CA2346693A1 - Pregnane glucuronides - Google Patents

Pregnane glucuronides Download PDF

Info

Publication number
CA2346693A1
CA2346693A1 CA002346693A CA2346693A CA2346693A1 CA 2346693 A1 CA2346693 A1 CA 2346693A1 CA 002346693 A CA002346693 A CA 002346693A CA 2346693 A CA2346693 A CA 2346693A CA 2346693 A1 CA2346693 A1 CA 2346693A1
Authority
CA
Canada
Prior art keywords
beta
glucuronide
pregnane
alpha
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002346693A
Other languages
English (en)
French (fr)
Inventor
Christopher Paul Miller
Bach Dinh Tran
Michael David Collini
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wyeth LLC
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2346693A1 publication Critical patent/CA2346693A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J17/00Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
    • C07J17/005Glycosides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07JSTEROIDS
    • C07J5/00Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond
    • C07J5/0007Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa
    • C07J5/0015Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane and substituted in position 21 by only one singly bound oxygen atom, i.e. only one oxygen bound to position 21 by a single bond not substituted in position 17 alfa not substituted in position 16

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA002346693A 1998-10-13 1999-10-07 Pregnane glucuronides Abandoned CA2346693A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US17034298A 1998-10-13 1998-10-13
US09/170,342 1998-10-13
PCT/US1999/023467 WO2000021977A1 (en) 1998-10-13 1999-10-07 Pregnane glucuronides

Publications (1)

Publication Number Publication Date
CA2346693A1 true CA2346693A1 (en) 2000-04-20

Family

ID=22619512

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002346693A Abandoned CA2346693A1 (en) 1998-10-13 1999-10-07 Pregnane glucuronides

Country Status (17)

Country Link
EP (1) EP1121376A1 (es)
JP (1) JP2002527448A (es)
KR (1) KR20010080102A (es)
CN (1) CN1330659A (es)
AR (1) AR020778A1 (es)
AU (1) AU751708B2 (es)
BR (1) BR9914521A (es)
CA (1) CA2346693A1 (es)
CZ (1) CZ20011343A3 (es)
EA (1) EA200100437A1 (es)
HU (1) HUP0103992A3 (es)
IL (1) IL142441A0 (es)
NO (1) NO20011825L (es)
PL (1) PL347270A1 (es)
TW (1) TW499435B (es)
WO (1) WO2000021977A1 (es)
ZA (1) ZA200103012B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0104423D0 (sv) * 2001-12-27 2001-12-27 Umecrine Ab Pregnane steroids and their use in the treatment of CNS disorders
KR100440607B1 (ko) * 2001-12-28 2004-07-15 주식회사 엘컴사이언스 프레그난 배당체 화합물 및 이를 유효성분으로 함유하는퇴행성 뇌신경계 질환의 예방 및 치료제

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2029011B (en) * 1978-09-01 1983-02-02 Coulson W Use of a synthetic bifunctional ligand for the immunimetric determination of the concentration ratio of two solutes

Also Published As

Publication number Publication date
EA200100437A1 (ru) 2001-10-22
TW499435B (en) 2002-08-21
KR20010080102A (ko) 2001-08-22
HUP0103992A3 (en) 2002-12-28
HUP0103992A2 (hu) 2002-04-29
WO2000021977A1 (en) 2000-04-20
IL142441A0 (en) 2002-03-10
AU751708B2 (en) 2002-08-22
ZA200103012B (en) 2002-07-11
BR9914521A (pt) 2001-06-26
NO20011825L (no) 2001-06-05
CZ20011343A3 (cs) 2002-04-17
AR020778A1 (es) 2002-05-29
EP1121376A1 (en) 2001-08-08
NO20011825D0 (no) 2001-04-10
AU6511599A (en) 2000-05-01
CN1330659A (zh) 2002-01-09
JP2002527448A (ja) 2002-08-27
PL347270A1 (en) 2002-03-25

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Legal Events

Date Code Title Description
FZDE Discontinued