TWI665192B - 製備二氫異唑衍生物之方法 - Google Patents

製備二氫異唑衍生物之方法 Download PDF

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Publication number
TWI665192B
TWI665192B TW104116745A TW104116745A TWI665192B TW I665192 B TWI665192 B TW I665192B TW 104116745 A TW104116745 A TW 104116745A TW 104116745 A TW104116745 A TW 104116745A TW I665192 B TWI665192 B TW I665192B
Authority
TW
Taiwan
Prior art keywords
formula
chlorine
acid
mixture
sodium
Prior art date
Application number
TW104116745A
Other languages
English (en)
Chinese (zh)
Other versions
TW201625567A (zh
Inventor
Guenter Hoemberger
岡特 漢伯格
Mark James Ford
馬克詹姆斯 弗德
Andreas Huegel
安德列斯 胡格爾
Tomoki Tsuchiya
土屋知己
Original Assignee
Bayer Cropscience Aktiengesellschaft
德商拜耳作物科學股份有限公司
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Aktiengesellschaft, 德商拜耳作物科學股份有限公司 filed Critical Bayer Cropscience Aktiengesellschaft
Publication of TW201625567A publication Critical patent/TW201625567A/zh
Application granted granted Critical
Publication of TWI665192B publication Critical patent/TWI665192B/zh

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
TW104116745A 2014-05-28 2015-05-26 製備二氫異唑衍生物之方法 TWI665192B (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
??14170155.7 2014-05-28
EP14170155 2014-05-28

Publications (2)

Publication Number Publication Date
TW201625567A TW201625567A (zh) 2016-07-16
TWI665192B true TWI665192B (zh) 2019-07-11

Family

ID=50828731

Family Applications (1)

Application Number Title Priority Date Filing Date
TW104116745A TWI665192B (zh) 2014-05-28 2015-05-26 製備二氫異唑衍生物之方法

Country Status (12)

Country Link
US (1) US9796690B2 (enExample)
EP (1) EP3148976B1 (enExample)
JP (1) JP6533798B2 (enExample)
KR (1) KR102337028B1 (enExample)
CN (1) CN106414417B (enExample)
BR (1) BR112016027824B1 (enExample)
DK (1) DK3148976T3 (enExample)
ES (1) ES2730048T3 (enExample)
IL (1) IL248568B (enExample)
MX (1) MX382631B (enExample)
TW (1) TWI665192B (enExample)
WO (1) WO2015181189A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX389099B (es) * 2015-03-05 2025-03-20 Bayer Cropscience Ag Proceso para la preparación de 3-cloro-2-vinilfenilsulfonatos.
ES2848200T3 (es) * 2016-12-05 2021-08-05 Bayer Cropscience Ag Procedimiento para la preparación de 2-vinilfenilsulfonatos 3-sustituidos
CN113891882B (zh) * 2019-06-14 2024-11-26 组合化学工业株式会社 二氢异噁唑的制造方法

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW201341382A (zh) * 2011-12-27 2013-10-16 拜耳智慧財產有限公司 作為殺真菌劑之雜芳基哌啶及哌□衍生物

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
OA09122A (en) 1988-07-08 1991-10-31 Schering Agrochemicals Ltd Triazole insecticides.
DE4331448A1 (de) 1993-09-16 1995-03-23 Hoechst Schering Agrevo Gmbh Substituierte Isoxazoline, Verfahren zu deren Herstellung, diese enthaltende Mittel und deren Verwendung als Safener
EP1878730A1 (en) 2006-07-12 2008-01-16 Bayer Schering Pharma Aktiengesellschaft Substituted isoxazolines, pharmaceutical compositions containing the same, methods of preparing the same, and uses of the same
WO2008013622A2 (en) * 2006-07-27 2008-01-31 E. I. Du Pont De Nemours And Company Fungicidal azocyclic amides
JP5529044B2 (ja) * 2008-01-25 2014-06-25 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー 殺菌性複素環化合物
WO2009094407A2 (en) * 2008-01-25 2009-07-30 E. I. Du Pont De Nemours And Company Fungicidal amides
CN102215820A (zh) 2008-11-17 2011-10-12 安龙制药公司 用于核酸输送系统的可释放融合脂质
ES2534516T3 (es) * 2010-01-07 2015-04-23 E.I. Du Pont De Nemours And Company Compuestos heterocíclicos fungicidas
IN2012DE00621A (enExample) * 2012-03-02 2015-07-17 Syngenta Participations Ag

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW201341382A (zh) * 2011-12-27 2013-10-16 拜耳智慧財產有限公司 作為殺真菌劑之雜芳基哌啶及哌□衍生物

Also Published As

Publication number Publication date
JP2017517513A (ja) 2017-06-29
US9796690B2 (en) 2017-10-24
CN106414417B (zh) 2019-04-16
BR112016027824B1 (pt) 2021-03-23
TW201625567A (zh) 2016-07-16
EP3148976A1 (en) 2017-04-05
EP3148976B1 (en) 2019-03-13
IL248568A0 (en) 2016-12-29
IL248568B (en) 2019-03-31
US20170247345A1 (en) 2017-08-31
KR20170012331A (ko) 2017-02-02
KR102337028B1 (ko) 2021-12-07
JP6533798B2 (ja) 2019-06-19
DK3148976T3 (da) 2019-05-27
ES2730048T3 (es) 2019-11-07
MX382631B (es) 2025-03-13
CN106414417A (zh) 2017-02-15
WO2015181189A1 (en) 2015-12-03
MX2016015623A (es) 2017-02-27

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