ZA200109785B - TH2 differentiation inhibitors. - Google Patents
TH2 differentiation inhibitors. Download PDFInfo
- Publication number
- ZA200109785B ZA200109785B ZA200109785A ZA200109785A ZA200109785B ZA 200109785 B ZA200109785 B ZA 200109785B ZA 200109785 A ZA200109785 A ZA 200109785A ZA 200109785 A ZA200109785 A ZA 200109785A ZA 200109785 B ZA200109785 B ZA 200109785B
- Authority
- ZA
- South Africa
- Prior art keywords
- optionally substituted
- ring
- compound
- lower alkyl
- substituted lower
- Prior art date
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Classifications
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- C07C251/32—Oximes
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C211/00—Compounds containing amino groups bound to a carbon skeleton
- C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
- C07C211/44—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring
- C07C211/49—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring having at least two amino groups bound to the carbon skeleton
- C07C211/50—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring having at least two amino groups bound to the carbon skeleton with at least two amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
- C07C217/78—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
- C07C217/80—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings
Landscapes
- Health & Medical Sciences (AREA)
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- Medicinal Chemistry (AREA)
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- Immunology (AREA)
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- Pulmonology (AREA)
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- Neurology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Endocrinology (AREA)
- Transplantation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
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Publications (1)
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| EP (1) | EP1206935A4 (tr) |
| KR (1) | KR20020012309A (tr) |
| CN (1) | CN1364080A (tr) |
| AU (1) | AU763976B2 (tr) |
| BR (1) | BR0012697A (tr) |
| CA (1) | CA2375982A1 (tr) |
| HK (1) | HK1046645A1 (tr) |
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| PL (1) | PL353476A1 (tr) |
| RU (1) | RU2230551C2 (tr) |
| TR (1) | TR200200099T2 (tr) |
| WO (1) | WO2001007032A1 (tr) |
| ZA (1) | ZA200109785B (tr) |
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| WO2001005768A1 (fr) * | 1999-07-19 | 2001-01-25 | Shionogi & Co., Ltd. | Composes tricycliques porteurs de pendants acyloxymethoxycarbonyle |
| WO2002057216A1 (fr) * | 2001-01-18 | 2002-07-25 | Shionogi & Co., Ltd. | Composes de terphenyle supportant des groupes amino substitues |
| JPWO2002057237A1 (ja) * | 2001-01-22 | 2004-05-20 | 塩野義製薬株式会社 | 置換アミノ基を有するヘテロ３環化合物 |
| US7186855B2 (en) | 2001-06-11 | 2007-03-06 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
| US8048917B2 (en) | 2005-04-06 | 2011-11-01 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
| US6818787B2 (en) | 2001-06-11 | 2004-11-16 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
| WO2003030905A1 (fr) * | 2001-10-01 | 2003-04-17 | Shionogi & Co., Ltd. | Inhibiteur de la dihydroorotate deshydrogenase |
| WO2003099284A1 (en) | 2002-05-22 | 2003-12-04 | Amgen Inc. | Amino-pyridine, -pyridine and pyridazine derivatives for use as vanilloid receptor ligands for the treatment of pain |
| NZ537952A (en) | 2002-08-08 | 2008-04-30 | Amgen Inc | Vanilloid receptor ligands and their use in treatments |
| US20050282814A1 (en) * | 2002-10-03 | 2005-12-22 | Targegen, Inc. | Vasculostatic agents and methods of use thereof |
| JP2007522233A (ja) | 2004-02-11 | 2007-08-09 | アムジエン・インコーポレーテツド | バニロイド受容体リガンド及び治療におけるそれらの使用 |
| MY139645A (en) | 2004-02-11 | 2009-10-30 | Amgen Inc | Vanilloid receptor ligands and their use in treatments |
| NZ588139A (en) | 2004-04-08 | 2012-02-24 | Targegen Inc | 7-Aryl-3-arylamino-benzo[1,2,4]triazine derivatives |
| MX2007002208A (es) | 2004-08-25 | 2007-05-08 | Targegen Inc | Compuestos hetrociclicos y metodos de uso. |
| AP2007004047A0 (en) | 2005-01-20 | 2007-06-30 | Pfizer Ltd | Substituted triazole derivatives as oxtocin antagonists |
| WO2006089311A1 (en) | 2005-02-15 | 2006-08-24 | Amgen Inc. | Vanilloid receptor ligands and their use in treatments |
| JP2006298775A (ja) * | 2005-04-15 | 2006-11-02 | Dainippon Sumitomo Pharma Co Ltd | 選択的Ｔｈ２免疫反応抑制剤 |
| PT1951684T (pt) | 2005-11-01 | 2016-10-13 | Targegen Inc | Inibidores de cinases de tipo biaril-meta-pirimidina |
| US8133900B2 (en) | 2005-11-01 | 2012-03-13 | Targegen, Inc. | Use of bi-aryl meta-pyrimidine inhibitors of kinases |
| US8604042B2 (en) | 2005-11-01 | 2013-12-10 | Targegen, Inc. | Bi-aryl meta-pyrimidine inhibitors of kinases |
| WO2009031627A1 (ja) * | 2007-09-04 | 2009-03-12 | Riken | パラテルフェニル化合物、その薬理学的に許容される塩、その製造方法及び用途 |
| UA103319C2 (en) | 2008-05-06 | 2013-10-10 | Глаксосмитклайн Ллк | Thiazole- and oxazole-benzene sulfonamide compounds |
| DK2509961T3 (en) | 2009-12-11 | 2016-05-17 | Autifony Therapeutics Ltd | Imidazolidinedione derivatives |
| EP2560488B1 (en) | 2010-04-23 | 2015-10-28 | Cytokinetics, Inc. | Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use |
| AR081626A1 (es) | 2010-04-23 | 2012-10-10 | Cytokinetics Inc | Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos |
| AR081331A1 (es) | 2010-04-23 | 2012-08-08 | Cytokinetics Inc | Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos |
| WO2012060847A1 (en) | 2010-11-07 | 2012-05-10 | Targegen, Inc. | Compositions and methods for treating myelofibrosis |
| EP2649066B1 (en) | 2010-12-06 | 2015-10-21 | Autifony Therapeutics Limited | Hydantoin derivatives useful as kv3 inhibitors |
| JP6008953B2 (ja) | 2011-06-07 | 2016-10-19 | アウトイフオンイ トヘラペウトイクス リミテッド | Ｋｖ３阻害剤としてのヒダントイン誘導体 |
| CN104334548A (zh) | 2012-05-22 | 2015-02-04 | 奥蒂福尼疗法有限公司 | 作为kv3抑制剂的乙内酰脲衍生物 |
| US9422252B2 (en) | 2012-05-22 | 2016-08-23 | Autifony Therapeutics Limited | Triazoles as Kv3 inhibitors |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5693611A (en) * | 1996-02-01 | 1997-12-02 | Eli Lilly And Company | Cyclic peptide antifungal agents |
| PT895981E (pt) | 1996-04-22 | 2001-05-31 | Shionogi & Co | Compostos de terfenilo e medicamentos contendo os mesmos |
| US7101915B1 (en) | 1996-07-31 | 2006-09-05 | Shionogi & Co., Ltd. | P-terphenyl compounds |
| HN1997000027A (es) * | 1996-12-06 | 1997-06-05 | Pfizer Prod Inc | Derivados de 6-fenil piridil - 2 amina |
| WO1998056785A1 (fr) * | 1997-06-12 | 1998-12-17 | Sumitomo Pharmaceuticals Co., Ltd. | Derives de pyrazole |
| US6003360A (en) | 1997-07-01 | 1999-12-21 | Wilson Tool International, Inc. | Press brake tool holder |
| WO1999038829A1 (fr) * | 1998-01-28 | 1999-08-05 | Shionogi & Co., Ltd. | Nouveau compose tricyclique |
| WO2001005768A1 (fr) * | 1999-07-19 | 2001-01-25 | Shionogi & Co., Ltd. | Composes tricycliques porteurs de pendants acyloxymethoxycarbonyle |
-
2000
- 2000-07-14 TR TR2002/00099T patent/TR200200099T2/tr unknown
- 2000-07-14 PL PL00353476A patent/PL353476A1/xx not_active Application Discontinuation
- 2000-07-14 MX MXPA01013452A patent/MXPA01013452A/es unknown
- 2000-07-14 RU RU2002103201/15A patent/RU2230551C2/ru not_active IP Right Cessation
- 2000-07-14 CN CN00810786A patent/CN1364080A/zh active Pending
- 2000-07-14 BR BR0012697-7A patent/BR0012697A/pt not_active IP Right Cessation
- 2000-07-14 US US09/980,475 patent/US7008954B1/en not_active Expired - Fee Related
- 2000-07-14 AU AU60159/00A patent/AU763976B2/en not_active Ceased
- 2000-07-14 CA CA002375982A patent/CA2375982A1/en not_active Abandoned
- 2000-07-14 KR KR1020027000498A patent/KR20020012309A/ko not_active Application Discontinuation
- 2000-07-14 EP EP00946316A patent/EP1206935A4/en not_active Withdrawn
- 2000-07-14 HU HU0203575A patent/HUP0203575A3/hu unknown
- 2000-07-14 WO PCT/JP2000/004725 patent/WO2001007032A1/ja not_active Application Discontinuation
-
2001
- 2001-11-28 ZA ZA200109785A patent/ZA200109785B/en unknown
- 2001-12-21 NO NO20016401A patent/NO20016401L/no not_active Application Discontinuation
-
2002
- 2002-11-18 HK HK02108343.5A patent/HK1046645A1/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BR0012697A (pt) | 2002-04-09 |
| AU6015900A (en) | 2001-02-13 |
| HUP0203575A3 (en) | 2003-11-28 |
| NO20016401L (no) | 2002-01-23 |
| PL353476A1 (en) | 2003-11-17 |
| TR200200099T2 (tr) | 2002-06-21 |
| US7008954B1 (en) | 2006-03-07 |
| WO2001007032A1 (fr) | 2001-02-01 |
| CA2375982A1 (en) | 2001-02-01 |
| HK1046645A1 (zh) | 2003-01-24 |
| MXPA01013452A (es) | 2002-07-02 |
| EP1206935A4 (en) | 2008-07-30 |
| RU2230551C2 (ru) | 2004-06-20 |
| HUP0203575A2 (hu) | 2003-02-28 |
| AU763976B2 (en) | 2003-08-07 |
| EP1206935A1 (en) | 2002-05-22 |
| CN1364080A (zh) | 2002-08-14 |
| KR20020012309A (ko) | 2002-02-15 |
| NO20016401D0 (no) | 2001-12-21 |
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