TW202132249A - 大麻二酚型大麻素化合物 - Google Patents

大麻二酚型大麻素化合物 Download PDF

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Publication number
TW202132249A
TW202132249A TW109140701A TW109140701A TW202132249A TW 202132249 A TW202132249 A TW 202132249A TW 109140701 A TW109140701 A TW 109140701A TW 109140701 A TW109140701 A TW 109140701A TW 202132249 A TW202132249 A TW 202132249A
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Taiwan
Prior art keywords
cbd
cannabidiol
dose
cannabinoids
compound
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Application number
TW109140701A
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English (en)
Chinese (zh)
Inventor
吉歐孚瑞 蓋
沃克 克納佩爾茲
班傑明 懷利
羅伯茨 瑪利 伍利
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英商吉偉研究有限公司
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Publication of TW202132249A publication Critical patent/TW202132249A/zh

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/658Medicinal preparations containing organic active ingredients o-phenolic cannabinoids, e.g. cannabidiol, cannabigerolic acid, cannabichromene or tetrahydrocannabinol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K36/00Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
    • A61K36/18Magnoliophyta (angiosperms)
    • A61K36/185Magnoliopsida (dicotyledons)
    • A61K36/348Cannabaceae
    • A61K36/3482Cannabis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C29/00Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
    • C07C29/132Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group
    • C07C29/136Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group of >C=O containing groups, e.g. —COOH
    • C07C29/143Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group of >C=O containing groups, e.g. —COOH of ketones
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C39/00Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a six-membered aromatic ring
    • C07C39/23Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a six-membered aromatic ring polycyclic, containing six-membered aromatic rings and other rings, with unsaturation outside the aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/12Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/16Systems containing only non-condensed rings with a six-membered ring the ring being unsaturated

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Natural Medicines & Medicinal Plants (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Pain & Pain Management (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Alternative & Traditional Medicine (AREA)
  • Biotechnology (AREA)
  • Mycology (AREA)
  • Botany (AREA)
  • Medical Informatics (AREA)
  • Microbiology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
TW109140701A 2019-11-21 2020-11-20 大麻二酚型大麻素化合物 TW202132249A (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GBGB1916974.7A GB201916974D0 (en) 2019-11-21 2019-11-21 Cannabidol-type cannabinoid compound
GB1916974.7 2019-11-21

Publications (1)

Publication Number Publication Date
TW202132249A true TW202132249A (zh) 2021-09-01

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ID=69137192

Family Applications (1)

Application Number Title Priority Date Filing Date
TW109140701A TW202132249A (zh) 2019-11-21 2020-11-20 大麻二酚型大麻素化合物

Country Status (17)

Country Link
US (1) US12383512B2 (https=)
EP (1) EP4061344B1 (https=)
JP (1) JP7741071B2 (https=)
KR (1) KR20220103996A (https=)
CN (1) CN114786656A (https=)
AU (1) AU2020389360A1 (https=)
BR (1) BR112022009539A2 (https=)
CA (1) CA3158182A1 (https=)
DK (1) DK4061344T3 (https=)
ES (1) ES2992665T3 (https=)
FI (1) FI4061344T3 (https=)
GB (2) GB201916974D0 (https=)
IL (1) IL293033A (https=)
MX (1) MX2022005995A (https=)
PY (1) PY2076940A (https=)
TW (1) TW202132249A (https=)
WO (1) WO2021099781A1 (https=)

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Publication number Publication date
GB2591567A (en) 2021-08-04
US20230000789A1 (en) 2023-01-05
KR20220103996A (ko) 2022-07-25
GB2591567B (en) 2022-11-16
FI4061344T3 (fi) 2024-07-01
CN114786656A (zh) 2022-07-22
CA3158182A1 (en) 2021-05-27
WO2021099781A1 (en) 2021-05-27
PY2076940A (es) 2021-07-16
GB202018135D0 (en) 2020-12-30
JP7741071B2 (ja) 2025-09-17
EP4061344B1 (en) 2024-05-29
GB201916974D0 (en) 2020-01-08
EP4061344A1 (en) 2022-09-28
MX2022005995A (es) 2022-06-17
GB2591567A9 (en) 2021-12-15
AU2020389360A1 (en) 2022-06-23
JP2023503303A (ja) 2023-01-27
IL293033A (en) 2022-07-01
ES2992665T3 (en) 2024-12-16
DK4061344T3 (da) 2024-07-08
BR112022009539A2 (pt) 2022-08-02
US12383512B2 (en) 2025-08-12

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