UA79073C2 - 8- hydrocarbyl-substituted estratrienes for use as selective estrogens, pharmaceutical composition based thereon - Google Patents
8- hydrocarbyl-substituted estratrienes for use as selective estrogens, pharmaceutical composition based thereon Download PDFInfo
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- UA79073C2 UA79073C2 UA2002118922A UA2002118922A UA79073C2 UA 79073 C2 UA79073 C2 UA 79073C2 UA 2002118922 A UA2002118922 A UA 2002118922A UA 2002118922 A UA2002118922 A UA 2002118922A UA 79073 C2 UA79073 C2 UA 79073C2
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- hydrogen atom
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- diol
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
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- C07J1/0074—Esters
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- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0072—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic
Landscapes
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- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
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- Endocrinology (AREA)
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- Neurosurgery (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Rheumatology (AREA)
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- Immunology (AREA)
- Hematology (AREA)
- Toxicology (AREA)
- Steroid Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE10019167A DE10019167A1 (de) | 2000-04-12 | 2000-04-12 | Substituierte Estratriene als selektiv wirksame Estrogene |
PCT/EP2001/004290 WO2001077139A1 (de) | 2000-04-12 | 2001-04-12 | 8.beta.-hydrocarbyl-substituierte estratriene als selektiv wirksame estrogene |
Publications (1)
Publication Number | Publication Date |
---|---|
UA79073C2 true UA79073C2 (en) | 2007-05-25 |
Family
ID=7639163
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
UA2002118922A UA79073C2 (en) | 2000-04-12 | 2001-12-04 | 8- hydrocarbyl-substituted estratrienes for use as selective estrogens, pharmaceutical composition based thereon |
Country Status (11)
Country | Link |
---|---|
JP (1) | JP4860880B2 (zh) |
KR (1) | KR100825534B1 (zh) |
AR (1) | AR028329A1 (zh) |
DE (2) | DE10019167A1 (zh) |
PE (1) | PE20011215A1 (zh) |
SI (1) | SI1272504T1 (zh) |
TW (1) | TWI288138B (zh) |
UA (1) | UA79073C2 (zh) |
UY (1) | UY26665A1 (zh) |
YU (1) | YU77302A (zh) |
ZA (1) | ZA200209149B (zh) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK1272504T3 (da) * | 2000-04-12 | 2007-10-01 | Bayer Schering Pharma Ag | 8.Beta-hydrocarbylsubstituerede östradiener til anvendelse som selektive östrogener |
DE10151114A1 (de) * | 2001-10-15 | 2003-04-17 | Schering Ag | 8ß-Substituierte-11ß-aryl-estra-2,3,5(10)-trienderivate |
JP2007512279A (ja) * | 2003-11-26 | 2007-05-17 | シエーリング アクチエンゲゼルシャフト | 選択的エストロゲン8β−ビニル−エストラ−1,3,5(10)−トリエン−3,17β−ジオール、及び17β−フルオル−9α−ビニル−エストラ−1,3,5(10)−トリエン−3,16α−ジオールによる高血圧性心疾患の予防及び治療 |
WO2008064133A1 (en) * | 2006-11-17 | 2008-05-29 | Trustees Of Dartmouth College | Synthesis and biological activities of new tricyclic-bis-enones (tbes) |
EP2014672A1 (en) * | 2007-07-12 | 2009-01-14 | Bayer Schering Pharma Aktiengesellschaft | 8-beta-substituted estratrienes as selectively active estrogens |
JP2012509286A (ja) * | 2008-11-21 | 2012-04-19 | バイエル ファーマ アクチエンゲゼルシャフト | 薬物送達システム |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3681407A (en) | 1969-06-18 | 1972-08-01 | American Cyanamid Co | 3-methoxy 8{62 -methylestra 1,3,5(10),9(11)-tetraene-17{62 -carboxylic acid lower alkyl ester and intermediates in the preparation thereof |
US3806546A (en) | 1969-06-18 | 1974-04-23 | American Cyanamid Co | Steroid-like compounds and method of synthesis |
US3736345A (en) | 1971-05-18 | 1973-05-29 | American Cyanamid Co | Steroid-like compounds and method of synthesis |
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2000
- 2000-04-12 DE DE10019167A patent/DE10019167A1/de not_active Withdrawn
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2001
- 2001-04-11 PE PE2001000335A patent/PE20011215A1/es not_active Application Discontinuation
- 2001-04-11 UY UY26665A patent/UY26665A1/es not_active Application Discontinuation
- 2001-04-11 AR ARP010101730A patent/AR028329A1/es active IP Right Grant
- 2001-04-12 KR KR1020027013665A patent/KR100825534B1/ko not_active IP Right Cessation
- 2001-04-12 JP JP2001575609A patent/JP4860880B2/ja not_active Expired - Fee Related
- 2001-04-12 TW TW090108786A patent/TWI288138B/zh not_active IP Right Cessation
- 2001-04-12 YU YU77302A patent/YU77302A/sh unknown
- 2001-04-12 DE DE50107204T patent/DE50107204D1/de not_active Expired - Fee Related
- 2001-04-12 SI SI200130752T patent/SI1272504T1/sl unknown
- 2001-12-04 UA UA2002118922A patent/UA79073C2/uk unknown
-
2002
- 2002-11-11 ZA ZA200209149A patent/ZA200209149B/en unknown
Also Published As
Publication number | Publication date |
---|---|
YU77302A (sh) | 2005-11-28 |
KR100825534B1 (ko) | 2008-04-25 |
UY26665A1 (es) | 2001-11-30 |
PE20011215A1 (es) | 2001-11-29 |
ZA200209149B (en) | 2007-10-31 |
AR028329A1 (es) | 2003-05-07 |
DE50107204D1 (de) | 2005-09-29 |
JP4860880B2 (ja) | 2012-01-25 |
KR20030028734A (ko) | 2003-04-10 |
TWI288138B (en) | 2007-10-11 |
SI1272504T1 (sl) | 2007-10-31 |
DE10019167A1 (de) | 2001-10-18 |
JP2003534248A (ja) | 2003-11-18 |
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