UY31514A1 - Una ciano piperidinil-fenil-oxazolidinona y uso de la misma - Google Patents

Una ciano piperidinil-fenil-oxazolidinona y uso de la misma

Info

Publication number
UY31514A1
UY31514A1 UY31514A UY31514A UY31514A1 UY 31514 A1 UY31514 A1 UY 31514A1 UY 31514 A UY31514 A UY 31514A UY 31514 A UY31514 A UY 31514A UY 31514 A1 UY31514 A1 UY 31514A1
Authority
UY
Uruguay
Prior art keywords
phenyl
compound
piperidinil
oxazolidinone
cyber
Prior art date
Application number
UY31514A
Other languages
English (en)
Inventor
Monserrat Cano
Guglietta Antonio
Palomer Albert
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of UY31514A1 publication Critical patent/UY31514A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

La invencion proporciona un compuesto de formula (I), o cualquiera de sus enantiomeros o mezclas de los mismos, o sus sales farmacéuticamente aceptables o solvatos, para uso como un medicamento. El compuesto de formula (I) es activo contra patogenos humanos y veterinarios Gram-positivos y algunos Gram-negativos con una actividad inhibidora débil de la monoamina oxidasa (MAO). Son utiles para el tratamiento de infecciones bacterianas. La invencion también describe formas del compuesto (S)-N.[3-[4-4-ciano-piperidin-1-il)-3-fluoro-fenil]-2-oxo-oxazolidin-5-ilmetil}-acetamida.
UY31514A 2007-12-17 2008-12-05 Una ciano piperidinil-fenil-oxazolidinona y uso de la misma UY31514A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP07150076A EP2072513A1 (en) 2007-12-17 2007-12-17 A cyano piperidinyl-phenil-oxazolidinone and use thereof

Publications (1)

Publication Number Publication Date
UY31514A1 true UY31514A1 (es) 2009-07-17

Family

ID=39472513

Family Applications (1)

Application Number Title Priority Date Filing Date
UY31514A UY31514A1 (es) 2007-12-17 2008-12-05 Una ciano piperidinil-fenil-oxazolidinona y uso de la misma

Country Status (7)

Country Link
EP (1) EP2072513A1 (es)
AR (1) AR069261A1 (es)
AU (1) AU2008337518A1 (es)
CL (1) CL2008003753A1 (es)
TW (1) TW200934492A (es)
UY (1) UY31514A1 (es)
WO (1) WO2009077484A2 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101128029B1 (ko) 2010-03-08 2012-03-29 주식회사 레고켐 바이오사이언스 (ｒ)-3-(3-플루오로-4-(1-메틸-5,6-다이하이드로-1,2,4-트리아진-4(1ｈ)-일)페닐)-5-(치환된 메틸)옥사졸리딘-2-온 유도체의 제조방법
WO2012121424A1 (ko) * 2011-03-04 2012-09-13 (주)레고켐바이오사이언스 사이클릭 아미드라존 기를 가지는 신규한 옥사졸리디논 유도체 및 이를 함유하는 의약 조성물

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1250538A (es) 1969-03-18 1971-10-20
US5668286A (en) * 1994-03-15 1997-09-16 Pharmacia & Upjohn Company Oxazolidinone derivatives and pharmaceutical compositions containing them
CA2492743A1 (en) * 2002-07-11 2004-01-22 Wockhardt Limited Antimicrobial oxazolidinones, process of their preparation, and pharmaceutical compositions containing them
US7687627B2 (en) * 2003-09-08 2010-03-30 Wockhardt Limited Substituted piperidino phenyloxazolidinones having antimicrobial activity with improved in vivo efficacy
PE20060619A1 (es) 2004-07-29 2006-07-11 Ferrer Int Derivados de oxazolidinona como antibacterianos
EP1912980A2 (en) 2005-06-20 2008-04-23 Wockhardt Limited Oxazolidinones bearing antimicrobial activity composition and methods of preparation

Also Published As

Publication number Publication date
AR069261A1 (es) 2010-01-13
CL2008003753A1 (es) 2009-05-29
WO2009077484A3 (en) 2009-10-01
WO2009077484A2 (en) 2009-06-25
TW200934492A (en) 2009-08-16
AU2008337518A1 (en) 2009-06-25
EP2072513A1 (en) 2009-06-24

Similar Documents

Publication Publication Date Title
ES2523968T3 (es) Terapia de combinación antibacteriana para el tratamiento de infecciones por bacterias Gram-positivas
CO2018010966A2 (es) Nuevos derivados de pirazolopirimidina
ECSP16073620A (es) Compuestos organicos de monobactam para el tratamiento de infecciones bacterianas
BR112012025844A2 (pt) uso de nanofibras snag
CL2021001042A1 (es) Nuevos compuestos antihelmínticos
CO6541645A2 (es) Compuestos de indol y su uso farmaceutico
ES2571998T3 (es) Composiciones y usos médicos de derivados del ajoeno
HK1138184A1 (en) Combination medicaments for treating bacterial infections
CO6620071A2 (es) Forma cristalina del fosfato de dihidrogeno r)-3-(4-(2-(2-metiltetrazol-5-il)piridin-5-il)-3-fluorofenil)-5-hidroximetil oxazolidin-2-ona
UY32462A (es) Derivados de bifenilo novedosos para el tratamiento de infección por virus de hepatitis c 644
UY33622A (es) Isoxazolín oximas como agentes antiparasitarios
ECSP11010949A (es) Inhibidores de las enzimas de proteína cinasa activadas por mitógeno p38
CL2009000990A1 (es) Uso de epotilona d para el tratamiento de enfermedades asociadas a tau, tal como enfermedad alzheimer, parkinson, entre otras.
UY31860A (es) Piridinas de tiazolo como inhibidoras de la adn girasa
ECSP10010704A (es) Sales y polimorfos de un compuesto de tetraticlina
UY30544A1 (es) Compuestos de pirrolo-piperidina y sales farmacéuticametne aceptables de los mismos, procesos de fabricacion, composiciones y aplicaciones
AR074604A1 (es) Derivados de 5-amino-2-(1-hidroxi-etil)-tetrahidropirano.
CR11825A (es) Derivados de urea heterociclicos para el tratamiento de infecciones bacterianas
GEP20186857B (en) Saturated nitrogen and n-acylated heterocycles potentiating the activity of an active antibiotic against mycobacteria
CU20100063A7 (es) Benzotiazoles como moduladores del receptor de grelina
CO6761349A2 (es) Proteína antimicrobiana
UY31514A1 (es) Una ciano piperidinil-fenil-oxazolidinona y uso de la misma
PA8640401A1 (es) Oxazolididonas y composiciones y metodos relacionados
CR9691A (es) Inhibidores de 6-alquilideno-peneme b-lactama biciclicos y combinacion antibiotica de b-lactama: un antibiotico de amplio espectro
UY31953A (es) 3-cianopirrolidinil-fenil-oxazolidinonas como agentes antibacterianos