UA88509C2 - Сублингвальная таблетка с покрытием, которое содержит опиоидный анальгетик - Google Patents

Сублингвальная таблетка с покрытием, которое содержит опиоидный анальгетик

Info

Publication number
UA88509C2
UA88509C2 UAA200710340A UAA200710340A UA88509C2 UA 88509 C2 UA88509 C2 UA 88509C2 UA A200710340 A UAA200710340 A UA A200710340A UA A200710340 A UAA200710340 A UA A200710340A UA 88509 C2 UA88509 C2 UA 88509C2
Authority
UA
Ukraine
Prior art keywords
opioid analgesic
coated tablet
sublingual coated
active substance
sublingual
Prior art date
Application number
UAA200710340A
Other languages
English (en)
Ukrainian (uk)
Inventor
Паскаль Ури
Гием Бенуа
Катрин Эрри
Йозеф Дювошель
Original Assignee
Этифарм
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Этифарм filed Critical Этифарм
Publication of UA88509C2 publication Critical patent/UA88509C2/ru

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/485—Morphinan derivatives, e.g. morphine, codeine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Zoology (AREA)
  • Emergency Medicine (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Oncology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Formation And Processing Of Food Products (AREA)

Abstract

Изобретение касается сублингвальной таблетки с покрытием, которая содержит сердцевину, свободную от фармацевтически активного вещества, содержащую один или более разбавителей, и покрытие, которое содержит, по меньшей мере, один опиоидный анальгетик, пригодный для сублингвального введения. Изобретение также касается способа получения такой таблетки и ее применения для лечения боли.
UAA200710340A 2005-03-18 2006-03-20 Сублингвальная таблетка с покрытием, которое содержит опиоидный анальгетик UA88509C2 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR0502727A FR2883179B1 (fr) 2005-03-18 2005-03-18 Comprime enrobe

Publications (1)

Publication Number Publication Date
UA88509C2 true UA88509C2 (ru) 2009-10-26

Family

ID=35309611

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA200710340A UA88509C2 (ru) 2005-03-18 2006-03-20 Сублингвальная таблетка с покрытием, которое содержит опиоидный анальгетик

Country Status (26)

Country Link
US (2) US20080226717A1 (ru)
EP (1) EP1858491B1 (ru)
JP (1) JP5138577B2 (ru)
KR (1) KR101239926B1 (ru)
CN (1) CN101141951B (ru)
AT (1) ATE507824T1 (ru)
AU (1) AU2006224690B2 (ru)
BR (1) BRPI0608505B8 (ru)
CA (1) CA2599502C (ru)
CY (1) CY1111729T1 (ru)
DE (1) DE602006021713D1 (ru)
DK (1) DK1858491T3 (ru)
ES (1) ES2365984T3 (ru)
FR (1) FR2883179B1 (ru)
HK (1) HK1109730A1 (ru)
IL (1) IL185626A (ru)
MX (1) MX2007011440A (ru)
NO (1) NO338771B1 (ru)
NZ (1) NZ561154A (ru)
PL (1) PL1858491T3 (ru)
PT (1) PT1858491E (ru)
RU (1) RU2403043C2 (ru)
SI (1) SI1858491T1 (ru)
UA (1) UA88509C2 (ru)
WO (1) WO2006097361A1 (ru)
ZA (1) ZA200707900B (ru)

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US8202535B2 (en) 2006-01-06 2012-06-19 Acelrx Pharmaceuticals, Inc. Small-volume oral transmucosal dosage forms
US8252328B2 (en) 2006-01-06 2012-08-28 Acelrx Pharmaceuticals, Inc. Bioadhesive drug formulations for oral transmucosal delivery
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Also Published As

Publication number Publication date
CY1111729T1 (el) 2015-10-07
EP1858491A1 (en) 2007-11-28
EP1858491B1 (en) 2011-05-04
NO20075345L (no) 2007-12-17
BRPI0608505B8 (pt) 2021-05-25
CA2599502A1 (en) 2006-09-21
NO338771B1 (no) 2016-10-17
CA2599502C (en) 2013-05-14
CN101141951A (zh) 2008-03-12
IL185626A0 (en) 2008-01-06
JP5138577B2 (ja) 2013-02-06
RU2007138647A (ru) 2009-04-27
KR20070114756A (ko) 2007-12-04
KR101239926B1 (ko) 2013-03-07
RU2403043C2 (ru) 2010-11-10
CN101141951B (zh) 2011-02-09
WO2006097361A1 (en) 2006-09-21
BRPI0608505B1 (pt) 2021-05-04
ATE507824T1 (de) 2011-05-15
HK1109730A1 (en) 2008-06-20
BRPI0608505A2 (pt) 2010-01-05
US20080226717A1 (en) 2008-09-18
DE602006021713D1 (de) 2011-06-16
MX2007011440A (es) 2007-11-14
ZA200707900B (en) 2009-01-28
AU2006224690A1 (en) 2006-09-21
ES2365984T3 (es) 2011-10-14
IL185626A (en) 2014-09-30
PT1858491E (pt) 2011-08-18
NZ561154A (en) 2010-12-24
US20060210632A1 (en) 2006-09-21
AU2006224690B2 (en) 2011-09-29
SI1858491T1 (sl) 2011-09-30
FR2883179A1 (fr) 2006-09-22
PL1858491T3 (pl) 2012-03-30
FR2883179B1 (fr) 2009-04-17
US8709479B2 (en) 2014-04-29
DK1858491T3 (da) 2011-08-22
JP2008533084A (ja) 2008-08-21

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