UY29366A1 - Derivados de la n-(4,5-difenil-2-tienil)metilamina, su preparacion y su aplicación en terapéutica - Google Patents

Derivados de la n-(4,5-difenil-2-tienil)metilamina, su preparacion y su aplicación en terapéutica

Info

Publication number
UY29366A1
UY29366A1 UY29366A UY29366A UY29366A1 UY 29366 A1 UY29366 A1 UY 29366A1 UY 29366 A UY29366 A UY 29366A UY 29366 A UY29366 A UY 29366A UY 29366 A1 UY29366 A1 UY 29366A1
Authority
UY
Uruguay
Prior art keywords
preparation
tienil
difenil
methylamine
therapeutics
Prior art date
Application number
UY29366A
Other languages
English (en)
Inventor
Barth Francis
Congy Christian
Rinaldi-Carmona Murielle
Ducoux Jean-Philippe
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of UY29366A1 publication Critical patent/UY29366A1/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
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    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
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  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Neurosurgery (AREA)
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  • Biomedical Technology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Addiction (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Hospice & Palliative Care (AREA)
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  • Pulmonology (AREA)
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  • Otolaryngology (AREA)

Abstract

La presente invención tiene por objeto compuestos que responden a la fórmulaque se menciona en el expediente: en la que: - X, R1, R2, R3, R4, R5, n y Alk son como se definieron en la memoria y reivindicaciones, procedimiento de preparación y aplicación en terapéutica.
UY29366A 2005-02-09 2006-02-08 Derivados de la n-(4,5-difenil-2-tienil)metilamina, su preparacion y su aplicación en terapéutica UY29366A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0501366A FR2881744B1 (fr) 2005-02-09 2005-02-09 Derives de n-[(4,5-diphenyl-2-thienyl)methyl]amine, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
UY29366A1 true UY29366A1 (es) 2006-10-02

Family

ID=34955350

Family Applications (1)

Application Number Title Priority Date Filing Date
UY29366A UY29366A1 (es) 2005-02-09 2006-02-08 Derivados de la n-(4,5-difenil-2-tienil)metilamina, su preparacion y su aplicación en terapéutica

Country Status (16)

Country Link
US (2) US7687537B2 (es)
EP (1) EP1858872A1 (es)
JP (1) JP4823236B2 (es)
KR (1) KR20070115941A (es)
CN (1) CN101128451A (es)
AR (1) AR052898A1 (es)
AU (1) AU2006212162A1 (es)
BR (1) BRPI0606942A2 (es)
CA (1) CA2596613A1 (es)
FR (1) FR2881744B1 (es)
IL (1) IL185035A0 (es)
MX (1) MX2007009439A (es)
RU (1) RU2007133602A (es)
TW (1) TW200639160A (es)
UY (1) UY29366A1 (es)
WO (1) WO2006084975A1 (es)

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FR2881744B1 (fr) * 2005-02-09 2007-04-27 Sanofi Aventis Sa Derives de n-[(4,5-diphenyl-2-thienyl)methyl]amine, leur preparation et leur application en therapeutique
JP2008534504A (ja) 2005-03-22 2008-08-28 アゼヴァン ファーマスーティカルズ，インコーポレイテッド 月経前障害を治療するためのβラクタミルアルカン酸
FR2894579B1 (fr) * 2005-12-12 2008-01-18 Sanofi Aventis Sa Derives diaryltriazolmethylamine, leur preparation et leur application en therapeutique.
US20100016274A1 (en) * 2006-09-14 2010-01-21 Koppel Gary A Beta-lactam cannabinoid receptor modulators
FR2908766B1 (fr) * 2006-11-20 2009-01-09 Sanofi Aventis Sa Derives de pyrrole,leur preparation et leur utilisation en therapeutique.
EP1939181A1 (en) * 2006-12-27 2008-07-02 sanofi-aventis Heteroaryl-substituted carboxamides and use thereof for the stimulation of the expression of NO synthase
EP2190822B1 (en) * 2007-09-28 2014-12-31 Takeda Pharmaceutical Company Limited 5-membered heterocyclic compounds as proton pump inhibitors
WO2009041447A1 (ja) * 2007-09-28 2009-04-02 Takeda Pharmaceutical Company Limited ５員複素環化合物
FR2934594B1 (fr) * 2008-08-01 2010-09-10 Sanofi Aventis Derives de thiophene-2-carboxamide, leur preparation et leur application en therapeutique.
FR2943672B1 (fr) * 2009-03-27 2011-03-25 Sanofi Aventis Derives de 3-alcoxy-4,5-diarylthiophene-2-carboxamide,leur preparation et leur application en therapeutique.
US8609663B2 (en) * 2009-11-18 2013-12-17 University Of Massachusetts Compounds for modulating TLR2
CN107007596A (zh) 2010-07-01 2017-08-04 阿泽凡药物公司 用于治疗创伤后应激障碍的方法
PL3122743T3 (pl) 2014-03-28 2023-05-02 Azevan Pharmaceuticals, Inc. Kompozycje i sposoby leczenia chorób neurodegeneracyjnych
AU2018333051B2 (en) 2017-09-15 2024-03-21 Azevan Pharmaceuticals, Inc. Compositions and methods for treating brain injury
AU2020308862A1 (en) * 2019-06-28 2022-01-20 Research Triangle Institute Urea derivatives as CB1 allosteric modulators

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EP0055471A1 (en) 1980-12-29 1982-07-07 E.I. Du Pont De Nemours And Company Antiinflammatory 4,5-diaryl-alpha,alpha-bis(polyhalomethyl)-2-thiophenemethanamines
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FR2881744B1 (fr) * 2005-02-09 2007-04-27 Sanofi Aventis Sa Derives de n-[(4,5-diphenyl-2-thienyl)methyl]amine, leur preparation et leur application en therapeutique

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RU2007133602A (ru) 2009-03-20
CA2596613A1 (fr) 2006-08-17
JP4823236B2 (ja) 2011-11-24
US20080009543A1 (en) 2008-01-10
US20100137402A1 (en) 2010-06-03
WO2006084975A1 (fr) 2006-08-17
IL185035A0 (en) 2007-12-03
KR20070115941A (ko) 2007-12-06
CN101128451A (zh) 2008-02-20
EP1858872A1 (fr) 2007-11-28
JP2008530060A (ja) 2008-08-07
MX2007009439A (es) 2008-03-06
FR2881744A1 (fr) 2006-08-11
AU2006212162A1 (en) 2006-08-17
BRPI0606942A2 (pt) 2009-07-28
TW200639160A (en) 2006-11-16
US7687537B2 (en) 2010-03-30
FR2881744B1 (fr) 2007-04-27
AR052898A1 (es) 2007-04-11

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