UY32043A - Nueva forma cristalina b de 4-(5-{ (1r)-1-[5-(3-clorofenil)isoxazol-3-il]etoxi} -4-metil-4h-1,2,4-triazol-3-il)piridina - Google Patents

Nueva forma cristalina b de 4-(5-{ (1r)-1-[5-(3-clorofenil)isoxazol-3-il]etoxi} -4-metil-4h-1,2,4-triazol-3-il)piridina

Info

Publication number
UY32043A
UY32043A UY0001032043A UY32043A UY32043A UY 32043 A UY32043 A UY 32043A UY 0001032043 A UY0001032043 A UY 0001032043A UY 32043 A UY32043 A UY 32043A UY 32043 A UY32043 A UY 32043A
Authority
UY
Uruguay
Prior art keywords
new crystalline
isoxazol
triazol
methyl
chlorophenil
Prior art date
Application number
UY0001032043A
Other languages
English (en)
Inventor
Hans Astroem
Profir Veronica
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of UY32043A publication Critical patent/UY32043A/es

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/422Oxazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P19/00Drugs for skeletal disorders
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    • A61P19/00Drugs for skeletal disorders
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    • A61P25/00Drugs for disorders of the nervous system
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
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  • Bioinformatics & Cheminformatics (AREA)
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  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
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  • Neurology (AREA)
  • Biomedical Technology (AREA)
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Abstract

La presente invención se refiere a una nueva forma cristalina de 4-(5-{(1R)-1-[5-(3- clorofenil)isoxazol-3-il] etoxi}-4-metil-4H-1,2,4-triazol-3-il)piridina. Además, la presente invención también se refiere al uso de una nueva forma cristalina para el tratamiento de trastornos digestivos, a composiciones farmacéuticas que la contienen así como a procesos para la preparación de la nueva forma cristalina.
UY0001032043A 2008-08-12 2009-08-11 Nueva forma cristalina b de 4-(5-{ (1r)-1-[5-(3-clorofenil)isoxazol-3-il]etoxi} -4-metil-4h-1,2,4-triazol-3-il)piridina UY32043A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US8805308P 2008-08-12 2008-08-12

Publications (1)

Publication Number Publication Date
UY32043A true UY32043A (es) 2010-03-26

Family

ID=41669086

Family Applications (1)

Application Number Title Priority Date Filing Date
UY0001032043A UY32043A (es) 2008-08-12 2009-08-11 Nueva forma cristalina b de 4-(5-{ (1r)-1-[5-(3-clorofenil)isoxazol-3-il]etoxi} -4-metil-4h-1,2,4-triazol-3-il)piridina

Country Status (15)

Country Link
US (1) US20100041706A1 (es)
EP (1) EP2324019A4 (es)
JP (1) JP2011530590A (es)
KR (1) KR20110040910A (es)
CN (1) CN102177158A (es)
AR (1) AR073268A1 (es)
AU (1) AU2009282523A1 (es)
BR (1) BRPI0917465A2 (es)
CA (1) CA2733922A1 (es)
IL (1) IL210923A0 (es)
MX (1) MX2011001549A (es)
RU (1) RU2011103224A (es)
TW (1) TW201011016A (es)
UY (1) UY32043A (es)
WO (1) WO2010019101A1 (es)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6627646B2 (en) * 2001-07-17 2003-09-30 Sepracor Inc. Norastemizole polymorphs
US7585881B2 (en) * 2004-02-18 2009-09-08 Astrazeneca Ab Additional heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
UY29796A1 (es) * 2005-09-29 2007-04-30 Astrazeneca Ab Nuevos compuestos para el tratamiento de trastornos neurológicos, psiquiátricos o del dolor
WO2007043939A1 (en) * 2005-10-07 2007-04-19 Astrazeneca Ab Novel crystalline form of 3,5-dibromo-n- [(2s)-2-(-4-fluorophenyl)-4-(3-morpholin-4-ylazetidin-1-yl)butyl] -n-methylbenzamide, modification a
TW200821305A (en) * 2006-10-05 2008-05-16 Astrazeneca Ab MGluR5 modulators

Also Published As

Publication number Publication date
AU2009282523A1 (en) 2010-02-18
RU2011103224A (ru) 2012-09-20
CN102177158A (zh) 2011-09-07
IL210923A0 (en) 2011-04-28
MX2011001549A (es) 2011-03-15
US20100041706A1 (en) 2010-02-18
WO2010019101A1 (en) 2010-02-18
JP2011530590A (ja) 2011-12-22
BRPI0917465A2 (pt) 2017-04-04
EP2324019A4 (en) 2011-10-05
KR20110040910A (ko) 2011-04-20
CA2733922A1 (en) 2010-02-18
TW201011016A (en) 2010-03-16
EP2324019A1 (en) 2011-05-25
AR073268A1 (es) 2010-10-28

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