YU33880B - Process for preparing estra-1,3,5-(10)-triens oxidized in positions 3 and 17 - Google Patents
Process for preparing estra-1,3,5-(10)-triens oxidized in positions 3 and 17Info
- Publication number
- YU33880B YU33880B YU1125/67A YU112567A YU33880B YU 33880 B YU33880 B YU 33880B YU 1125/67 A YU1125/67 A YU 1125/67A YU 112567 A YU112567 A YU 112567A YU 33880 B YU33880 B YU 33880B
- Authority
- YU
- Yugoslavia
- Prior art keywords
- triens
- estra
- oxidized
- preparing
- positions
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/566—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol having an oxo group in position 17, e.g. estrone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A61K31/567—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in position 17 alpha, e.g. mestranol, norethandrolone
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J75/00—Processes for the preparation of steroids in general
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (6)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR64481A FR5519M (de) | 1966-06-07 | 1966-06-07 | |
FR75528A FR1514122A (fr) | 1966-06-07 | 1966-09-07 | Dérivés stéroïdes substitués en position 11 à noyau a aromatique et procédé de préparation |
FR86879A FR6021M (de) | 1966-06-07 | 1966-12-09 | |
FR91611A FR6030M (de) | 1966-06-07 | 1967-01-18 | |
FR96848A FR6182M (de) | 1966-06-07 | 1967-02-28 | |
FR98154A FR1540942A (fr) | 1966-06-07 | 1967-03-09 | Dérivés stéroïdes substitués en positions 11 et 17 à noyau a aromatique et procédé de préparation |
Publications (2)
Publication Number | Publication Date |
---|---|
YU112567A YU112567A (en) | 1977-12-31 |
YU33880B true YU33880B (en) | 1978-06-30 |
Family
ID=27546052
Family Applications (6)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
YU1125/67A YU33880B (en) | 1966-06-07 | 1967-06-03 | Process for preparing estra-1,3,5-(10)-triens oxidized in positions 3 and 17 |
YU1758/67A YU33882B (en) | 1966-06-07 | 1967-09-07 | Process for preparing estradiol derivatives |
YU2408/67A YU33725B (en) | 1966-06-07 | 1967-12-08 | Process for preparing 3,17 oxidized esters of1,3,5(10)-trienes |
YU109/68A YU34050B (en) | 1966-06-07 | 1968-01-17 | Process for preparing 3817beta-dihydroxy-11beta-ethoxy-estra-1,2,3(10)-trienes |
YU455/68A YU33883B (en) | 1966-06-07 | 1968-02-27 | Process for preparing 3,17-dihydro-11beta-methoxy-17delta-ethinyl-estra-1,3,5-(10)-trienes |
YU545/68A YU33972B (en) | 1966-06-07 | 1968-03-08 | Process for preparing 3,17beta-dihydroxy-11 beta-ethoxy-17 delta-ethynyl-estra-1,3,5(10)-triene |
Family Applications After (5)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
YU1758/67A YU33882B (en) | 1966-06-07 | 1967-09-07 | Process for preparing estradiol derivatives |
YU2408/67A YU33725B (en) | 1966-06-07 | 1967-12-08 | Process for preparing 3,17 oxidized esters of1,3,5(10)-trienes |
YU109/68A YU34050B (en) | 1966-06-07 | 1968-01-17 | Process for preparing 3817beta-dihydroxy-11beta-ethoxy-estra-1,2,3(10)-trienes |
YU455/68A YU33883B (en) | 1966-06-07 | 1968-02-27 | Process for preparing 3,17-dihydro-11beta-methoxy-17delta-ethinyl-estra-1,3,5-(10)-trienes |
YU545/68A YU33972B (en) | 1966-06-07 | 1968-03-08 | Process for preparing 3,17beta-dihydroxy-11 beta-ethoxy-17 delta-ethynyl-estra-1,3,5(10)-triene |
Country Status (14)
Country | Link |
---|---|
US (2) | US3526648A (de) |
AT (3) | AT301037B (de) |
BE (2) | BE699394A (de) |
CH (3) | CH474495A (de) |
DE (1) | DE1618830C3 (de) |
DK (2) | DK121857B (de) |
ES (5) | ES341435A1 (de) |
FR (6) | FR5519M (de) |
GB (2) | GB1151404A (de) |
IL (2) | IL28112A (de) |
NL (2) | NL6707903A (de) |
SE (2) | SE335979B (de) |
SU (2) | SU483828A3 (de) |
YU (6) | YU33880B (de) |
Families Citing this family (28)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2140258B1 (de) * | 1971-06-07 | 1974-08-23 | Roussel Uclaf | |
US3906096A (en) * | 1971-11-23 | 1975-09-16 | Roussel Uclaf | Novel 11{62 -alkoxy steroids |
FR2183555B1 (de) * | 1972-05-10 | 1975-06-20 | Roussel Uclaf | |
NL7613248A (nl) * | 1976-11-26 | 1978-05-30 | Akzo Nv | Werkwijze voor het bereiden van nieuwe steroid- esters. |
FR2401173A1 (fr) * | 1977-06-27 | 1979-03-23 | Roussel Uclaf | Nouveaux steroides, leur procede de preparation et leur application dans la synthese de steroides marques au tritium |
US4568673A (en) * | 1984-03-20 | 1986-02-04 | Wayne State University | Compositions inhibiting murine MXT ductal carcinoma |
US4636496A (en) * | 1984-03-20 | 1987-01-13 | Wayne State University | Compositions inhibiting murine MXT ductal carcinoma |
US4668668A (en) * | 1984-03-20 | 1987-05-26 | Wayne State University | Compositions inhibiting murine MXT ductal carcinoma |
US4705783A (en) * | 1985-06-25 | 1987-11-10 | Sri International | 9α, 11β-substituted and 11β-substituted estranes |
WO2002022645A2 (en) * | 2000-09-14 | 2002-03-21 | Accelerated Pharmaceuticals, Inc. | Method of making 7alpha-methyl-11beta-methoxy estradiol and related compounds with estrogenic activity |
LT2782584T (lt) | 2011-11-23 | 2021-09-10 | Therapeuticsmd, Inc. | Natūralios kombinuotos pakaitinės hormonų terapijos kompozicijos ir gydymas |
US9301920B2 (en) | 2012-06-18 | 2016-04-05 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
US20150196640A1 (en) | 2012-06-18 | 2015-07-16 | Therapeuticsmd, Inc. | Progesterone formulations having a desirable pk profile |
US10806740B2 (en) | 2012-06-18 | 2020-10-20 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
US10806697B2 (en) | 2012-12-21 | 2020-10-20 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US20130338122A1 (en) | 2012-06-18 | 2013-12-19 | Therapeuticsmd, Inc. | Transdermal hormone replacement therapies |
US10537581B2 (en) | 2012-12-21 | 2020-01-21 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US11266661B2 (en) | 2012-12-21 | 2022-03-08 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US10568891B2 (en) | 2012-12-21 | 2020-02-25 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US10471072B2 (en) | 2012-12-21 | 2019-11-12 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
US9180091B2 (en) | 2012-12-21 | 2015-11-10 | Therapeuticsmd, Inc. | Soluble estradiol capsule for vaginal insertion |
US11246875B2 (en) | 2012-12-21 | 2022-02-15 | Therapeuticsmd, Inc. | Vaginal inserted estradiol pharmaceutical compositions and methods |
AU2015264003A1 (en) | 2014-05-22 | 2016-11-17 | Therapeuticsmd, Inc. | Natural combination hormone replacement formulations and therapies |
CA3006267C (en) * | 2014-11-26 | 2023-08-29 | The Regents Of The University Of California | Estrogen receptor modulators |
US10328087B2 (en) | 2015-07-23 | 2019-06-25 | Therapeuticsmd, Inc. | Formulations for solubilizing hormones |
US10286077B2 (en) | 2016-04-01 | 2019-05-14 | Therapeuticsmd, Inc. | Steroid hormone compositions in medium chain oils |
WO2017173071A1 (en) | 2016-04-01 | 2017-10-05 | Therapeuticsmd, Inc. | Steroid hormone pharmaceutical composition |
US11633405B2 (en) | 2020-02-07 | 2023-04-25 | Therapeuticsmd, Inc. | Steroid hormone pharmaceutical formulations |
-
1966
- 1966-06-07 FR FR64481A patent/FR5519M/fr not_active Expired
- 1966-09-07 FR FR75528A patent/FR1514122A/fr not_active Expired
- 1966-12-09 FR FR86879A patent/FR6021M/fr not_active Expired
-
1967
- 1967-01-18 FR FR91611A patent/FR6030M/fr not_active Expired
- 1967-02-28 FR FR96848A patent/FR6182M/fr not_active Expired
- 1967-03-09 FR FR98154A patent/FR1540942A/fr not_active Expired
- 1967-06-01 GB GB25314/67A patent/GB1151404A/en not_active Expired
- 1967-06-01 GB GB25315/67A patent/GB1152226A/en not_active Expired
- 1967-06-02 US US643061A patent/US3526648A/en not_active Expired - Lifetime
- 1967-06-02 BE BE699394D patent/BE699394A/xx not_active IP Right Cessation
- 1967-06-02 BE BE699393D patent/BE699393A/xx unknown
- 1967-06-03 YU YU1125/67A patent/YU33880B/xx unknown
- 1967-06-05 SE SE07862/67A patent/SE335979B/xx unknown
- 1967-06-05 SE SE07863/67A patent/SE335980B/xx unknown
- 1967-06-06 DK DK294467AA patent/DK121857B/da not_active IP Right Cessation
- 1967-06-06 SU SU1161494A patent/SU483828A3/ru active
- 1967-06-06 ES ES341435A patent/ES341435A1/es not_active Expired
- 1967-06-06 DK DK294567AA patent/DK119925B/da not_active IP Right Cessation
- 1967-06-06 SU SU1250885A patent/SU432714A3/ru active
- 1967-06-07 CH CH806367A patent/CH474495A/fr not_active IP Right Cessation
- 1967-06-07 DE DE1618830A patent/DE1618830C3/de not_active Expired
- 1967-06-07 CH CH806467A patent/CH475965A/fr not_active IP Right Cessation
- 1967-06-07 CH CH450769A patent/CH490361A/fr not_active IP Right Cessation
- 1967-06-07 NL NL6707903A patent/NL6707903A/xx unknown
- 1967-06-07 AT AT532367A patent/AT301037B/de not_active IP Right Cessation
- 1967-06-07 AT AT532267A patent/AT279815B/de not_active IP Right Cessation
- 1967-06-07 NL NL6707906A patent/NL6707906A/xx unknown
- 1967-06-07 AT AT1252868A patent/AT290023B/de not_active IP Right Cessation
- 1967-06-08 IL IL28112A patent/IL28112A/en unknown
- 1967-06-08 IL IL28113A patent/IL28113A/en unknown
- 1967-09-06 ES ES344805A patent/ES344805A1/es not_active Expired
- 1967-09-07 YU YU1758/67A patent/YU33882B/xx unknown
- 1967-12-07 ES ES348057A patent/ES348057A1/es not_active Expired
- 1967-12-08 YU YU2408/67A patent/YU33725B/xx unknown
-
1968
- 1968-01-17 YU YU109/68A patent/YU34050B/xx unknown
- 1968-02-27 ES ES350987A patent/ES350987A1/es not_active Expired
- 1968-02-27 YU YU455/68A patent/YU33883B/xx unknown
- 1968-03-08 ES ES351368A patent/ES351368A1/es not_active Expired
- 1968-03-08 YU YU545/68A patent/YU33972B/xx unknown
-
1969
- 1969-08-25 US US852905A patent/US3579545A/en not_active Expired - Lifetime
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