WO2003026425A1 - Composition antiparasitaire - Google Patents

Composition antiparasitaire Download PDF

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Publication number
WO2003026425A1
WO2003026425A1 PCT/JP2002/008638 JP0208638W WO03026425A1 WO 2003026425 A1 WO2003026425 A1 WO 2003026425A1 JP 0208638 W JP0208638 W JP 0208638W WO 03026425 A1 WO03026425 A1 WO 03026425A1
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WO
WIPO (PCT)
Prior art keywords
methyl
compound
pyridyl
phenyl
tetrahydro
Prior art date
Application number
PCT/JP2002/008638
Other languages
English (en)
Japanese (ja)
Inventor
Naoki Sato
Original Assignee
Sumitomo Chemical Company, Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sumitomo Chemical Company, Limited filed Critical Sumitomo Chemical Company, Limited
Publication of WO2003026425A1 publication Critical patent/WO2003026425A1/fr

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Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines

Definitions

  • the present invention relates to pest control compositions.
  • the present invention provides a compound represented by the formula (I):
  • N * N0 represented by 2 3- [(2-Black port thiazole one rule 5 I) methyl] one 5-methyl-4 double Troy plasminogen perhydro 3, 5- Okisajin (hereinafter, described as Compound (II). ) And formula (III)
  • a pest control composition contained as a component, and a compound (A) and a compound selected from the group consisting of compound (1), compound (II) and compound (III) 1 Treating pests or pest habitats with one or more compounds And a method for controlling pests.
  • the compound (A) in the present invention is a compound described in US Pat. No. 5,498,612, and can be produced according to the description in the publication.
  • Compound (I) in the present invention is a compound described in US Pat. No. 5,304,566, and compound (II) is a compound described in US Pat. No. 5,852,012.
  • the compound (III) is a compound described in US Pat. No. 5,434,181 and can be produced according to the method described in the publication.
  • insect pests to which the composition of the present invention has a controlling effect include the following insects, arthropods such as mites, and nematodes such as nematodes.
  • Hemiptera pests Black-footed deer (Laodelphax striatellus), Brown-footed deer
  • Leafhoppers Nephotettix virescens and other leafhoppers, Aphis gossypii, peach aphids (Myzus persicae), orange aphids (Aphis citricola), aphids aphids (Lipaphis pserudobrassicae), Aphids such as Aphid aphid (Toxoptera aurantii) and Citrus aphid (Toxoptera ciidius)
  • Stink bugs such as Riptortus clavetus and Plaitia stali; Trialeurodes vaporariorum Aonidiella aurantii)
  • Lepidopteran pests Chilo suppressalis, Cnaphalocrocis medinalis, Ostrinia nubilalis, Hellula undalis, Parapediasia teterrella, Notanoa dero vide Species such as Madame Larvae (Plodia interpunctel la), Spodoptera litura, Psyudaletia (Pseudaletia separata), Spodoptera (Maraestra brassicae), Tamanayaga (Agrotis ipsilon), genus Trichophelio Rupa, etc., White butterfly (Pieris rapae), etc., White butterfly (Pieris rapae), etc., Adoxophyes, Graphholita molesta, Codling moths (Cydia pomonella), etc .; Lepidoptera, Limantria, Hupro Species of the genus Cutis, etc .; Suga, such as Plutella xylostella;
  • Pests such as Acaie (Culex pipiens pal lens) and Koga Acaie (Culex tritaeniorhynchus), Aedes spp. Anopheles sinensis and other anopheles, mussuri, Musca domes tica, Musca stabulans and other house flies, blowflies, mosquitoes, gypsophila, and flies (Delia platura) (Anti qua), Flies, such as Liriomyza trifolii, Fruit flies, Flies, Drosophila, Drosophila, Bu, Flies, Flies, etc.
  • Hymenoptera pests such as the wasps (Athalia rosae), mifushi honeybees such as the terrestrial wasp (Arge pagana), wasps (Vespa simillima), wasps such as the hornet wasp (Polites chinensis), and omnivorous monkeys such as the mosquitoes Moni or spores Moni ) Etc., Ariga evening bees etc.
  • Pests such as Western Corn Loom Worm (Diabrotica virgifera virgifera) Southern Corn Lemon (Diabrotica undecimpunctaia howardi) Tortworms, Scarabaeids such as Anomala cuprea, Anomala rufocuprea, etc., Sitophilus zeamais, Lissorhoptrus oryzophilus, Why cis cissis (Hyper) Weevil such as Tenebrio inolitor, Tribolium castaneum, and other beetles; Aulacophora femoralis; And epilacunas such as Epilachna vigintioctopunctata, and other insects, such as the beetles, the locust beetles, and the opal beetle OPaederus fuscipes.
  • Bots such as Western Corn Loom Worm (Diabrotica virgifera virgifera) Southern Corn Lemon (Dia
  • Cockroach pests Blattella germanica, Black cockroach (Periplaneta fuliginosa), Black cockroach (Periplaneta americana), Black cockroach (Periplaneta brunnea), Black cockroach (Blatta oriental is) and the like.
  • Thistle pests Thrips palmi thrips (Thrips palii), Nepal thrips (Thrips tabaci), Thrips thrips (Thrips hawaiiensis), Chestnut yellow thistles Thrips (Frankliniella occidental is), Power thrips (Ponticulothrips diospyrosu).
  • Orthoptera Pests, grasshoppers, etc.
  • Lepidopteran pests cat flea (Ctenocephalides felis), wild flea (Ctenocephalides canis), human flea (Pulex irritans) and the like.
  • Pests of the louse Lice lice (Pediculus humanus humanus), white lice (Pediculus humanus corporis) ⁇ lice (Phthirus pubis), etc.
  • Coleoptera Coleoptera (Porcellio scaber), Coleoptera cricket (Porcel 1 ionides pruinosus), talented Dankomushi (Armadillidium vulgare).
  • Centipedes Centipedes: Tobism Kade (Scolopendra subspinipes mutilans), Aozum Kade (Scolopendra subspinipes japonica), Akasum Kade (Scolopendra subspinipes raul tidens), Geji (There Lord oda hilgendorf i) and the like.
  • Millipede Oyster Millet (Oxidus gracilis), Obiba Bay Millet (Parafontaria laminata laminata) etc.
  • Pests of the order Acarina Tetranyc us urticae, Tetranychus kanzawai> Citrus spider mite (Panonychus citri) Linnino, mites (Panonychus ulm re, Oligonicus spp., Aculops lycos pelis culs Aculops lycosper cul (Ph.
  • Dermatophagoids Calacarus carinatus
  • Polyphagotarsonemus latus Polyphagotarsonemus latus
  • Scarabidae Coldadae
  • Dermatophagoides Ticks
  • Dermatophagoides farinae And mites Chelacaropsis moorei
  • mites mites and the like.
  • Nematodes such as southern exotic (Pratylenchus coffeae), northern exotic (Pratylenchus fallax), prawn (Pratylenchus loosi), and walnut (Pratylenchus vulnus) Nematodes such as cysts (Heterodera glycines) and potato cysts (Globodera rostochiensis), Meloidogyne hapla, Meloidogyne incognita and others , Aphelenchoides besseyi, Aphelenchoides fragarieae, etc., Afelencoides, Ishukusenyu, Pengsenyu, Pincentiuyu, Longidurus, Trichodorus and the like.
  • compound (A) and one or more compounds selected from the group consisting of compound (1), compound (II) and compound (III) (hereinafter, referred to as compound (B)).
  • the ratio is not limited as long as it exhibits a synergistic effect. Specifically, for example, the ratio by weight is usually 30: 1 to 1:30, preferably the ratio is 20: 1 to 1:20, More preferably, the ratio is 10: 1 to 1:10.
  • composition of the present invention can be used in the form of a mixture of the compound (A) and the compound (B) as it is, but usually, a solid alone, a liquid carrier and / or a gaseous carrier are added, Add surfactants and other formulation auxiliaries as needed to make oils, emulsions, flowables, granules, powders, aerosols, microcapsules, ULVs, sheet formulations, smoke Formulated into smoke, spot-on, pour-on, shampoo, bait, etc.
  • the total amount of compound (A) and compound (B) is usually from 01 to 90% by weight.
  • solid carriers used in the formulation include clays (kaolin clay, diatomaceous earth, synthetic hydrous silicon oxide, bentonite, fupasami clay, acid clay, etc.), talc, ceramics, and other inorganic minerals (sericite, quartz) , Sulfur, activated carbon, calcium carbonate, hydrated silica, etc.) and fine powders and granular materials such as chemical fertilizers (ammonium sulfate, phosphorous ammonium, ammonium nitrate, urea, salt ammonium, etc.).
  • liquid carriers examples include water, alcohols (methanol, ethanol, etc.), ketones (acetone, methylethyl ketone, etc.), aromatic hydrocarbons (benzene, toluene, xylene, ethylbenzene, methylnaphthalene, etc.), fats Group hydrocarbons (hexane, cyclohexane, kerosene, gas oil, etc.), esters (ethyl acetate, butyl acetate, etc.), nitriles (acetonitrile, isoptyronitrile, etc.), ethers (diisopropyl ether, dioxane) Acid amides (N, N-dimethylformamide, N, N-dimethylacetamide, etc.), halogenated hydrocarbons (dichloromethane, trichloroethane, carbon tetrachloride, etc.), dimethyl sulfoxide and vegetable oils (soybean oil
  • gaseous carrier examples include fluorocarbon, butane gas, LPG (liquefied petroleum gas), dimethyl ether, and carbon dioxide gas.
  • surfactant examples include alkyl sulfates, alkyl sulfonates, alkyl sulfonates, alkyl aryl ethers and their polyoxyethylenes, polyethylene glycol ethers, polyhydric alcohol esters, and sugars. Alcohol derivatives are mentioned.
  • Other pharmaceutical auxiliaries include fixing agents, dispersants and stabilizers, such as casein, gelatin, polysaccharides (starch, gum arabic, cellulose derivatives, alginic acid, etc.), lignin derivatives, bentonite, Saccharides, synthetic water-soluble polymers (polyvinyl alcohol, polyvinylpyrrolidone, polyacrylic acids, etc.), PAP (isopropyl oxyphosphate), BHT (2,6-di-tert-butyl-4-methylphenol), BHA ( Two — A mixture of tert-butyl-4-methoxyphenol and 3-iert-butyl-4-methoxyphenol), vegetable oils, mineral oils, fatty acids and fatty acid esters.
  • fixing agents such as casein, gelatin, polysaccharides (starch, gum arabic, cellulose derivatives, alginic acid, etc.), lignin derivatives, bentonite, Saccharides, synthetic water-soluble polymers (polyvinyl alcohol,
  • Base materials for poison bait include, for example, feed ingredients such as cereal flour, vegetable oil, sugar, and crystalline cellulose; antioxidants such as dibutylhydroxytoluene and nordihydroguaiaretic acid; preservatives such as dehydroacetic acid; and pepper powder.
  • Infant-inducing agents such as children and pets, cheese flavor, evening onion flavor, and pest-inducing flavors such as peanut oil.
  • the composition of the present invention can also be prepared, depending on the form of the preparation, by mixing a preparation of the compound (A) with a preparation of the compound (B). Furthermore, it can also be prepared by mixing a diluent of the compound (A) formulated and a diluent of the compound (B) formulated at the time of application.
  • the method for controlling pests of the present invention is usually carried out by applying the composition of the present invention to a pest or a habitat of the pests.
  • the effect of the composition of the present invention can be obtained by applying the composition to a habitat of a pest.
  • the ratio of the compound (A) to the compound (B) is usually 30: 1 to 1:30 by weight, preferably 20: 1 to 1:20, more preferably The ratio is 10: 1 to 1:10.
  • the application amount is 0.1 to 1 in terms of the total amount of the compound (A) and the compound (B) per 100 m 2 . 0 0 0 g.
  • Emulsions, flowables and the like are usually diluted with water so as to have an active ingredient concentration of 10 to 1000 ppm, and granules and powders are usually applied as they are.
  • These preparations may be directly applied to plants such as crops to be protected from pests, and by treating these preparations with soil, pests that inhabit the soil can be controlled.
  • composition of the present invention can be used together with other insecticides, nematicides, acaricides, fungicides, herbicides, plant growth regulators, synergists, fertilizers, soil conditioners, animal feeds, etc. it can.
  • the present invention will be described in more detail with reference to Formulation Examples of the present mixed composition and Examples of the method of the present invention, but the present invention is not limited to these Examples. First, formulation examples of the composition of the present invention will be described. In addition, parts represent parts by weight.
  • Emulsion was prepared by uniformly mixing 5 parts of compound (A), 5 parts of any of compounds (I) to (III), 8 parts of polyoxyethylene styrene, 2 parts of calcium dodecylbenzenesulfonate, and 80 parts of xylene. obtain.
  • test examples show that the composition of the present invention is useful as a pest control composition.
  • the cucumber was air-dried, the pot was placed in a plastic cup, covered, and cultivated in a greenhouse (room temperature: 25 ° C) for 7 days. Seven days after the application of the spray solution, the number of adult larvae (adults + larvae) infesting the cucumber was investigated.
  • T 7DAT Number of insects 7 days after treatment in treated plants
  • T pre number of insects before treatment in treated plants
  • C 7DAT Number of insects 7 days after treatment in untreated plants
  • composition of the present invention has an excellent controlling effect on pests and can effectively control pests.

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  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

L'invention concerne une composition antiparasitaire qui contient en tant qu'ingrédients actifs le composé 5-chloro-6-(1-fluoroéthyl)-N-[2-[4-(trifluorométhoxy)phényl]éthyl]pyrimidin-4-ylamine, représenté par la formule (A), et au moins un composé choisi dans le groupe comprenant N1[(6-chloro-3-pyridyl)méthyl]-N2-cyano-N1-méthylacétamidine, 3-[(2-chlorothiazol-5-yl)méthyl]-5-méthyl-4-nitroiminoperhydro-1, 3, 5-oxidiazine, et 1-[(tétrahydro-3-furanyl)méthyl]-2-nitro-3-méthylguanidine.
PCT/JP2002/008638 2001-09-07 2002-08-28 Composition antiparasitaire WO2003026425A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2001-271535 2001-09-07
JP2001271535 2001-09-07

Publications (1)

Publication Number Publication Date
WO2003026425A1 true WO2003026425A1 (fr) 2003-04-03

Family

ID=19097029

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/JP2002/008638 WO2003026425A1 (fr) 2001-09-07 2002-08-28 Composition antiparasitaire

Country Status (1)

Country Link
WO (1) WO2003026425A1 (fr)

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0057440A1 (fr) * 1981-01-29 1982-08-11 Sankyo Company Limited Dérivés de l'aminopyrimidine, leurs procédés de préparation et compositions fongicides, insecticides et acaricides les contenant
EP0665225A1 (fr) * 1994-02-01 1995-08-02 Ube Industries, Ltd. 4-Phénylaminopyrimidines, procédé pour leur préparation et pesticides pour l'agriculture et l'horticulture les contenant
JP2000080005A (ja) * 1998-06-22 2000-03-21 Sumitomo Chem Co Ltd 木材害虫駆除組成物

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0057440A1 (fr) * 1981-01-29 1982-08-11 Sankyo Company Limited Dérivés de l'aminopyrimidine, leurs procédés de préparation et compositions fongicides, insecticides et acaricides les contenant
EP0665225A1 (fr) * 1994-02-01 1995-08-02 Ube Industries, Ltd. 4-Phénylaminopyrimidines, procédé pour leur préparation et pesticides pour l'agriculture et l'horticulture les contenant
JP2000080005A (ja) * 1998-06-22 2000-03-21 Sumitomo Chem Co Ltd 木材害虫駆除組成物

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