UA93868C2 - Лекарственное средство для перорального введения, kotopoe содержит ингибитор циклооксигеназы-2, и способ его получения - Google Patents
Лекарственное средство для перорального введения, kotopoe содержит ингибитор циклооксигеназы-2, и способ его полученияInfo
- Publication number
- UA93868C2 UA93868C2 UAA200709319A UAA200709319A UA93868C2 UA 93868 C2 UA93868 C2 UA 93868C2 UA A200709319 A UAA200709319 A UA A200709319A UA A200709319 A UAA200709319 A UA A200709319A UA 93868 C2 UA93868 C2 UA 93868C2
- Authority
- UA
- Ukraine
- Prior art keywords
- agglomerate
- inhibitor
- medicament
- cyclooxygenase
- preparation
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/417—Imidazole-alkylamines, e.g. histamine, phentolamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Изобретение касается лекарственного средства, предназначенного для перорального введения, которое содержит ингибитор циклооксигеназы-2 и имеет повышенную биодоступность, а также способа получения такого лекарственного средства.Лекарственное средство по изобретению содержит агломерат на базе инертных твердых частиц, состав которых базируется как минимум на одном вспомогательном веществе, причем указанный агломерат содержит ингибитор циклооксигеназы-2 и как минимум один гидрофильный полимер.Согласно изобретению, агломерат содержит аэрозоль, нанесенный �
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR0500708A FR2881049B1 (fr) | 2005-01-24 | 2005-01-24 | Medicament destine a etre administre par voie orale comprenant un inhibiteur de la cyclo-oxygenase-2, et son procede de preparation |
Publications (1)
Publication Number | Publication Date |
---|---|
UA93868C2 true UA93868C2 (ru) | 2011-03-25 |
Family
ID=34954944
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UAA200709319A UA93868C2 (ru) | 2005-01-24 | 2006-01-23 | Лекарственное средство для перорального введения, kotopoe содержит ингибитор циклооксигеназы-2, и способ его получения |
Country Status (17)
Country | Link |
---|---|
US (1) | US20080213376A1 (ru) |
EP (1) | EP1845959B1 (ru) |
JP (1) | JP5106119B2 (ru) |
KR (2) | KR20080007543A (ru) |
CN (1) | CN101119712B (ru) |
AU (1) | AU2006207396B2 (ru) |
BR (1) | BRPI0607372B8 (ru) |
CA (1) | CA2595496C (ru) |
FR (1) | FR2881049B1 (ru) |
IL (1) | IL184759A (ru) |
MX (1) | MX2007008878A (ru) |
NZ (1) | NZ556707A (ru) |
PL (1) | PL1845959T3 (ru) |
RU (1) | RU2391099C2 (ru) |
UA (1) | UA93868C2 (ru) |
WO (1) | WO2006077334A2 (ru) |
ZA (1) | ZA200705996B (ru) |
Family Cites Families (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU670567B2 (en) * | 1992-03-05 | 1996-07-25 | American Home Products Corporation | Pharmaceutical coated cores |
AR024222A1 (es) * | 1998-10-16 | 2002-09-25 | Palau Pharma Sa | Imidazoles con actividad antiinflamatoria un procedimiento para su preparacion y composiciones farmaceuticas que lo contienen |
BR0008058A (pt) * | 1999-12-08 | 2002-03-26 | Pharmacia Corp | Forma de estado sólido de celecoxib tendo biodisposnibilidade melhorada |
EP1239857B1 (en) * | 1999-12-22 | 2006-04-19 | Pharmacia Corporation | Dual-release compositions of a cyclooxygenase-2- inhibitor |
CA2394222A1 (en) * | 1999-12-22 | 2001-06-28 | Pharmacia Corporation | Sustained-release formulation of a cyclooxygenase-2 inhibitor |
EP1330239A2 (en) * | 2000-10-26 | 2003-07-30 | MEHTA, Atul M. | Delayed and sustained release formulations and method of use thereof |
-
2005
- 2005-01-24 FR FR0500708A patent/FR2881049B1/fr not_active Expired - Fee Related
-
2006
- 2006-01-23 WO PCT/FR2006/000144 patent/WO2006077334A2/fr active Application Filing
- 2006-01-23 EP EP06709146.2A patent/EP1845959B1/fr active Active
- 2006-01-23 RU RU2007132017/15A patent/RU2391099C2/ru active
- 2006-01-23 KR KR1020077019460A patent/KR20080007543A/ko not_active Application Discontinuation
- 2006-01-23 KR KR1020137028765A patent/KR20130128019A/ko not_active Application Discontinuation
- 2006-01-23 BR BRPI0607372A patent/BRPI0607372B8/pt not_active IP Right Cessation
- 2006-01-23 UA UAA200709319A patent/UA93868C2/ru unknown
- 2006-01-23 CA CA2595496A patent/CA2595496C/fr not_active Expired - Fee Related
- 2006-01-23 AU AU2006207396A patent/AU2006207396B2/en not_active Ceased
- 2006-01-23 JP JP2007551709A patent/JP5106119B2/ja active Active
- 2006-01-23 PL PL06709146T patent/PL1845959T3/pl unknown
- 2006-01-23 CN CN2006800050019A patent/CN101119712B/zh not_active Expired - Fee Related
- 2006-01-23 MX MX2007008878A patent/MX2007008878A/es active IP Right Grant
- 2006-01-23 NZ NZ556707A patent/NZ556707A/en not_active IP Right Cessation
- 2006-01-23 US US11/814,626 patent/US20080213376A1/en not_active Abandoned
-
2007
- 2007-07-17 ZA ZA200705996A patent/ZA200705996B/xx unknown
- 2007-07-22 IL IL184759A patent/IL184759A/en not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
CA2595496C (fr) | 2014-06-03 |
RU2391099C2 (ru) | 2010-06-10 |
KR20080007543A (ko) | 2008-01-22 |
MX2007008878A (es) | 2007-10-11 |
ZA200705996B (en) | 2009-03-25 |
BRPI0607372B1 (pt) | 2019-04-30 |
BRPI0607372A2 (pt) | 2009-09-01 |
CN101119712A (zh) | 2008-02-06 |
RU2007132017A (ru) | 2009-02-27 |
WO2006077334A3 (fr) | 2007-04-12 |
FR2881049A1 (fr) | 2006-07-28 |
WO2006077334A2 (fr) | 2006-07-27 |
IL184759A (en) | 2012-10-31 |
BRPI0607372B8 (pt) | 2021-05-25 |
EP1845959B1 (fr) | 2015-04-15 |
AU2006207396B2 (en) | 2011-05-19 |
JP5106119B2 (ja) | 2012-12-26 |
CN101119712B (zh) | 2013-05-01 |
EP1845959A2 (fr) | 2007-10-24 |
KR20130128019A (ko) | 2013-11-25 |
JP2008528462A (ja) | 2008-07-31 |
US20080213376A1 (en) | 2008-09-04 |
AU2006207396A1 (en) | 2006-07-27 |
CA2595496A1 (fr) | 2006-07-27 |
PL1845959T3 (pl) | 2015-10-30 |
IL184759A0 (en) | 2007-12-03 |
FR2881049B1 (fr) | 2008-12-26 |
NZ556707A (en) | 2010-05-28 |
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