UY30511A1 - Agonistas de ep2 - Google Patents
Agonistas de ep2Info
- Publication number
- UY30511A1 UY30511A1 UY30511A UY30511A UY30511A1 UY 30511 A1 UY30511 A1 UY 30511A1 UY 30511 A UY30511 A UY 30511A UY 30511 A UY30511 A UY 30511A UY 30511 A1 UY30511 A1 UY 30511A1
- Authority
- UY
- Uruguay
- Prior art keywords
- agonists
- compounds
- methods
- preparation
- provides
- Prior art date
Links
- 239000000556 agonist Substances 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 208000010412 Glaucoma Diseases 0.000 abstract 1
- 230000004410 intraocular pressure Effects 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
- C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C311/03—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C311/04—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by singly-bound oxygen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/01—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms
- C07C311/02—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C311/03—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C311/06—Sulfonamides having sulfur atoms of sulfonamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atoms of the sulfonamide groups bound to hydrogen atoms or to acyclic carbon atoms to acyclic carbon atoms of hydrocarbon radicals substituted by carboxyl groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Ophthalmology & Optometry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
- Pyridine Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Heterocyclic Compounds Containing Sulfur Atoms (AREA)
Abstract
La invencion proporciona agonistas de EP2, procedimientos para su preparacion, composiciones farmacéuticas que contienen estos compuestos y procedimientos de uso de estos compuestos y composiciones para reducir la presion intraocular y tratar así el glaucoma.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US83390706P | 2006-07-28 | 2006-07-28 | |
US94192307P | 2007-06-04 | 2007-06-04 |
Publications (1)
Publication Number | Publication Date |
---|---|
UY30511A1 true UY30511A1 (es) | 2008-02-29 |
Family
ID=38896126
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UY30511A UY30511A1 (es) | 2006-07-28 | 2007-07-27 | Agonistas de ep2 |
Country Status (26)
Country | Link |
---|---|
US (2) | US7622475B2 (es) |
EP (1) | EP2059507B1 (es) |
JP (1) | JP4583500B2 (es) |
KR (1) | KR101088942B1 (es) |
AP (1) | AP2009004754A0 (es) |
AR (1) | AR062122A1 (es) |
AU (1) | AU2007280130B2 (es) |
BR (1) | BRPI0714683A2 (es) |
CA (1) | CA2659184C (es) |
CL (1) | CL2007002207A1 (es) |
CR (1) | CR10554A (es) |
EA (1) | EA200970067A1 (es) |
EC (1) | ECSP099071A (es) |
GT (1) | GT200700064A (es) |
HK (1) | HK1133876A1 (es) |
IL (1) | IL196355A0 (es) |
MA (1) | MA30604B1 (es) |
MX (1) | MX2009001062A (es) |
NO (1) | NO20090738L (es) |
NZ (1) | NZ573964A (es) |
PE (1) | PE20080408A1 (es) |
RS (1) | RS20090002A (es) |
TN (1) | TN2009000028A1 (es) |
TW (1) | TWI372757B (es) |
UY (1) | UY30511A1 (es) |
WO (1) | WO2008015517A2 (es) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SI2264009T1 (sl) * | 2008-03-12 | 2019-05-31 | Ube Industries, Ltd. | Spojina piridilaminoocetne kisline |
US8685986B2 (en) | 2009-03-30 | 2014-04-01 | Ube Industries, Ltd. | Medical composition for treatment or prophylaxis of glaucoma |
WO2011030865A1 (ja) * | 2009-09-11 | 2011-03-17 | 宇部興産株式会社 | 置換ベンジル化合物 |
KR20120068902A (ko) * | 2009-09-11 | 2012-06-27 | 우베 고산 가부시키가이샤 | 아닐린 화합물 |
WO2011030872A1 (ja) * | 2009-09-11 | 2011-03-17 | 宇部興産株式会社 | スルホンアミド化合物 |
AU2010293410A1 (en) * | 2009-09-11 | 2012-05-03 | Ube Industries, Ltd. | Substituted carbonyl compounds |
WO2011030871A1 (ja) * | 2009-09-11 | 2011-03-17 | 宇部興産株式会社 | N-置換ヘテロアリール化合物 |
WO2011030873A1 (ja) * | 2009-09-11 | 2011-03-17 | 宇部興産株式会社 | ベンジル化合物 |
WO2011078303A1 (ja) | 2009-12-25 | 2011-06-30 | 宇部興産株式会社 | アミノピリジン化合物 |
SG187861A1 (en) * | 2010-08-17 | 2013-03-28 | Allergan Inc | Ep2 or ep4 agonists for treating corneal haze |
PE20142083A1 (es) | 2011-09-16 | 2014-12-30 | Fovea Pharmaceuticals | Derivados de anilina, su preparacion y su aplicacion terapeutica |
EP2804605A4 (en) * | 2012-01-20 | 2015-07-08 | Acucela Inc | SUBSTITUTED HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF DISEASES |
EP2844638A1 (en) | 2012-05-03 | 2015-03-11 | Takeda GmbH | Novel ep2 receptor agonists |
US9339496B2 (en) * | 2012-07-13 | 2016-05-17 | Santen Pharmaceutical Co., Ltd. | Composition for treating or preventing glaucoma comprising a sulfonamide compound, and a beta-receptor antagonist |
EP2980075A4 (en) * | 2013-03-28 | 2016-08-10 | Ube Industries | SUBSTITUTED BIARYL CONNECTION |
JP2017206443A (ja) * | 2014-09-26 | 2017-11-24 | 宇部興産株式会社 | 置換ビアリール化合物及び他の医薬の組み合わせ |
JP2017206445A (ja) * | 2014-09-26 | 2017-11-24 | 宇部興産株式会社 | 呼吸器疾患の治療及び/又は予防のための医薬組成物 |
CA2991015A1 (en) * | 2015-07-01 | 2017-01-05 | Santen Pharmaceutical Co., Ltd. | Depot preparation containing citric acid ester |
Family Cites Families (13)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4599353A (en) * | 1982-05-03 | 1986-07-08 | The Trustees Of Columbia University In The City Of New York | Use of eicosanoids and their derivatives for treatment of ocular hypertension and glaucoma |
US5296504A (en) * | 1988-09-06 | 1994-03-22 | Kabi Pharmacia | Prostaglandin derivatives for the treatment of glaucoma or ocular hypertension |
UA59384C2 (uk) * | 1996-12-20 | 2003-09-15 | Пфайзер, Інк. | Похідні сульфонамідів та амідів як агоністи простагландину, фармацевтична композиція та способи лікування на їх основі |
UA67754C2 (uk) | 1997-10-10 | 2004-07-15 | Пфайзер, Інк. | Агоністи простагландину, фармацевтична композиція на їх основі (варіанти), спосіб нарощення та збереження кісткової маси у хребетних та спосіб лікування (варіанти) |
EP1000619A3 (en) * | 1998-06-23 | 2002-07-24 | Pfizer Products Inc. | Method for treating glaucoma |
IL139941A0 (en) | 1999-12-02 | 2002-02-10 | Pfizer Prod Inc | Use of prostaglandin agonists to treat erectile dysfunction or impotence |
US20020161026A1 (en) * | 2000-11-07 | 2002-10-31 | Paralkar Vishwas M. | Combination therapies for the stimulation of bone growth |
EP1448182A1 (en) * | 2001-11-30 | 2004-08-25 | Pfizer Products Inc. | Pharmaceutical compositions and methods for administering ep 2 receptor selective agonists |
CN1625549A (zh) * | 2002-01-31 | 2005-06-08 | 辉瑞产品公司 | (3-{[4-叔丁基-苄基)-(吡啶-3-磺酰基)-氨基]-甲基}-苯氧基)-乙酸的代谢物 |
JP2006519250A (ja) | 2003-03-04 | 2006-08-24 | ファイザー・プロダクツ・インク | 医療処置におけるep2選択的受容体アゴニストの使用 |
US20050203086A1 (en) * | 2004-03-04 | 2005-09-15 | Pfizer Inc. | Methods of treatment using an EP2 selective receptor agonist |
US7915316B2 (en) * | 2005-08-22 | 2011-03-29 | Allergan, Inc | Sulfonamides |
US7696235B2 (en) * | 2005-08-29 | 2010-04-13 | Allergan, Inc. | EP2 receptor agonists for treating glaucoma |
-
2007
- 2007-07-16 CA CA2659184A patent/CA2659184C/en not_active Expired - Fee Related
- 2007-07-16 AP AP2009004754A patent/AP2009004754A0/xx unknown
- 2007-07-16 NZ NZ573964A patent/NZ573964A/en not_active IP Right Cessation
- 2007-07-16 RS RSP-2009/0002A patent/RS20090002A/sr unknown
- 2007-07-16 MX MX2009001062A patent/MX2009001062A/es active IP Right Grant
- 2007-07-16 EP EP07766635A patent/EP2059507B1/en not_active Not-in-force
- 2007-07-16 WO PCT/IB2007/002044 patent/WO2008015517A2/en active Application Filing
- 2007-07-16 KR KR1020097001522A patent/KR101088942B1/ko not_active IP Right Cessation
- 2007-07-16 BR BRPI0714683-3A patent/BRPI0714683A2/pt not_active IP Right Cessation
- 2007-07-16 JP JP2009522350A patent/JP4583500B2/ja not_active Expired - Fee Related
- 2007-07-16 AU AU2007280130A patent/AU2007280130B2/en not_active Ceased
- 2007-07-16 EA EA200970067A patent/EA200970067A1/ru unknown
- 2007-07-26 AR ARP070103330A patent/AR062122A1/es unknown
- 2007-07-26 PE PE2007000967A patent/PE20080408A1/es not_active Application Discontinuation
- 2007-07-27 CL CL200702207A patent/CL2007002207A1/es unknown
- 2007-07-27 UY UY30511A patent/UY30511A1/es not_active Application Discontinuation
- 2007-07-27 US US11/829,176 patent/US7622475B2/en not_active Expired - Fee Related
- 2007-07-27 GT GT200700064A patent/GT200700064A/es unknown
- 2007-07-27 TW TW096127590A patent/TWI372757B/zh not_active IP Right Cessation
-
2009
- 2009-01-05 IL IL196355A patent/IL196355A0/en unknown
- 2009-01-13 CR CR10554A patent/CR10554A/es not_active Application Discontinuation
- 2009-01-14 EC EC2009009071A patent/ECSP099071A/es unknown
- 2009-01-26 TN TN2009000028A patent/TN2009000028A1/fr unknown
- 2009-01-28 MA MA31593A patent/MA30604B1/fr unknown
- 2009-02-16 NO NO20090738A patent/NO20090738L/no not_active Application Discontinuation
- 2009-10-07 US US12/575,373 patent/US20100105905A1/en not_active Abandoned
- 2009-11-10 HK HK09110479.0A patent/HK1133876A1/xx not_active IP Right Cessation
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
109 | Application deemed to be withdrawn |
Effective date: 20170724 |