TWI433838B - 作為趨化因子受體活性調節劑之六氫吡啶衍生物 - Google Patents
作為趨化因子受體活性調節劑之六氫吡啶衍生物 Download PDFInfo
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US7539408P | 2008-06-25 | 2008-06-25 | |
| US12/490,477 US8299098B2 (en) | 2008-06-25 | 2009-06-24 | Piperidinyl derivative as a modulator of chemokine receptor activity |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| TW201004927A TW201004927A (en) | 2010-02-01 |
| TWI433838B true TWI433838B (zh) | 2014-04-11 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| TW098120298A TWI433838B (zh) | 2008-06-25 | 2009-06-17 | 作為趨化因子受體活性調節劑之六氫吡啶衍生物 |
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| EP (1) | EP2323983B1 (enExample) |
| JP (1) | JP5357965B2 (enExample) |
| KR (1) | KR20110023865A (enExample) |
| CN (1) | CN102076663B (enExample) |
| AU (1) | AU2009262219B2 (enExample) |
| BR (1) | BRPI0914539A2 (enExample) |
| CA (1) | CA2729016A1 (enExample) |
| CL (1) | CL2010001566A1 (enExample) |
| CO (1) | CO6321247A2 (enExample) |
| CY (1) | CY1114994T1 (enExample) |
| DK (1) | DK2323983T3 (enExample) |
| EA (1) | EA021224B1 (enExample) |
| ES (1) | ES2447740T3 (enExample) |
| HR (1) | HRP20140071T1 (enExample) |
| IL (1) | IL209832A (enExample) |
| MX (1) | MX2010013664A (enExample) |
| NZ (1) | NZ589909A (enExample) |
| PE (1) | PE20110103A1 (enExample) |
| PL (1) | PL2323983T3 (enExample) |
| PT (1) | PT2323983E (enExample) |
| SI (1) | SI2323983T1 (enExample) |
| TW (1) | TWI433838B (enExample) |
| WO (1) | WO2009158452A1 (enExample) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI433838B (zh) * | 2008-06-25 | 2014-04-11 | 必治妥美雅史谷比公司 | 作為趨化因子受體活性調節劑之六氫吡啶衍生物 |
| US8410139B2 (en) * | 2009-10-07 | 2013-04-02 | Bristol-Myers Squibb Company | Prodrugs of a piperidinyl derivative as modulators of chemokine receptor activity |
| WO2011044197A1 (en) * | 2009-10-07 | 2011-04-14 | Bristol-Myers Squibb Company | Spirocyclic compounds as modulators of chemokine receptor activity |
| US8642622B2 (en) | 2010-06-16 | 2014-02-04 | Bristol-Myers Squibb Company | Piperidinyl compound as a modulator of chemokine receptor activity |
| AR087277A1 (es) | 2011-07-21 | 2014-03-12 | Bristol Myers Squibb Co | Composiciones biodisponibles de compuestos amorfos de piperidinilo, composicion farmaceutica, metodos |
| US20150225790A1 (en) | 2012-04-25 | 2015-08-13 | Bristol-Myers Squibb Company | Methods for identifying subjects with an increased likelihood of responding to ccr1 antagonist |
| US9257178B1 (en) * | 2014-11-26 | 2016-02-09 | Taiwan Semiconductor Manufacturing Company Limited | Devices and methods for writing to a memory cell of a memory |
| EP3507830A4 (en) * | 2016-08-31 | 2020-04-01 | Micron Technology, Inc. | MEMORY CELLS AND MEMORY MATRICES |
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| CA2249601A1 (en) | 1996-04-03 | 1997-10-23 | Thorsten E. Fisher | Inhibitors of farnesyl-protein transferase |
| AU721035C (en) * | 1996-09-10 | 2004-09-02 | Dr. Karl Thomae Gmbh | Modified aminoacids, pharmaceuticals containing these compounds and method for their production |
| JP4024309B2 (ja) | 1996-10-22 | 2007-12-19 | 第一三共株式会社 | 新規な感染症治療薬 |
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| DE69925160T2 (de) | 1998-12-17 | 2006-02-16 | Wyeth | Arylpiperidin- und aryl-1,2,5,6-tetrahydropyridinamid-derivate mit 5ht1a rezeptor aktivität |
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| US7615556B2 (en) * | 2006-01-27 | 2009-11-10 | Bristol-Myers Squibb Company | Piperazinyl derivatives as modulators of chemokine receptor activity |
| JP5292400B2 (ja) | 2007-07-24 | 2013-09-18 | ブリストル−マイヤーズ スクイブ カンパニー | ケモカイン受容体活性のモジュレーターとしてのピペリジン誘導体 |
| EP2173713B1 (en) | 2007-07-24 | 2016-02-17 | Bristol-Myers Squibb Company | Piperidinyl derivatives as modulators of chemokine receptor activity |
| TWI433838B (zh) * | 2008-06-25 | 2014-04-11 | 必治妥美雅史谷比公司 | 作為趨化因子受體活性調節劑之六氫吡啶衍生物 |
| AR087277A1 (es) | 2011-07-21 | 2014-03-12 | Bristol Myers Squibb Co | Composiciones biodisponibles de compuestos amorfos de piperidinilo, composicion farmaceutica, metodos |
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2009
- 2009-06-17 TW TW098120298A patent/TWI433838B/zh not_active IP Right Cessation
- 2009-06-24 US US12/490,477 patent/US8299098B2/en active Active
- 2009-06-25 PL PL09770985T patent/PL2323983T3/pl unknown
- 2009-06-25 ES ES09770985.1T patent/ES2447740T3/es active Active
- 2009-06-25 JP JP2011516635A patent/JP5357965B2/ja not_active Expired - Fee Related
- 2009-06-25 DK DK09770985.1T patent/DK2323983T3/da active
- 2009-06-25 PE PE2010001176A patent/PE20110103A1/es not_active Application Discontinuation
- 2009-06-25 PT PT97709851T patent/PT2323983E/pt unknown
- 2009-06-25 CA CA2729016A patent/CA2729016A1/en not_active Abandoned
- 2009-06-25 HR HRP20140071AT patent/HRP20140071T1/hr unknown
- 2009-06-25 EA EA201100088A patent/EA021224B1/ru not_active IP Right Cessation
- 2009-06-25 MX MX2010013664A patent/MX2010013664A/es active IP Right Grant
- 2009-06-25 AU AU2009262219A patent/AU2009262219B2/en not_active Ceased
- 2009-06-25 NZ NZ589909A patent/NZ589909A/en not_active IP Right Cessation
- 2009-06-25 KR KR1020107029082A patent/KR20110023865A/ko not_active Withdrawn
- 2009-06-25 SI SI200930827T patent/SI2323983T1/sl unknown
- 2009-06-25 CN CN2009801245643A patent/CN102076663B/zh not_active Expired - Fee Related
- 2009-06-25 BR BRPI0914539A patent/BRPI0914539A2/pt not_active IP Right Cessation
- 2009-06-25 WO PCT/US2009/048564 patent/WO2009158452A1/en not_active Ceased
- 2009-06-25 EP EP09770985.1A patent/EP2323983B1/en not_active Not-in-force
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- 2010-12-14 CO CO10157214A patent/CO6321247A2/es active IP Right Grant
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