ZA200109785B - TH2 differentiation inhibitors. - Google Patents
TH2 differentiation inhibitors. Download PDFInfo
- Publication number
- ZA200109785B ZA200109785B ZA200109785A ZA200109785A ZA200109785B ZA 200109785 B ZA200109785 B ZA 200109785B ZA 200109785 A ZA200109785 A ZA 200109785A ZA 200109785 A ZA200109785 A ZA 200109785A ZA 200109785 B ZA200109785 B ZA 200109785B
- Authority
- ZA
- South Africa
- Prior art keywords
- optionally substituted
- ring
- compound
- lower alkyl
- substituted lower
- Prior art date
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Classifications
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- C07C251/32—Oximes
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C211/00—Compounds containing amino groups bound to a carbon skeleton
- C07C211/43—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
- C07C211/44—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring
- C07C211/49—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring having at least two amino groups bound to the carbon skeleton
- C07C211/50—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton having amino groups bound to only one six-membered aromatic ring having at least two amino groups bound to the carbon skeleton with at least two amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C217/00—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton
- C07C217/78—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton
- C07C217/80—Compounds containing amino and etherified hydroxy groups bound to the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of six-membered aromatic rings of the same carbon skeleton having amino groups and etherified hydroxy groups bound to carbon atoms of non-condensed six-membered aromatic rings
Landscapes
- Health & Medical Sciences (AREA)
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- General Health & Medical Sciences (AREA)
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- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
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- Bioinformatics & Cheminformatics (AREA)
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- Chemical Kinetics & Catalysis (AREA)
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- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Immunology (AREA)
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- Pulmonology (AREA)
- Reproductive Health (AREA)
- Neurology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Endocrinology (AREA)
- Transplantation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
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| JP20929899 | 1999-07-23 |
Publications (1)
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| ZA200109785B true ZA200109785B (en) | 2002-11-28 |
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| ZA200109785A ZA200109785B (en) | 1999-07-23 | 2001-11-28 | TH2 differentiation inhibitors. |
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| US (1) | US7008954B1 (no) |
| EP (1) | EP1206935A4 (no) |
| KR (1) | KR20020012309A (no) |
| CN (1) | CN1364080A (no) |
| AU (1) | AU763976B2 (no) |
| BR (1) | BR0012697A (no) |
| CA (1) | CA2375982A1 (no) |
| HK (1) | HK1046645A1 (no) |
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| MX (1) | MXPA01013452A (no) |
| NO (1) | NO20016401L (no) |
| PL (1) | PL353476A1 (no) |
| RU (1) | RU2230551C2 (no) |
| TR (1) | TR200200099T2 (no) |
| WO (1) | WO2001007032A1 (no) |
| ZA (1) | ZA200109785B (no) |
Families Citing this family (31)
| Publication number | Priority date | Publication date | Assignee | Title |
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| CA2375909A1 (en) * | 1999-07-19 | 2001-01-25 | Shionogi & Co., Ltd. | Tricyclic compounds bearing acyloxymethoxycarbonyl pendants |
| WO2002057216A1 (fr) * | 2001-01-18 | 2002-07-25 | Shionogi & Co., Ltd. | Composes de terphenyle supportant des groupes amino substitues |
| US20040087604A1 (en) * | 2001-01-22 | 2004-05-06 | Tatsuo Tsuri | Hetero-tricyclic compounds having substituted amino groups |
| US6818787B2 (en) | 2001-06-11 | 2004-11-16 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
| US8048917B2 (en) | 2005-04-06 | 2011-11-01 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
| US7186855B2 (en) | 2001-06-11 | 2007-03-06 | Xenoport, Inc. | Prodrugs of GABA analogs, compositions and uses thereof |
| WO2003030905A1 (fr) * | 2001-10-01 | 2003-04-17 | Shionogi & Co., Ltd. | Inhibiteur de la dihydroorotate deshydrogenase |
| ES2355472T3 (es) | 2002-05-22 | 2011-03-28 | Amgen Inc. | Derivados de aminopirimidina para su uso como ligandos del receptor vaniloide para el tratamiento del dolor. |
| TW200410945A (en) | 2002-08-08 | 2004-07-01 | Amgen Inc | Vanilloid receptor ligands and their use in treatments" |
| US20050282814A1 (en) * | 2002-10-03 | 2005-12-22 | Targegen, Inc. | Vasculostatic agents and methods of use thereof |
| MY139645A (en) | 2004-02-11 | 2009-10-30 | Amgen Inc | Vanilloid receptor ligands and their use in treatments |
| EP1745034A1 (en) | 2004-02-11 | 2007-01-24 | Amgen Inc. | Vanilloid receptor ligands and their use in treatments |
| US7456176B2 (en) | 2004-04-08 | 2008-11-25 | Targegen, Inc. | Benzotriazine inhibitors of kinases |
| MX2007002208A (es) | 2004-08-25 | 2007-05-08 | Targegen Inc | Compuestos hetrociclicos y metodos de uso. |
| AP2007004047A0 (en) | 2005-01-20 | 2007-06-30 | Pfizer Ltd | Substituted triazole derivatives as oxtocin antagonists |
| WO2006089311A1 (en) | 2005-02-15 | 2006-08-24 | Amgen Inc. | Vanilloid receptor ligands and their use in treatments |
| JP2006298775A (ja) * | 2005-04-15 | 2006-11-02 | Dainippon Sumitomo Pharma Co Ltd | 選択的Ｔｈ２免疫反応抑制剤 |
| US8133900B2 (en) | 2005-11-01 | 2012-03-13 | Targegen, Inc. | Use of bi-aryl meta-pyrimidine inhibitors of kinases |
| US7528143B2 (en) | 2005-11-01 | 2009-05-05 | Targegen, Inc. | Bi-aryl meta-pyrimidine inhibitors of kinases |
| US8604042B2 (en) | 2005-11-01 | 2013-12-10 | Targegen, Inc. | Bi-aryl meta-pyrimidine inhibitors of kinases |
| JP5408660B2 (ja) * | 2007-09-04 | 2014-02-05 | 学校法人東京農業大学 | パラテルフェニル化合物、その薬理学的に許容される塩、その製造方法及び用途 |
| UA103319C2 (en) | 2008-05-06 | 2013-10-10 | Глаксосмитклайн Ллк | Thiazole- and oxazole-benzene sulfonamide compounds |
| CA2781685C (en) | 2009-12-11 | 2018-09-04 | Autifony Therapeutics Limited | Imidazolidinedione derivatives |
| US9133123B2 (en) | 2010-04-23 | 2015-09-15 | Cytokinetics, Inc. | Certain amino-pyridines and amino-triazines, compositions thereof, and methods for their use |
| AR081626A1 (es) | 2010-04-23 | 2012-10-10 | Cytokinetics Inc | Compuestos amino-piridazinicos, composiciones farmaceuticas que los contienen y uso de los mismos para tratar trastornos musculares cardiacos y esqueleticos |
| AR081331A1 (es) | 2010-04-23 | 2012-08-08 | Cytokinetics Inc | Amino- pirimidinas composiciones de las mismas y metodos para el uso de los mismos |
| WO2012060847A1 (en) | 2010-11-07 | 2012-05-10 | Targegen, Inc. | Compositions and methods for treating myelofibrosis |
| EP2649066B1 (en) | 2010-12-06 | 2015-10-21 | Autifony Therapeutics Limited | Hydantoin derivatives useful as kv3 inhibitors |
| CN103596943B (zh) | 2011-06-07 | 2016-10-12 | 奥蒂福尼疗法有限公司 | 用作kv3抑制剂的乙内酰脲衍生物 |
| US9669030B2 (en) | 2012-05-22 | 2017-06-06 | Autifony Therapeutics Limited | Hydantoin derivatives as Kv3 inhibitors |
| EP2852589B1 (en) | 2012-05-22 | 2021-04-28 | Autifony Therapeutics Limited | Triazoles as kv3 inhibitors |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5693611A (en) * | 1996-02-01 | 1997-12-02 | Eli Lilly And Company | Cyclic peptide antifungal agents |
| KR19990087816A (ko) * | 1996-04-22 | 1999-12-27 | 시오노 요시히코 | 신규 테르페닐 화합물 및 이를 함유한 약제 |
| CN1232443A (zh) * | 1996-07-31 | 1999-10-20 | 盐野义制药株式会社 | 新的对三联苯化合物 |
| HN1997000027A (es) * | 1996-12-06 | 1997-06-05 | Pfizer Prod Inc | Derivados de 6-fenil piridil - 2 amina |
| AU7553198A (en) * | 1997-06-12 | 1998-12-30 | Sumitomo Pharmaceuticals Company, Limited | Pyrazole derivatives |
| US6003360A (en) | 1997-07-01 | 1999-12-21 | Wilson Tool International, Inc. | Press brake tool holder |
| WO1999038829A1 (fr) | 1998-01-28 | 1999-08-05 | Shionogi & Co., Ltd. | Nouveau compose tricyclique |
| CA2375909A1 (en) * | 1999-07-19 | 2001-01-25 | Shionogi & Co., Ltd. | Tricyclic compounds bearing acyloxymethoxycarbonyl pendants |
-
2000
- 2000-07-14 US US09/980,475 patent/US7008954B1/en not_active Expired - Fee Related
- 2000-07-14 PL PL00353476A patent/PL353476A1/xx not_active Application Discontinuation
- 2000-07-14 CN CN00810786A patent/CN1364080A/zh active Pending
- 2000-07-14 KR KR1020027000498A patent/KR20020012309A/ko not_active Application Discontinuation
- 2000-07-14 MX MXPA01013452A patent/MXPA01013452A/es unknown
- 2000-07-14 RU RU2002103201/15A patent/RU2230551C2/ru not_active IP Right Cessation
- 2000-07-14 TR TR2002/00099T patent/TR200200099T2/xx unknown
- 2000-07-14 AU AU60159/00A patent/AU763976B2/en not_active Ceased
- 2000-07-14 CA CA002375982A patent/CA2375982A1/en not_active Abandoned
- 2000-07-14 BR BR0012697-7A patent/BR0012697A/pt not_active IP Right Cessation
- 2000-07-14 WO PCT/JP2000/004725 patent/WO2001007032A1/ja not_active Application Discontinuation
- 2000-07-14 HU HU0203575A patent/HUP0203575A3/hu unknown
- 2000-07-14 EP EP00946316A patent/EP1206935A4/en not_active Withdrawn
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2001
- 2001-11-28 ZA ZA200109785A patent/ZA200109785B/en unknown
- 2001-12-21 NO NO20016401A patent/NO20016401L/no not_active Application Discontinuation
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2002
- 2002-11-18 HK HK02108343.5A patent/HK1046645A1/zh unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NO20016401D0 (no) | 2001-12-21 |
| MXPA01013452A (es) | 2002-07-02 |
| AU6015900A (en) | 2001-02-13 |
| NO20016401L (no) | 2002-01-23 |
| KR20020012309A (ko) | 2002-02-15 |
| WO2001007032A1 (fr) | 2001-02-01 |
| TR200200099T2 (tr) | 2002-06-21 |
| BR0012697A (pt) | 2002-04-09 |
| AU763976B2 (en) | 2003-08-07 |
| CN1364080A (zh) | 2002-08-14 |
| HUP0203575A2 (hu) | 2003-02-28 |
| RU2230551C2 (ru) | 2004-06-20 |
| HK1046645A1 (zh) | 2003-01-24 |
| PL353476A1 (en) | 2003-11-17 |
| EP1206935A1 (en) | 2002-05-22 |
| US7008954B1 (en) | 2006-03-07 |
| HUP0203575A3 (en) | 2003-11-28 |
| EP1206935A4 (en) | 2008-07-30 |
| CA2375982A1 (en) | 2001-02-01 |
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