ZA200402621B - Intermediates for preparing glycogen phosphorylase inhibitors. - Google Patents
Intermediates for preparing glycogen phosphorylase inhibitors. Download PDFInfo
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- ZA200402621B ZA200402621B ZA200402621A ZA200402621A ZA200402621B ZA 200402621 B ZA200402621 B ZA 200402621B ZA 200402621 A ZA200402621 A ZA 200402621A ZA 200402621 A ZA200402621 A ZA 200402621A ZA 200402621 B ZA200402621 B ZA 200402621B
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- South Africa
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- compound
- acid
- mixture
- reaction
- solution
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- 108010046163 Glycogen Phosphorylase Proteins 0.000 title description 10
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Indole Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US34964702P | 2002-01-18 | 2002-01-18 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200402621B true ZA200402621B (en) | 2005-05-27 |
Family
ID=23373348
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ZA200402621A ZA200402621B (en) | 2002-01-18 | 2004-04-02 | Intermediates for preparing glycogen phosphorylase inhibitors. |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US6696574B2 (xx) |
| EP (1) | EP1470128A1 (xx) |
| JP (1) | JP2005514460A (xx) |
| KR (1) | KR20040072730A (xx) |
| CN (1) | CN1592749A (xx) |
| AU (1) | AU2003200853A1 (xx) |
| BR (1) | BR0307006A (xx) |
| CA (1) | CA2472205A1 (xx) |
| HU (1) | HUP0500513A3 (xx) |
| IL (1) | IL161507A0 (xx) |
| MX (1) | MXPA04006937A (xx) |
| PL (1) | PL371408A1 (xx) |
| RU (1) | RU2004121986A (xx) |
| TW (1) | TW200302220A (xx) |
| WO (1) | WO2003059910A1 (xx) |
| ZA (1) | ZA200402621B (xx) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2006059163A1 (en) * | 2004-12-02 | 2006-06-08 | Prosidion Limited | Treatment of diabetes with glycogen phosphorylase inhibitors |
| PE20080251A1 (es) | 2006-05-04 | 2008-04-25 | Boehringer Ingelheim Int | Usos de inhibidores de dpp iv |
| ES2699773T3 (es) * | 2011-05-31 | 2019-02-12 | Theravance Biopharma R&D Ip Llc | Inhibidores de neprilisina |
| CN103626845B (zh) * | 2013-09-30 | 2015-11-11 | 承德医学院 | 作为糖原磷酸化酶抑制剂的芳基并吡咯-2-甲酰胺二肽衍生物、其制备方法及医药用途 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX9709874A (es) * | 1995-06-06 | 1998-03-31 | Pfizer | N-(INDOL-2-CARBONIL) beta-ALANILAMIDAS SUSTITUIDAS Y DERIVADOS COMO INHIBIDORES DE GLUCOGENO FOSFORILASA, USO DE LOS MISMOS Y COMPOSICIONES QUE LOS CONTIENEN. |
| DE69523182T2 (de) | 1995-06-06 | 2002-02-07 | Pfizer | Substituierte n-(indol-2-carbonyl)-glycinamide und derivate als glycogen phosphorylase inhibitoren |
| US6277877B1 (en) | 2000-08-15 | 2001-08-21 | Pfizer, Inc. | Substituted n-(indole-2-carbonyl)glycinamides and derivates as glycogen phosphorylase inhibitors |
-
2003
- 2003-01-06 CA CA002472205A patent/CA2472205A1/en not_active Abandoned
- 2003-01-06 CN CNA038015455A patent/CN1592749A/zh active Pending
- 2003-01-06 BR BR0307006-9A patent/BR0307006A/pt not_active Application Discontinuation
- 2003-01-06 WO PCT/IB2003/000034 patent/WO2003059910A1/en not_active Application Discontinuation
- 2003-01-06 KR KR10-2004-7011084A patent/KR20040072730A/ko not_active Application Discontinuation
- 2003-01-06 AU AU2003200853A patent/AU2003200853A1/en not_active Abandoned
- 2003-01-06 PL PL03371408A patent/PL371408A1/xx not_active Application Discontinuation
- 2003-01-06 HU HU0500513A patent/HUP0500513A3/hu unknown
- 2003-01-06 JP JP2003560013A patent/JP2005514460A/ja active Pending
- 2003-01-06 MX MXPA04006937A patent/MXPA04006937A/es unknown
- 2003-01-06 EP EP03700024A patent/EP1470128A1/en not_active Withdrawn
- 2003-01-06 RU RU2004121986/04A patent/RU2004121986A/ru not_active Application Discontinuation
- 2003-01-06 IL IL16150703A patent/IL161507A0/xx unknown
- 2003-01-13 TW TW092100616A patent/TW200302220A/zh unknown
- 2003-01-16 US US10/345,661 patent/US6696574B2/en not_active Expired - Fee Related
-
2004
- 2004-04-02 ZA ZA200402621A patent/ZA200402621B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL161507A0 (en) | 2004-09-27 |
| US20030187051A1 (en) | 2003-10-02 |
| KR20040072730A (ko) | 2004-08-18 |
| EP1470128A1 (en) | 2004-10-27 |
| US6696574B2 (en) | 2004-02-24 |
| WO2003059910A1 (en) | 2003-07-24 |
| MXPA04006937A (es) | 2004-12-06 |
| BR0307006A (pt) | 2004-11-03 |
| CA2472205A1 (en) | 2003-07-24 |
| HUP0500513A3 (en) | 2006-07-28 |
| TW200302220A (en) | 2003-08-01 |
| RU2004121986A (ru) | 2005-11-20 |
| PL371408A1 (en) | 2005-06-13 |
| HUP0500513A2 (hu) | 2005-11-28 |
| CN1592749A (zh) | 2005-03-09 |
| AU2003200853A1 (en) | 2003-07-30 |
| JP2005514460A (ja) | 2005-05-19 |
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