TW202233178A - 固體配製物 - Google Patents
固體配製物 Download PDFInfo
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- TW202233178A TW202233178A TW110140905A TW110140905A TW202233178A TW 202233178 A TW202233178 A TW 202233178A TW 110140905 A TW110140905 A TW 110140905A TW 110140905 A TW110140905 A TW 110140905A TW 202233178 A TW202233178 A TW 202233178A
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- pharmaceutical formulation
- formulation
- api
- pharmaceutical
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- JUQGWKYSEXPRGL-UHFFFAOYSA-M sodium;tetradecanoate Chemical compound [Na+].CCCCCCCCCCCCCC([O-])=O JUQGWKYSEXPRGL-UHFFFAOYSA-M 0.000 description 1
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- 239000011877 solvent mixture Substances 0.000 description 1
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- 235000015523 tannic acid Nutrition 0.000 description 1
- 229940033123 tannic acid Drugs 0.000 description 1
- 229920002258 tannic acid Polymers 0.000 description 1
- 239000011975 tartaric acid Substances 0.000 description 1
- 229960001367 tartaric acid Drugs 0.000 description 1
- 235000002906 tartaric acid Nutrition 0.000 description 1
- 229940095064 tartrate Drugs 0.000 description 1
- WBWWGRHZICKQGZ-GIHLXUJPSA-N taurocholic acid Chemical compound C([C@@H]1C[C@H]2O)[C@@H](O)CC[C@]1(C)[C@@H]1[C@@H]2[C@@H]2CC[C@@H]([C@@H](CCC(=O)NCCS(O)(=O)=O)C)[C@@]2(C)[C@H](O)C1 WBWWGRHZICKQGZ-GIHLXUJPSA-N 0.000 description 1
- MHXBHWLGRWOABW-UHFFFAOYSA-N tetradecyl octadecanoate Chemical compound CCCCCCCCCCCCCCCCCC(=O)OCCCCCCCCCCCCCC MHXBHWLGRWOABW-UHFFFAOYSA-N 0.000 description 1
- 150000003567 thiocyanates Chemical class 0.000 description 1
- 238000011200 topical administration Methods 0.000 description 1
- 239000006208 topical dosage form Substances 0.000 description 1
- 238000012546 transfer Methods 0.000 description 1
- ODLHGICHYURWBS-LKONHMLTSA-N trappsol cyclo Chemical compound CC(O)COC[C@H]([C@H]([C@@H]([C@H]1O)O)O[C@H]2O[C@@H]([C@@H](O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O[C@H]3O[C@H](COCC(C)O)[C@H]([C@@H]([C@H]3O)O)O3)[C@H](O)[C@H]2O)COCC(O)C)O[C@@H]1O[C@H]1[C@H](O)[C@@H](O)[C@@H]3O[C@@H]1COCC(C)O ODLHGICHYURWBS-LKONHMLTSA-N 0.000 description 1
- LENZDBCJOHFCAS-UHFFFAOYSA-N tris Chemical compound OCC(N)(CO)CO LENZDBCJOHFCAS-UHFFFAOYSA-N 0.000 description 1
- 229960004418 trolamine Drugs 0.000 description 1
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- 229960002703 undecylenic acid Drugs 0.000 description 1
- 229940070710 valerate Drugs 0.000 description 1
- NQPDZGIKBAWPEJ-UHFFFAOYSA-N valeric acid Chemical compound CCCCC(O)=O NQPDZGIKBAWPEJ-UHFFFAOYSA-N 0.000 description 1
- 229940124549 vasodilator Drugs 0.000 description 1
- 239000003071 vasodilator agent Substances 0.000 description 1
- 239000003981 vehicle Substances 0.000 description 1
- 229940053446 vitamin E d-alpha Drugs 0.000 description 1
- 239000000341 volatile oil Substances 0.000 description 1
- 239000003871 white petrolatum Substances 0.000 description 1
- 239000000230 xanthan gum Substances 0.000 description 1
- 235000010493 xanthan gum Nutrition 0.000 description 1
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- 229940082509 xanthan gum Drugs 0.000 description 1
- 229950000339 xinafoate Drugs 0.000 description 1
- 239000010457 zeolite Substances 0.000 description 1
- UGZADUVQMDAIAO-UHFFFAOYSA-L zinc hydroxide Chemical compound [OH-].[OH-].[Zn+2] UGZADUVQMDAIAO-UHFFFAOYSA-L 0.000 description 1
- 229940007718 zinc hydroxide Drugs 0.000 description 1
- 229910021511 zinc hydroxide Inorganic materials 0.000 description 1
- 239000002076 α-tocopherol Substances 0.000 description 1
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- GVJHHUAWPYXKBD-IEOSBIPESA-N α-tocopherol Chemical compound OC1=C(C)C(C)=C2O[C@@](CCC[C@H](C)CCC[C@H](C)CCCC(C)C)(C)CCC2=C1C GVJHHUAWPYXKBD-IEOSBIPESA-N 0.000 description 1
Images
Classifications
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- A—HUMAN NECESSITIES
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- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
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- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
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- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
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- Veterinary Medicine (AREA)
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- Communicable Diseases (AREA)
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- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
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PCT/CN2020/126596 WO2022094816A1 (fr) | 2020-11-04 | 2020-11-04 | Formulation solide |
WOPCT/CN2020/126596 | 2020-11-04 |
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TW202233178A true TW202233178A (zh) | 2022-09-01 |
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TW110140905A TW202233178A (zh) | 2020-11-04 | 2021-11-03 | 固體配製物 |
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US (1) | US20240000749A1 (fr) |
EP (1) | EP4240331A1 (fr) |
JP (1) | JP2023548348A (fr) |
KR (1) | KR20230104226A (fr) |
CN (1) | CN116685317A (fr) |
AU (1) | AU2021376584A1 (fr) |
CA (1) | CA3200538A1 (fr) |
CO (1) | CO2023005726A2 (fr) |
CR (1) | CR20230192A (fr) |
DO (1) | DOP2023000084A (fr) |
MX (1) | MX2023005219A (fr) |
PE (1) | PE20231946A1 (fr) |
TW (1) | TW202233178A (fr) |
UY (1) | UY39503A (fr) |
WO (2) | WO2022094816A1 (fr) |
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WO2024080308A1 (fr) * | 2022-10-12 | 2024-04-18 | 中外製薬株式会社 | Composition contenant un peptide, un tensioactif et un polymère |
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WO2015103230A1 (fr) * | 2013-12-31 | 2015-07-09 | Ascendia Pharmaceuticals, Llc | Compositions pharmaceutiques pour composés faiblement hydrosolubles |
JOP20160086B1 (ar) * | 2015-05-08 | 2021-08-17 | 2 Katholieke Univ Leuven Ku Leuven Research And Development | مشتقات اندول مستبدلة احاديا او ثنائيا بصفتها مانعات للتكاثر الفيروسي لحمى الفنك |
EP3305289A1 (fr) * | 2016-10-06 | 2018-04-11 | Philipps-Universität Marburg | Utilisation de silvestrol, épisilvestrol et silvestrol analoga pour le traitement d'infections virales provoquées par des virus avec traduction dépendante de la coiffe |
KR102295179B1 (ko) * | 2017-09-14 | 2021-08-30 | 피닉스 바이오테크놀러지 인코포레이티드. | 바이러스 감염 치료를 위한 방법 및 조성물 |
US20190365738A1 (en) * | 2018-05-21 | 2019-12-05 | Cadila Healthcare Limited | Amorphous solid dispersion of valbenazine tosylate and process for preparation thereof |
AU2019344905A1 (en) * | 2018-09-18 | 2021-04-29 | Metacrine, Inc. | Crystalline forms of a farnesoid X receptor agonist |
KR102173092B1 (ko) * | 2018-11-20 | 2020-11-02 | 중앙대학교 산학협력단 | 루테인 장용성 고체분산체를 유효성분으로 함유하는 위산보호용 조성물 및 이를 포함하는 경구용 제제 |
CN111407728B (zh) * | 2020-04-16 | 2022-02-22 | 重庆市畜牧科学院 | 一种替米考星肠溶性固体分散体及其制备方法和应用 |
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2020
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2021
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- 2021-11-03 MX MX2023005219A patent/MX2023005219A/es unknown
- 2021-11-03 AU AU2021376584A patent/AU2021376584A1/en active Pending
- 2021-11-03 TW TW110140905A patent/TW202233178A/zh unknown
- 2021-11-03 US US18/035,279 patent/US20240000749A1/en active Pending
- 2021-11-03 JP JP2023526557A patent/JP2023548348A/ja active Pending
- 2021-11-03 EP EP21809914.1A patent/EP4240331A1/fr active Pending
- 2021-11-03 CN CN202180088975.2A patent/CN116685317A/zh active Pending
- 2021-11-03 PE PE2023001555A patent/PE20231946A1/es unknown
- 2021-11-03 CA CA3200538A patent/CA3200538A1/fr active Pending
- 2021-11-03 CR CR20230192A patent/CR20230192A/es unknown
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- 2021-11-03 KR KR1020237018792A patent/KR20230104226A/ko unknown
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2023
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- 2023-05-05 CO CONC2023/0005726A patent/CO2023005726A2/es unknown
Also Published As
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JP2023548348A (ja) | 2023-11-16 |
UY39503A (es) | 2022-05-31 |
WO2022094816A1 (fr) | 2022-05-12 |
AU2021376584A1 (en) | 2023-06-29 |
DOP2023000084A (es) | 2023-11-15 |
EP4240331A1 (fr) | 2023-09-13 |
WO2022095913A1 (fr) | 2022-05-12 |
CA3200538A1 (fr) | 2022-05-12 |
CO2023005726A2 (es) | 2023-05-29 |
US20240000749A1 (en) | 2024-01-04 |
CR20230192A (es) | 2023-10-26 |
KR20230104226A (ko) | 2023-07-07 |
MX2023005219A (es) | 2023-07-25 |
CN116685317A (zh) | 2023-09-01 |
PE20231946A1 (es) | 2023-12-05 |
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