TWI673049B - 治療及/或預防纖維性疾病之胺基萘醌化合物 - Google Patents

治療及/或預防纖維性疾病之胺基萘醌化合物 Download PDF

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TWI673049B
TWI673049B TW105137577A TW105137577A TWI673049B TW I673049 B TWI673049 B TW I673049B TW 105137577 A TW105137577 A TW 105137577A TW 105137577 A TW105137577 A TW 105137577A TW I673049 B TWI673049 B TW I673049B
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methyl
dioxo
chloro
dihydronaphthalen
alkyl
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TW105137577A
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TW201720433A (zh
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雲 閻
劉景平
林建煌
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臺北醫學大學
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    • A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
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TW105137577A 2015-11-17 2016-11-17 治療及/或預防纖維性疾病之胺基萘醌化合物 TWI673049B (zh)

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Kai Xu et al,"Design and synthesis of naphthoquinone derivatives as antiproliferative agents and 20S proteasome inhibitors", Bioorganic & Medicinal Chemistry Letters, Vol 22(8), 15 April 2012, pages 2772-2774. Pingaew R et al,"Novel 1,4-naphthoquinone-based sulfonamides: Synthesis, QSAR, anticancer and antimalarial studies", Eur J Med Chem., Vol 22(8), 5 Sep 2015. *
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