UY28730A1 - Procedimiento mejorado para la preparacion de un derivado de 2-(etoximetil)-tropano - Google Patents

Procedimiento mejorado para la preparacion de un derivado de 2-(etoximetil)-tropano

Info

Publication number
UY28730A1
UY28730A1 UY28730A UY28730A UY28730A1 UY 28730 A1 UY28730 A1 UY 28730A1 UY 28730 A UY28730 A UY 28730A UY 28730 A UY28730 A UY 28730A UY 28730 A1 UY28730 A1 UY 28730A1
Authority
UY
Uruguay
Prior art keywords
preparation
etoximethyl
tropane
derivative
improved procedure
Prior art date
Application number
UY28730A
Other languages
English (en)
Spanish (es)
Inventor
Dr Richard Ehlenz
Dr Oliver Meyer
Sascha Wagner
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of UY28730A1 publication Critical patent/UY28730A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Psychology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
UY28730A 2004-01-31 2005-01-28 Procedimiento mejorado para la preparacion de un derivado de 2-(etoximetil)-tropano UY28730A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE102004004965A DE102004004965B4 (de) 2004-01-31 2004-01-31 Verfahren zur Herstellung eines 2-(Ethoxymethyl)-tropanderivates

Publications (1)

Publication Number Publication Date
UY28730A1 true UY28730A1 (es) 2005-09-30

Family

ID=34801391

Family Applications (1)

Application Number Title Priority Date Filing Date
UY28730A UY28730A1 (es) 2004-01-31 2005-01-28 Procedimiento mejorado para la preparacion de un derivado de 2-(etoximetil)-tropano

Country Status (16)

Country Link
US (1) US7544802B2 (https=)
EP (1) EP1713800B1 (https=)
JP (1) JP2007519660A (https=)
CN (1) CN1910180B (https=)
AR (1) AR047515A1 (https=)
AT (1) ATE449095T1 (https=)
AU (1) AU2005209382B2 (https=)
CA (1) CA2554125A1 (https=)
DE (2) DE102004004965B4 (https=)
DK (1) DK1713800T3 (https=)
MY (1) MY141935A (https=)
NZ (1) NZ548092A (https=)
PE (1) PE20050770A1 (https=)
TW (1) TWI338690B (https=)
UY (1) UY28730A1 (https=)
WO (1) WO2005073228A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX381130B (es) 2016-09-07 2025-03-12 Saniona As Composiciones de tesofensina.
CN115572289A (zh) * 2022-10-24 2023-01-06 龙曦宁(上海)医药科技有限公司 一种特索芬辛的合成方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3238414B2 (ja) * 1996-02-22 2001-12-17 ニューロサーチ・アクティーゼルスカブ トロパン―誘導体、その製造方法及びその使用方法
JP2005508872A (ja) * 2001-05-23 2005-04-07 ニューロサーチ、アクティーゼルスカブ トロパン誘導体及びこれをモノアミン神経伝達物質再取り込み阻害剤として使用する方法
US7381733B2 (en) * 2001-11-30 2008-06-03 Neurosearch A/S Tropane derivatives having dopamine reuptake inhibitor activity for the treatment of ischemic diseases
WO2021028011A1 (en) 2019-08-09 2021-02-18 Quintus Technologies Ab System and method for handling and isostatic pressure treatment of a load

Also Published As

Publication number Publication date
NZ548092A (en) 2009-07-31
HK1097845A1 (zh) 2007-07-06
TW200538455A (en) 2005-12-01
PE20050770A1 (es) 2005-11-10
AR047515A1 (es) 2006-01-25
US7544802B2 (en) 2009-06-09
JP2007519660A (ja) 2007-07-19
ATE449095T1 (de) 2009-12-15
WO2005073228A1 (de) 2005-08-11
CN1910180B (zh) 2010-05-12
US20050171145A1 (en) 2005-08-04
CN1910180A (zh) 2007-02-07
CA2554125A1 (en) 2005-08-11
MY141935A (en) 2010-07-30
TWI338690B (en) 2011-03-11
DE102004004965A1 (de) 2005-09-01
AU2005209382B2 (en) 2011-02-17
WO2005073228A8 (de) 2005-10-27
EP1713800B1 (de) 2009-11-18
DE102004004965B4 (de) 2006-01-05
DK1713800T3 (da) 2010-03-29
EP1713800A2 (de) 2006-10-25
DE502005008535D1 (de) 2009-12-31
AU2005209382A1 (en) 2005-08-11

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20160419