TW499435B - Pregnane glucuronides - Google Patents

Pregnane glucuronides Download PDF

Info

Publication number
TW499435B
TW499435B TW088117305A TW88117305A TW499435B TW 499435 B TW499435 B TW 499435B TW 088117305 A TW088117305 A TW 088117305A TW 88117305 A TW88117305 A TW 88117305A TW 499435 B TW499435 B TW 499435B
Authority
TW
Taiwan
Prior art keywords
pregnane
compound
salt
scope
carbon atoms
Prior art date
Application number
TW088117305A
Other languages
English (en)
Chinese (zh)
Inventor
Christopher P Miller
Bach D Tran
Michael D Collini
Original Assignee
Wyeth Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth Corp filed Critical Wyeth Corp
Application granted granted Critical
Publication of TW499435B publication Critical patent/TW499435B/zh

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J17/00Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J17/005Glycosides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C07J5/0007Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa
    • C07J5/0015Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa not substituted in position 16

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
TW088117305A 1998-10-13 1999-10-07 Pregnane glucuronides TW499435B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US17034298A 1998-10-13 1998-10-13

Publications (1)

Publication Number Publication Date
TW499435B true TW499435B (en) 2002-08-21

Family

ID=22619512

Family Applications (1)

Application Number Title Priority Date Filing Date
TW088117305A TW499435B (en) 1998-10-13 1999-10-07 Pregnane glucuronides

Country Status (17)

Country Link
EP (1) EP1121376A1 (es)
JP (1) JP2002527448A (es)
KR (1) KR20010080102A (es)
CN (1) CN1330659A (es)
AR (1) AR020778A1 (es)
AU (1) AU751708B2 (es)
BR (1) BR9914521A (es)
CA (1) CA2346693A1 (es)
CZ (1) CZ20011343A3 (es)
EA (1) EA200100437A1 (es)
HU (1) HUP0103992A3 (es)
IL (1) IL142441A0 (es)
NO (1) NO20011825L (es)
PL (1) PL347270A1 (es)
TW (1) TW499435B (es)
WO (1) WO2000021977A1 (es)
ZA (1) ZA200103012B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0104423D0 (sv) * 2001-12-27 2001-12-27 Umecrine Ab Pregnane steroids and their use in the treatment of CNS disorders
KR100440607B1 (ko) * 2001-12-28 2004-07-15 주식회사 엘컴사이언스 프레그난 배당체 화합물 및 이를 유효성분으로 함유하는퇴행성 뇌신경계 질환의 예방 및 치료제

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2029011B (en) * 1978-09-01 1983-02-02 Coulson W Use of a synthetic bifunctional ligand for the immunimetric determination of the concentration ratio of two solutes

Also Published As

Publication number Publication date
EA200100437A1 (ru) 2001-10-22
KR20010080102A (ko) 2001-08-22
HUP0103992A3 (en) 2002-12-28
HUP0103992A2 (hu) 2002-04-29
WO2000021977A1 (en) 2000-04-20
CA2346693A1 (en) 2000-04-20
IL142441A0 (en) 2002-03-10
AU751708B2 (en) 2002-08-22
ZA200103012B (en) 2002-07-11
BR9914521A (pt) 2001-06-26
NO20011825L (no) 2001-06-05
CZ20011343A3 (cs) 2002-04-17
AR020778A1 (es) 2002-05-29
EP1121376A1 (en) 2001-08-08
NO20011825D0 (no) 2001-04-10
AU6511599A (en) 2000-05-01
CN1330659A (zh) 2002-01-09
JP2002527448A (ja) 2002-08-27
PL347270A1 (en) 2002-03-25

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