TWI331606B - Piperidine derivatives useful as ccr5 antagonists - Google Patents
Piperidine derivatives useful as ccr5 antagonists Download PDFInfo
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- TWI331606B TWI331606B TW092135748A TW92135748A TWI331606B TW I331606 B TWI331606 B TW I331606B TW 092135748 A TW092135748 A TW 092135748A TW 92135748 A TW92135748 A TW 92135748A TW I331606 B TWI331606 B TW I331606B
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- cycloalkyl
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
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Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US43430602P | 2002-12-18 | 2002-12-18 |
Publications (2)
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| TW200427682A TW200427682A (en) | 2004-12-16 |
| TWI331606B true TWI331606B (en) | 2010-10-11 |
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| Application Number | Title | Priority Date | Filing Date |
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| TW092135748A TWI331606B (en) | 2002-12-18 | 2003-12-17 | Piperidine derivatives useful as ccr5 antagonists |
Country Status (16)
| Country | Link |
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| US (2) | US7307081B2 (https=) |
| EP (1) | EP1581494A2 (https=) |
| JP (1) | JP4589728B2 (https=) |
| KR (1) | KR20050085700A (https=) |
| CN (2) | CN100591678C (https=) |
| AR (1) | AR042481A1 (https=) |
| AU (1) | AU2003297400B2 (https=) |
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| PE (1) | PE20040769A1 (https=) |
| TW (1) | TWI331606B (https=) |
| WO (1) | WO2004056770A2 (https=) |
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| BRPI0509803A (pt) | 2004-04-13 | 2007-09-18 | Incyte Corp | derivados de piperazinilpiperidina como antagonistas de receptor de quimiocina |
| US7635698B2 (en) | 2004-12-29 | 2009-12-22 | Millennium Pharmaceuticals, Inc. | Compounds useful as chemokine receptor antagonists |
| US7880002B2 (en) | 2004-12-29 | 2011-02-01 | Millennium Pharmaceuticals, Inc. | Substituted piperazinyl-pyrrolidine compounds useful as chemokine receptor antagonists |
| JP4769257B2 (ja) * | 2005-02-23 | 2011-09-07 | シェーリング コーポレイション | ケモカインレセプターのインヒビターとして有用なピペリジニルピペラジン誘導体 |
| EP1858886A1 (en) * | 2005-02-23 | 2007-11-28 | Schering Corporation | Piperidinyl piperidine derivatives useful as inhibitors of chemokine receptors |
| US20070123538A1 (en) * | 2005-11-30 | 2007-05-31 | Schering Corporation | Compositions comprising a combination of CCR5 and CXCR4 antagonists |
| US20080108586A1 (en) * | 2006-09-06 | 2008-05-08 | Incyte Corporation | Combination therapy for human immunodeficiency virus infection |
| US20100063280A1 (en) * | 2006-12-22 | 2010-03-11 | Schering Corporation | Process for preparing ccr-5 receptor antagonists utilizing 4-substituted 1-cyclopropane-sulfonyl-piperidinyl compounds |
| JP7611949B2 (ja) * | 2023-01-27 | 2025-01-10 | 株式会社Ｓｃｒｅｅｎホールディングス | 基板保持装置及びそれを備えた基板処理装置 |
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| IL117149A0 (en) | 1995-02-23 | 1996-06-18 | Schering Corp | Muscarinic antagonists |
| US5889006A (en) | 1995-02-23 | 1999-03-30 | Schering Corporation | Muscarinic antagonists |
| DE19614204A1 (de) * | 1996-04-10 | 1997-10-16 | Thomae Gmbh Dr K | Carbonsäurederivate, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung |
| US5952349A (en) | 1996-07-10 | 1999-09-14 | Schering Corporation | Muscarinic antagonists for treating memory loss |
| US5977138A (en) | 1996-08-15 | 1999-11-02 | Schering Corporation | Ether muscarinic antagonists |
| CA2371583C (en) * | 1999-05-04 | 2005-09-13 | Schering Corporation | Piperazine derivatives useful as ccr5 antagonists |
| HK1039330B (en) * | 1999-05-04 | 2005-12-09 | Schering Corporation | Piperidine derivatives useful as ccr5 antagonists |
| PL364560A1 (en) * | 2001-03-29 | 2004-12-13 | Schering Corporation | Ccr5 antagonists useful for treating aids |
| EP1373206B1 (en) * | 2001-03-29 | 2008-12-24 | Schering Corporation | Aryl oxime-piperazines useful as ccr5 antagonists |
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Also Published As
| Publication number | Publication date |
|---|---|
| JP2006515851A (ja) | 2006-06-08 |
| AR042481A1 (es) | 2005-06-22 |
| KR20050085700A (ko) | 2005-08-29 |
| ZA200504772B (en) | 2006-03-29 |
| CN1729186A (zh) | 2006-02-01 |
| MXPA05006580A (es) | 2005-08-16 |
| CL2003002637A1 (es) | 2005-04-08 |
| CN101768152A (zh) | 2010-07-07 |
| US20040132711A1 (en) | 2004-07-08 |
| WO2004056770A3 (en) | 2004-08-12 |
| NZ540452A (en) | 2008-12-24 |
| TW200427682A (en) | 2004-12-16 |
| WO2004056770A2 (en) | 2004-07-08 |
| AU2003297400B2 (en) | 2010-03-11 |
| JP4589728B2 (ja) | 2010-12-01 |
| AU2003297400A1 (en) | 2004-07-14 |
| CA2510027A1 (en) | 2004-07-08 |
| CN100591678C (zh) | 2010-02-24 |
| US20080095740A1 (en) | 2008-04-24 |
| MY147899A (en) | 2013-01-31 |
| PE20040769A1 (es) | 2004-11-06 |
| EP1581494A2 (en) | 2005-10-05 |
| US7307081B2 (en) | 2007-12-11 |
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| MM4A | Annulment or lapse of patent due to non-payment of fees |