TW202241846A - 具有ep拮抗活性之化合物的鹽、溶劑合物及結晶 - Google Patents

具有ep拮抗活性之化合物的鹽、溶劑合物及結晶 Download PDF

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TW202241846A
TW202241846A TW110148402A TW110148402A TW202241846A TW 202241846 A TW202241846 A TW 202241846A TW 110148402 A TW110148402 A TW 110148402A TW 110148402 A TW110148402 A TW 110148402A TW 202241846 A TW202241846 A TW 202241846A
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Taiwan
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crystal
compound
powder
cancer
ray diffraction
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TW110148402A
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Chinese (zh)
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大谷修平
藤戸貴之
西馬直希
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日商小野藥品工業股份有限公司
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    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
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    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/42Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/44Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C07C235/56Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring

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TW110148402A 2020-12-24 2021-12-23 具有ep拮抗活性之化合物的鹽、溶劑合物及結晶 TW202241846A (zh)

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Application Number Priority Date Filing Date Title
JP2020-214481 2020-12-24
JP2020214481 2020-12-24

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TW202241846A true TW202241846A (zh) 2022-11-01

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TW110148402A TW202241846A (zh) 2020-12-24 2021-12-23 具有ep拮抗活性之化合物的鹽、溶劑合物及結晶

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JP (1) JPWO2022138792A1 (enrdf_load_stackoverflow)
TW (1) TW202241846A (enrdf_load_stackoverflow)
WO (1) WO2022138792A1 (enrdf_load_stackoverflow)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2004268839A1 (en) * 2003-09-03 2005-03-10 Pfizer Inc. Phenyl or pyridyl amide compounds as prostaglandin E2 antagonists
US7326732B2 (en) * 2004-02-12 2008-02-05 Pharmagene Laboratories Limited EP2 receptor agonists
TW201326154A (zh) * 2011-11-28 2013-07-01 拜耳知識產權公司 作為ep2受體拮抗劑之新穎2h-吲唑
WO2013164326A1 (en) * 2012-05-03 2013-11-07 Takeda Gmbh Novel ep2 receptor agonists
TW202114985A (zh) * 2019-06-28 2021-04-16 日商小野藥品工業股份有限公司 Ep拮抗劑

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JPWO2022138792A1 (enrdf_load_stackoverflow) 2022-06-30

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