ZA200300588B - Use of dopamine D2/D3 receptor agonists to treat fibromyalgia. - Google Patents
Use of dopamine D2/D3 receptor agonists to treat fibromyalgia. Download PDFInfo
- Publication number
- ZA200300588B ZA200300588B ZA200300588A ZA200300588A ZA200300588B ZA 200300588 B ZA200300588 B ZA 200300588B ZA 200300588 A ZA200300588 A ZA 200300588A ZA 200300588 A ZA200300588 A ZA 200300588A ZA 200300588 B ZA200300588 B ZA 200300588B
- Authority
- ZA
- South Africa
- Prior art keywords
- group
- fibromyalgia
- phenyl
- alkyl group
- dopamine
- Prior art date
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/428—Thiazoles condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Neurology (AREA)
- Physical Education & Sports Medicine (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US09/617,177 US6277875B1 (en) | 2000-07-17 | 2000-07-17 | Use of dopamine D2/D3 receptor agonists to treat fibromyalgia |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ZA200300588B true ZA200300588B (en) | 2004-04-22 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| ZA200300588A ZA200300588B (en) | 2000-07-17 | 2003-01-22 | Use of dopamine D2/D3 receptor agonists to treat fibromyalgia. |
Country Status (17)
| Country | Link |
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| US (2) | US6277875B1 (no) |
| EP (1) | EP1311251A2 (no) |
| JP (1) | JP2004503587A (no) |
| KR (1) | KR100797603B1 (no) |
| CN (1) | CN1443066A (no) |
| AU (2) | AU2001271910B2 (no) |
| BR (1) | BR0112476A (no) |
| CA (1) | CA2414774C (no) |
| CZ (1) | CZ2003417A3 (no) |
| HU (1) | HUP0301305A3 (no) |
| IL (1) | IL153915A0 (no) |
| MX (1) | MXPA03000336A (no) |
| NO (1) | NO20030213L (no) |
| NZ (1) | NZ523926A (no) |
| PL (1) | PL360121A1 (no) |
| WO (1) | WO2002005797A2 (no) |
| ZA (1) | ZA200300588B (no) |
Families Citing this family (32)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| BR0110188A (pt) * | 2000-04-21 | 2003-03-05 | Upjohn Co | Compostos selecionados para o tratamento de sìndromes de fibromialgia e de fadiga crÈnica |
| DE10041479A1 (de) * | 2000-08-24 | 2002-03-14 | Sanol Arznei Schwarz Gmbh | Neue pharmazeutische Zusammensetzung zur Verabreichung von N-0923 |
| US20020165246A1 (en) * | 2001-03-05 | 2002-11-07 | Andrew Holman | Administration of sleep restorative agents |
| DE10137162A1 (de) * | 2001-07-30 | 2003-02-20 | Hexal Ag | Matrixkontrolliertes transdermales therapeutisches System zur Anwendung von Pramiprexol und Ropinirol |
| DE10138275A1 (de) * | 2001-08-10 | 2003-02-27 | Boehringer Ingelheim Pharma | Verbindungen zur Beseitigung der Anhedonie |
| GB0125088D0 (en) * | 2001-10-18 | 2001-12-12 | Smithkline Beecham Cork Ltd | New use |
| US7079888B2 (en) * | 2002-04-11 | 2006-07-18 | Ansar, Inc. | Method and apparatus for monitoring the autonomic nervous system using non-stationary spectral analysis of heart rate and respiratory activity |
| US20040048779A1 (en) * | 2002-05-06 | 2004-03-11 | Erwin Schollmayer | Use of rotigotine for treating the restless leg syndrome |
| AR040680A1 (es) * | 2002-07-25 | 2005-04-13 | Pharmacia Corp | Composicion de tabletas de liberacion sostenida |
| MY142204A (en) * | 2002-07-25 | 2010-10-29 | Pharmacia Corp | Pramipexole once-daily dosage form |
| US20050226926A1 (en) * | 2002-07-25 | 2005-10-13 | Pfizer Inc | Sustained-release tablet composition of pramipexole |
| US20040092504A1 (en) * | 2002-11-12 | 2004-05-13 | Anuthep Benja-Athon | Definitive medications for treating fibromyalgia |
| ES2239196T3 (es) * | 2002-12-02 | 2005-09-16 | Schwarz Pharma Ag | Suministro iontoforetico de rotigotina para el tratamiento de la enfermedad de parkinson. |
| DE10334188B4 (de) * | 2003-07-26 | 2007-07-05 | Schwarz Pharma Ag | Verwendung von Rotigotin zur Behandlung von Depressionen |
| DE10334187A1 (de) * | 2003-07-26 | 2005-03-03 | Schwarz Pharma Ag | Substituierte 2-Aminotetraline zur Behandlung von Depressionen |
| SI1781260T2 (sl) * | 2004-08-13 | 2014-08-29 | Boehringer Ingelheim International Gmbh | Tabletna formulacija s podaljšanim sproščanjem, ki vsebuje pramipeksol ali njegovo farmacevtsko sprejemljivo sol, postopek za izdelavo le-te in njena uporaba |
| CN101843597A (zh) * | 2004-08-13 | 2010-09-29 | 贝林格尔·英格海姆国际有限公司 | 包含普拉克索或其可药用盐的延长释放小球制剂、其制备方法及其用途 |
| WO2007048034A2 (en) * | 2005-10-21 | 2007-04-26 | Caritas St. Elizabeth Medical Center Of Boston, Inc. | Use of androgens for the treatment of parkinson' s disease |
| WO2007090883A1 (en) * | 2006-02-10 | 2007-08-16 | Boehringer Ingelheim International Gmbh | Extended release formulation |
| WO2007090881A2 (en) * | 2006-02-10 | 2007-08-16 | Boehringer Ingelheim International Gmbh | Modified release formulation |
| TWI392670B (zh) * | 2006-06-22 | 2013-04-11 | Ucb Pharma Gmbh | 經取代的２-胺基萘滿之於製造用於預防、減緩及／或治療各種類型疼痛之藥物上的用途 |
| CN1944647B (zh) * | 2006-08-23 | 2010-05-12 | 华东师范大学 | 多巴胺受体新亚型d5b基因及编码的蛋白与应用 |
| GB0700786D0 (en) * | 2007-01-15 | 2007-02-21 | Pfizer Ltd | Morpholine dopamine agonists for the treatment of pain |
| EP1987815A1 (en) * | 2007-05-04 | 2008-11-05 | Schwarz Pharma Ag | Oronasopharyngeally deliverable pharmaceutical compositions of dopamine agonists for the prevention and/or treatment of restless limb disorders |
| US20110195117A1 (en) * | 2008-09-01 | 2011-08-11 | Lupin Limited | Controlled release compositions of ropinirole |
| US20110262537A1 (en) | 2008-09-29 | 2011-10-27 | Premchand Nakhat | Extended release dosage form of ropinirole |
| WO2010044108A2 (en) | 2008-10-17 | 2010-04-22 | Rubicon Research Private Limited | Controlled release formulations of ropinirole |
| AU2011248904B2 (en) | 2010-04-30 | 2014-02-27 | Teikoku Seiyaku Co., Ltd. | Propynylaminoindan transdermal compositions |
| WO2012129429A2 (en) | 2011-03-24 | 2012-09-27 | Teikoku Pharma Usa, Inc. | Transdermal compositions comprising an active agent layer and an active agent conversion layer |
| JP5913614B2 (ja) | 2011-11-09 | 2016-04-27 | テイコク ファーマ ユーエスエー インコーポレーテッド | 皮膚新生物の処置方法 |
| AU2013338243B2 (en) | 2012-11-02 | 2016-09-29 | Teikoku Seiyaku Co., Ltd. | Propynylaminoindan transdermal compositions |
| MA41125A (fr) * | 2014-12-05 | 2017-10-10 | Purdue Pharma Lp | Dérivés de 6.7-cyclomorphinane et leur utilisation |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4414224A (en) * | 1980-08-22 | 1983-11-08 | Smithkline Beckman Corporation | Pharmaceutical composition and methods for producing dopamine agonist activity |
| US4879391A (en) * | 1982-09-20 | 1989-11-07 | Pfizer Inc. | 1-Phenyl-2(1H,3H)-indolone psychotherapeutic agents |
| US4452808A (en) * | 1982-12-07 | 1984-06-05 | Smithkline Beckman Corporation | 4-Aminoalkyl-2(3H)-indolones |
| DE3447075A1 (de) * | 1984-12-22 | 1986-07-03 | Dr. Karl Thomae Gmbh, 7950 Biberach | Tetrahydro-benzthiazole, deren herstellung und deren verwendung als zwischenprodukte oder als arzneimittel |
| ATE45735T1 (de) * | 1984-12-22 | 1989-09-15 | Thomae Gmbh Dr K | Tetrahydro-benzthiazole, deren herstellung und deren verwendung als zwischenprodukte oder als arnzneimittel. |
| GB8712073D0 (en) * | 1987-05-21 | 1987-06-24 | Smith Kline French Lab | Medicament |
| US5498610A (en) * | 1992-11-06 | 1996-03-12 | Pfizer Inc. | Neuroprotective indolone and related derivatives |
| US5696128A (en) | 1994-07-07 | 1997-12-09 | The Board Of Supervisors Of Louisiana University And Agricultural And Mechanical College | Method of regulating immune function |
| US5658955A (en) | 1994-11-01 | 1997-08-19 | Hitzig; Pietr | Combined use of dopamine and serotonin agonists in the treatment of immune disorders |
| BR0110188A (pt) * | 2000-04-21 | 2003-03-05 | Upjohn Co | Compostos selecionados para o tratamento de sìndromes de fibromialgia e de fadiga crÈnica |
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2000
- 2000-07-17 US US09/617,177 patent/US6277875B1/en not_active Expired - Lifetime
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2001
- 2001-05-07 US US09/850,901 patent/US6300365B1/en not_active Expired - Fee Related
- 2001-07-05 JP JP2002511730A patent/JP2004503587A/ja active Pending
- 2001-07-05 IL IL15391501A patent/IL153915A0/xx unknown
- 2001-07-05 AU AU2001271910A patent/AU2001271910B2/en not_active Ceased
- 2001-07-05 CZ CZ2003417A patent/CZ2003417A3/cs unknown
- 2001-07-05 NZ NZ523926A patent/NZ523926A/en unknown
- 2001-07-05 CN CN01812983A patent/CN1443066A/zh active Pending
- 2001-07-05 HU HU0301305A patent/HUP0301305A3/hu unknown
- 2001-07-05 KR KR1020037000785A patent/KR100797603B1/ko not_active IP Right Cessation
- 2001-07-05 BR BR0112476-5A patent/BR0112476A/pt not_active IP Right Cessation
- 2001-07-05 CA CA2414774A patent/CA2414774C/en not_active Expired - Fee Related
- 2001-07-05 PL PL36012101A patent/PL360121A1/xx unknown
- 2001-07-05 WO PCT/US2001/021530 patent/WO2002005797A2/en active IP Right Grant
- 2001-07-05 AU AU7191001A patent/AU7191001A/xx active Pending
- 2001-07-05 MX MXPA03000336A patent/MXPA03000336A/es active IP Right Grant
- 2001-07-05 EP EP01950966A patent/EP1311251A2/en not_active Withdrawn
-
2003
- 2003-01-16 NO NO20030213A patent/NO20030213L/no not_active Application Discontinuation
- 2003-01-22 ZA ZA200300588A patent/ZA200300588B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2414774A1 (en) | 2002-01-24 |
| BR0112476A (pt) | 2003-07-22 |
| CA2414774C (en) | 2010-09-07 |
| MXPA03000336A (es) | 2005-04-19 |
| AU2001271910B2 (en) | 2005-07-28 |
| US6277875B1 (en) | 2001-08-21 |
| HUP0301305A3 (en) | 2008-03-28 |
| WO2002005797A2 (en) | 2002-01-24 |
| KR100797603B1 (ko) | 2008-01-28 |
| WO2002005797A8 (en) | 2003-03-06 |
| KR20030029625A (ko) | 2003-04-14 |
| NO20030213L (no) | 2003-03-11 |
| EP1311251A2 (en) | 2003-05-21 |
| AU7191001A (en) | 2002-01-30 |
| PL360121A1 (en) | 2004-09-06 |
| JP2004503587A (ja) | 2004-02-05 |
| IL153915A0 (en) | 2003-07-31 |
| CN1443066A (zh) | 2003-09-17 |
| US6300365B1 (en) | 2001-10-09 |
| CZ2003417A3 (cs) | 2003-08-13 |
| NO20030213D0 (no) | 2003-01-16 |
| HUP0301305A2 (hu) | 2003-08-28 |
| NZ523926A (en) | 2006-05-26 |
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