UY37315A - Procedimiento para la preparación de derivados de piridina halogenados - Google Patents
Procedimiento para la preparación de derivados de piridina halogenadosInfo
- Publication number
- UY37315A UY37315A UY0001037315A UY37315A UY37315A UY 37315 A UY37315 A UY 37315A UY 0001037315 A UY0001037315 A UY 0001037315A UY 37315 A UY37315 A UY 37315A UY 37315 A UY37315 A UY 37315A
- Authority
- UY
- Uruguay
- Prior art keywords
- preparation
- halogenated
- procedure
- formula
- halogen
- Prior art date
Links
- 229910052736 halogen Inorganic materials 0.000 abstract 3
- 125000005843 halogen group Chemical group 0.000 abstract 2
- 125000004169 (C1-C6) alkyl group Chemical group 0.000 abstract 1
- 125000000171 (C1-C6) haloalkyl group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 150000002367 halogens Chemical class 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 150000003222 pyridines Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/79—Acids; Esters
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D213/79—Acids; Esters
- C07D213/803—Processes of preparation
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F3/00—Compounds containing elements of Groups 2 or 12 of the Periodic Table
- C07F3/06—Zinc compounds
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyridine Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Abstract
La presente invención se refiere a un procedimiento para la preparación de derivados de piridina halogenados de la fórmula (II) partiendo de compuestos de fórmula (I) a través de compuestos intermedios de la fórmula (IIIa) o (IIIb) en el que los radicales Q y W son independientemente halógeno, R2 es halógeno o –O-pivaloilo e Y es halógeno, CO2R1 o NO2, donde R1 es (C1-C6)-alquilo o (C1-C6)-haloalquilo.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP16178022 | 2016-07-05 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY37315A true UY37315A (es) | 2018-01-31 |
Family
ID=56363777
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY0001037315A UY37315A (es) | 2016-07-05 | 2017-07-03 | Procedimiento para la preparación de derivados de piridina halogenados |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US10766909B2 (es) |
| EP (1) | EP3481805B1 (es) |
| JP (1) | JP7034953B2 (es) |
| KR (1) | KR102408111B1 (es) |
| CN (1) | CN109476601B (es) |
| AR (1) | AR108943A1 (es) |
| BR (1) | BR112019000213B1 (es) |
| DK (1) | DK3481805T3 (es) |
| ES (1) | ES2941903T3 (es) |
| FI (1) | FI3481805T3 (es) |
| IL (1) | IL263970B (es) |
| MX (1) | MX2019000254A (es) |
| TW (1) | TWI766872B (es) |
| UY (1) | UY37315A (es) |
| WO (1) | WO2018007224A1 (es) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI820231B (zh) | 2018-10-11 | 2023-11-01 | 德商拜耳廠股份有限公司 | 用於製備經取代咪唑衍生物之方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3947457A (en) | 1974-12-27 | 1976-03-30 | The Dow Chemical Company | Method for preparing 2,5-dihalo- and 2,5,6-trihalopyridines |
| US8569337B2 (en) * | 2008-07-23 | 2013-10-29 | Vertex Pharmaceuticals Incorporated | Tri-cyclic pyrazolopyridine kinase inhibitors |
| EP2630134B9 (en) | 2010-10-20 | 2018-04-18 | Pfizer Inc | Pyridine-2- derivatives as smoothened receptor modulators |
| WO2016010897A1 (en) | 2014-07-14 | 2016-01-21 | Incyte Corporation | Bicyclic heteroaromatic carboxamide compounds useful as pim kinase inhibitors |
-
2017
- 2017-06-28 MX MX2019000254A patent/MX2019000254A/es unknown
- 2017-06-28 CN CN201780041677.1A patent/CN109476601B/zh active Active
- 2017-06-28 ES ES17736603T patent/ES2941903T3/es active Active
- 2017-06-28 BR BR112019000213-8A patent/BR112019000213B1/pt active IP Right Grant
- 2017-06-28 DK DK17736603.6T patent/DK3481805T3/da active
- 2017-06-28 WO PCT/EP2017/065989 patent/WO2018007224A1/de unknown
- 2017-06-28 KR KR1020197001561A patent/KR102408111B1/ko active IP Right Grant
- 2017-06-28 FI FIEP17736603.6T patent/FI3481805T3/fi active
- 2017-06-28 EP EP17736603.6A patent/EP3481805B1/de active Active
- 2017-06-28 US US16/312,568 patent/US10766909B2/en active Active
- 2017-06-28 JP JP2018567735A patent/JP7034953B2/ja active Active
- 2017-07-03 UY UY0001037315A patent/UY37315A/es not_active Application Discontinuation
- 2017-07-03 TW TW106122177A patent/TWI766872B/zh active
- 2017-07-03 AR ARP170101838A patent/AR108943A1/es unknown
-
2018
- 2018-12-26 IL IL263970A patent/IL263970B/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| US10766909B2 (en) | 2020-09-08 |
| IL263970B (en) | 2021-06-30 |
| CN109476601A (zh) | 2019-03-15 |
| KR20190025626A (ko) | 2019-03-11 |
| TW201811747A (zh) | 2018-04-01 |
| DK3481805T3 (da) | 2023-04-11 |
| IL263970A (en) | 2019-01-31 |
| MX2019000254A (es) | 2019-05-27 |
| AR108943A1 (es) | 2018-10-10 |
| TWI766872B (zh) | 2022-06-11 |
| CN109476601B (zh) | 2022-10-28 |
| US20190330241A1 (en) | 2019-10-31 |
| ES2941903T3 (es) | 2023-05-26 |
| BR112019000213A2 (pt) | 2019-04-16 |
| FI3481805T3 (fi) | 2023-04-25 |
| EP3481805A1 (de) | 2019-05-15 |
| WO2018007224A1 (de) | 2018-01-11 |
| KR102408111B1 (ko) | 2022-06-10 |
| EP3481805B1 (de) | 2023-01-18 |
| JP2019521123A (ja) | 2019-07-25 |
| BR112019000213B1 (pt) | 2022-10-25 |
| JP7034953B2 (ja) | 2022-03-14 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 109 | Application deemed to be withdrawn |
Effective date: 20230626 |