043110L/no not_active Application Discontinuation
-
2005
- 2005-07-26 US US11/190,393 patent/US7070811B2/en not_active Expired - Fee Related
- 2005-08-26 US US11/213,022 patent/US20060024364A1/en not_active Abandoned
- 2005-08-26 US US11/212,332 patent/US20060024363A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| KR20040066175A (ko) | 2004-07-23 |
| CN1668282A (zh) | 2005-09-14 |
| NZ532707A (en) | 2006-07-28 |
| MXPA04005105A (es) | 2004-08-19 |
| US20060024363A1 (en) | 2006-02-02 |
| AU2002348884A1 (en) | 2003-07-09 |
| BR0215193A (pt) | 2004-11-16 |
| RU2004118709A (ru) | 2005-04-20 |
| TW200301138A (en) | 2003-07-01 |
| PE20030591A1 (es) | 2003-07-12 |
| US20050287209A1 (en) | 2005-12-29 |
| RU2277914C2 (ru) | 2006-06-20 |
| US20030165563A1 (en) | 2003-09-04 |
| AR037930A1 (es) | 2004-12-22 |
| KR100632339B1 (ko) | 2006-10-12 |
| EP1455758A1 (en) | 2004-09-15 |
| PA8562201A1 (es) | 2003-07-28 |
| CA2469246A1 (en) | 2003-07-03 |
| NO20043110L (no) | 2004-07-20 |
| IL161996A0 (en) | 2005-11-20 |
| PL371259A1 (en) | 2005-06-13 |
| WO2003053416A1 (en) | 2003-07-03 |
| JP2005513099A (ja) | 2005-05-12 |
| US7070811B2 (en) | 2006-07-04 |
| US20060024364A1 (en) | 2006-02-02 |
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