UY29366A1 - Derivados de la n-(4,5-difenil-2-tienil)metilamina, su preparacion y su aplicación en terapéutica - Google Patents

Derivados de la n-(4,5-difenil-2-tienil)metilamina, su preparacion y su aplicación en terapéutica

Info

Publication number
UY29366A1
UY29366A1 UY29366A UY29366A UY29366A1 UY 29366 A1 UY29366 A1 UY 29366A1 UY 29366 A UY29366 A UY 29366A UY 29366 A UY29366 A UY 29366A UY 29366 A1 UY29366 A1 UY 29366A1
Authority
UY
Uruguay
Prior art keywords
preparation
tienil
difenil
methylamine
therapeutics
Prior art date
Application number
UY29366A
Other languages
English (en)
Inventor
Barth Francis
Congy Christian
Rinaldi-Carmona Murielle
Ducoux Jean-Philippe
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of UY29366A1 publication Critical patent/UY29366A1/es

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
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    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381—Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
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  • Biomedical Technology (AREA)
  • Diabetes (AREA)
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  • Addiction (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Obesity (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Reproductive Health (AREA)
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  • Child & Adolescent Psychology (AREA)

Abstract

La presente invención tiene por objeto compuestos que responden a la fórmulaque se menciona en el expediente: en la que: - X, R1, R2, R3, R4, R5, n y Alk son como se definieron en la memoria y reivindicaciones, procedimiento de preparación y aplicación en terapéutica.
UY29366A 2005-02-09 2006-02-08 Derivados de la n-(4,5-difenil-2-tienil)metilamina, su preparacion y su aplicación en terapéutica UY29366A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0501366A FR2881744B1 (fr) 2005-02-09 2005-02-09 Derives de n-[(4,5-diphenyl-2-thienyl)methyl]amine, leur preparation et leur application en therapeutique

Publications (1)

Publication Number Publication Date
UY29366A1 true UY29366A1 (es) 2006-10-02

Family

ID=34955350

Family Applications (1)

Application Number Title Priority Date Filing Date
UY29366A UY29366A1 (es) 2005-02-09 2006-02-08 Derivados de la n-(4,5-difenil-2-tienil)metilamina, su preparacion y su aplicación en terapéutica

Country Status (16)

Country Link
US (2) US7687537B2 (es)
EP (1) EP1858872A1 (es)
JP (1) JP4823236B2 (es)
KR (1) KR20070115941A (es)
CN (1) CN101128451A (es)
AR (1) AR052898A1 (es)
AU (1) AU2006212162A1 (es)
BR (1) BRPI0606942A2 (es)
CA (1) CA2596613A1 (es)
FR (1) FR2881744B1 (es)
IL (1) IL185035A0 (es)
MX (1) MX2007009439A (es)
RU (1) RU2007133602A (es)
TW (1) TW200639160A (es)
UY (1) UY29366A1 (es)
WO (1) WO2006084975A1 (es)

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FR2881744B1 (fr) * 2005-02-09 2007-04-27 Sanofi Aventis Sa Derives de n-[(4,5-diphenyl-2-thienyl)methyl]amine, leur preparation et leur application en therapeutique
CN104922117A (zh) 2005-03-22 2015-09-23 阿泽范药品公司 用于治疗月经前病症的β-内酰氨基链烷酸
FR2894579B1 (fr) * 2005-12-12 2008-01-18 Sanofi Aventis Sa Derives diaryltriazolmethylamine, leur preparation et leur application en therapeutique.
US20100016274A1 (en) * 2006-09-14 2010-01-21 Koppel Gary A Beta-lactam cannabinoid receptor modulators
FR2908766B1 (fr) * 2006-11-20 2009-01-09 Sanofi Aventis Sa Derives de pyrrole,leur preparation et leur utilisation en therapeutique.
EP1939181A1 (en) 2006-12-27 2008-07-02 sanofi-aventis Heteroaryl-substituted carboxamides and use thereof for the stimulation of the expression of NO synthase
CL2008002834A1 (es) * 2007-09-28 2009-09-11 Takeda Pharmaceuticals Co Compuestos heterociclicos de 5 miembros, composicion farmaceutica, util para el tratamiento de la ulcera peptidica, sindrome de zollinger-ellison, gastritis, esofagitis por reflujo, enfermedad sintomatica por reflujo gastroesofagico, esofago de barrett, cancer gastrico, hiperacidez gastrica o ulcera debido a estres posquirurgico.
KR101559597B1 (ko) * 2007-09-28 2015-10-12 다케다 야쿠힌 고교 가부시키가이샤 ５―원 헤테로시클릭 화합물
FR2934594B1 (fr) * 2008-08-01 2010-09-10 Sanofi Aventis Derives de thiophene-2-carboxamide, leur preparation et leur application en therapeutique.
FR2943672B1 (fr) * 2009-03-27 2011-03-25 Sanofi Aventis Derives de 3-alcoxy-4,5-diarylthiophene-2-carboxamide,leur preparation et leur application en therapeutique.
US8609663B2 (en) 2009-11-18 2013-12-17 University Of Massachusetts Compounds for modulating TLR2
US9376424B2 (en) 2010-07-01 2016-06-28 Azevan Pharmaceuticals, Inc. Methods for treating post traumatic stress disorder
FI3122743T3 (fi) 2014-03-28 2023-03-02 Azevan Pharmaceuticals Inc Koostumuksia ja menetelmiä hermostoa rappeuttavien sairauksien hoitamiseksi
JP2020534274A (ja) 2017-09-15 2020-11-26 アゼヴァン ファーマシューティカルズ，インコーポレイテッド 脳損傷を治療するための組成物及び方法
WO2020264176A1 (en) * 2019-06-28 2020-12-30 Rti International Urea derivatives as cb1 allosteric modulators

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FR2881744B1 (fr) * 2005-02-09 2007-04-27 Sanofi Aventis Sa Derives de n-[(4,5-diphenyl-2-thienyl)methyl]amine, leur preparation et leur application en therapeutique

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US7687537B2 (en) 2010-03-30
AR052898A1 (es) 2007-04-11
IL185035A0 (en) 2007-12-03
FR2881744A1 (fr) 2006-08-11
JP2008530060A (ja) 2008-08-07
JP4823236B2 (ja) 2011-11-24
US20080009543A1 (en) 2008-01-10
KR20070115941A (ko) 2007-12-06
FR2881744B1 (fr) 2007-04-27
RU2007133602A (ru) 2009-03-20
TW200639160A (en) 2006-11-16
WO2006084975A1 (fr) 2006-08-17
US20100137402A1 (en) 2010-06-03
AU2006212162A1 (en) 2006-08-17
MX2007009439A (es) 2008-03-06
EP1858872A1 (fr) 2007-11-28
CN101128451A (zh) 2008-02-20
BRPI0606942A2 (pt) 2009-07-28
CA2596613A1 (fr) 2006-08-17

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