TW252044B - - Google Patents

Info

Publication number
TW252044B
TW252044B TW082106170A TW82106170A TW252044B TW 252044 B TW252044 B TW 252044B TW 082106170 A TW082106170 A TW 082106170A TW 82106170 A TW82106170 A TW 82106170A TW 252044 B TW252044 B TW 252044B
Authority
TW
Taiwan
Application number
TW082106170A
Other languages
Chinese (zh)
Inventor
Muller Enzio
Original Assignee
Boehringer Ingelheim Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg
Application granted granted Critical
Publication of TW252044B publication Critical patent/TW252044B/zh

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/08Vasodilators for multiple indications
TW082106170A 1992-08-10 1993-08-02 TW252044B (US20050026921A1-20050203-C00021.png)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE4226371 1992-08-10
DE4238423 1992-11-13

Publications (1)

Publication Number Publication Date
TW252044B true TW252044B (US20050026921A1-20050203-C00021.png) 1995-07-21

Family

ID=25917371

Family Applications (1)

Application Number Title Priority Date Filing Date
TW082106170A TW252044B (US20050026921A1-20050203-C00021.png) 1992-08-10 1993-08-02

Country Status (21)

Country Link
US (1) US5719279A (US20050026921A1-20050203-C00021.png)
EP (1) EP0654033A1 (US20050026921A1-20050203-C00021.png)
JP (1) JPH08500344A (US20050026921A1-20050203-C00021.png)
KR (1) KR950702988A (US20050026921A1-20050203-C00021.png)
CN (1) CN1043348C (US20050026921A1-20050203-C00021.png)
AU (1) AU681348B2 (US20050026921A1-20050203-C00021.png)
BG (1) BG62618B1 (US20050026921A1-20050203-C00021.png)
CA (1) CA2140883A1 (US20050026921A1-20050203-C00021.png)
CZ (1) CZ286459B6 (US20050026921A1-20050203-C00021.png)
FI (1) FI950542A0 (US20050026921A1-20050203-C00021.png)
HU (1) HUT65734A (US20050026921A1-20050203-C00021.png)
IL (1) IL106624A (US20050026921A1-20050203-C00021.png)
MX (1) MX9304819A (US20050026921A1-20050203-C00021.png)
NZ (1) NZ254804A (US20050026921A1-20050203-C00021.png)
PL (1) PL176389B1 (US20050026921A1-20050203-C00021.png)
RU (1) RU2138500C1 (US20050026921A1-20050203-C00021.png)
SG (1) SG55038A1 (US20050026921A1-20050203-C00021.png)
SK (1) SK18595A3 (US20050026921A1-20050203-C00021.png)
TW (1) TW252044B (US20050026921A1-20050203-C00021.png)
UA (1) UA46697C2 (US20050026921A1-20050203-C00021.png)
WO (1) WO1994003456A1 (US20050026921A1-20050203-C00021.png)

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US7407955B2 (en) 2002-08-21 2008-08-05 Boehringer Ingelheim Pharma Gmbh & Co., Kg 8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions
US7569574B2 (en) 2002-08-22 2009-08-04 Boehringer Ingelheim Pharma Gmbh & Co. Kg Purine derivatives, the preparation thereof and their use as pharmaceutical compositions
US7495005B2 (en) 2002-08-22 2009-02-24 Boehringer Ingelheim Pharma Gmbh & Co. Kg Xanthine derivatives, their preparation and their use in pharmaceutical compositions
US7482337B2 (en) * 2002-11-08 2009-01-27 Boehringer Ingelheim Pharma Gmbh & Co. Kg Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions
DE10254304A1 (de) 2002-11-21 2004-06-03 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Xanthinderivate, deren Herstellung und deren Verwendung als Arzneimittel
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JP2007506804A (ja) * 2003-06-09 2007-03-22 エンダセア, インコーポレイテッド A1アデノシンレセプターアンタゴニスト
US7566707B2 (en) 2003-06-18 2009-07-28 Boehringer Ingelheim International Gmbh Imidazopyridazinone and imidazopyridone derivatives, the preparation thereof and their use as pharmaceutical compositions
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DE102004009039A1 (de) 2004-02-23 2005-09-08 Boehringer Ingelheim Pharma Gmbh & Co. Kg 8-[3-Amino-piperidin-1-yl]-xanthine, deren Herstellung und Verwendung als Arzneimittel
US7393847B2 (en) 2004-03-13 2008-07-01 Boehringer Ingleheim International Gmbh Imidazopyridazinediones, their preparation and their use as pharmaceutical compositions
US7179809B2 (en) * 2004-04-10 2007-02-20 Boehringer Ingelheim International Gmbh 2-Amino-imidazo[4,5-d]pyridazin-4-ones, their preparation and their use as pharmaceutical compositions
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EA015687B1 (ru) 2006-05-04 2011-10-31 Бёрингер Ингельхайм Интернациональ Гмбх Полиморфы
WO2008017670A1 (en) * 2006-08-08 2008-02-14 Boehringer Ingelheim International Gmbh Pyrrolo [3, 2 -d] pyrimidines as dpp-iv inhibitors for the treatment of diabetes mellitus
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KR20190016601A (ko) 2008-08-06 2019-02-18 베링거 인겔하임 인터내셔날 게엠베하 메트포르민 요법이 부적합한 환자에서의 당뇨병 치료
CN103816158A (zh) * 2008-08-15 2014-05-28 勃林格殷格翰国际有限公司 用于治疗fab-相关疾病的嘌呤衍生物
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US20200155558A1 (en) 2018-11-20 2020-05-21 Boehringer Ingelheim International Gmbh Treatment for diabetes in patients with insufficient glycemic control despite therapy with an oral antidiabetic drug
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WO2013174767A1 (en) 2012-05-24 2013-11-28 Boehringer Ingelheim International Gmbh A xanthine derivative as dpp -4 inhibitor for use in modifying food intake and regulating food preference
JP6615109B2 (ja) 2014-02-28 2019-12-04 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Dpp−4阻害薬の医学的使用
WO2017211979A1 (en) 2016-06-10 2017-12-14 Boehringer Ingelheim International Gmbh Combinations of linagliptin and metformin
RU2643336C1 (ru) * 2016-10-03 2018-01-31 Общество с Ограниченной Ответственностью "Компания "ЭЛТА" СРЕДСТВО, ПРОЯВЛЯЮЩЕЕ АНТИТРОМБОТИЧЕСКИЙ ЭФФЕКТ ПОСРЕДСТВОМ БЛОКИРОВАНИЯ РЕЦЕПТОРОВ ТРОМБОЦИТОВ ГП IIb-IIIa (ВАРИАНТЫ)
CN109796453A (zh) * 2019-02-12 2019-05-24 南京纽邦生物科技有限公司 一种1,7-二甲基黄嘌呤的制备方法
US20240002416A1 (en) 2020-10-15 2024-01-04 Rheinische-Friedrich-Wilhelms-Universität Bonn MRGPRX4 Agonists and Antagonists

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Also Published As

Publication number Publication date
SG55038A1 (en) 1998-12-21
RU95109100A (ru) 1996-12-27
HU9302302D0 (en) 1993-10-28
SK18595A3 (en) 1995-07-11
BG99489A (bg) 1996-01-31
FI950542A (fi) 1995-02-08
NZ254804A (en) 1997-01-29
IL106624A (en) 1999-01-26
BG62618B1 (bg) 2000-03-31
CN1086818A (zh) 1994-05-18
AU681348B2 (en) 1997-08-28
WO1994003456A1 (de) 1994-02-17
CN1043348C (zh) 1999-05-12
KR950702988A (ko) 1995-08-23
CA2140883A1 (en) 1994-02-17
IL106624A0 (en) 1993-12-08
AU4707193A (en) 1994-03-03
FI950542A0 (fi) 1995-02-08
RU2138500C1 (ru) 1999-09-27
MX9304819A (es) 1994-02-28
EP0654033A1 (de) 1995-05-24
CZ34895A3 (en) 1995-10-18
PL176389B1 (pl) 1999-05-31
PL307397A1 (en) 1995-05-15
UA46697C2 (uk) 2002-06-17
US5719279A (en) 1998-02-17
HUT65734A (en) 1994-07-28
CZ286459B6 (en) 2000-04-12
JPH08500344A (ja) 1996-01-16

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