TW202120094A - 淚液分泌促進用眼科組成物 - Google Patents
淚液分泌促進用眼科組成物 Download PDFInfo
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- TW202120094A TW202120094A TW109126866A TW109126866A TW202120094A TW 202120094 A TW202120094 A TW 202120094A TW 109126866 A TW109126866 A TW 109126866A TW 109126866 A TW109126866 A TW 109126866A TW 202120094 A TW202120094 A TW 202120094A
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- ophthalmic composition
- salt
- digotinib
- eye
- tear secretion
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Images
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
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- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
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- Organic Chemistry (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JPJP2019-145670 | 2019-08-07 | ||
| JP2019145670 | 2019-08-07 | ||
| JPJP2019-239605 | 2019-12-27 | ||
| JP2019239605 | 2019-12-27 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW202120094A true TW202120094A (zh) | 2021-06-01 |
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| TW109126866A TW202120094A (zh) | 2019-08-07 | 2020-08-07 | 淚液分泌促進用眼科組成物 |
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| EP4176882A4 (en) * | 2020-07-30 | 2024-01-10 | Rohto Pharmaceutical Co., Ltd. | AQUEOUS COMPOSITION |
| JP2025014078A (ja) * | 2021-11-30 | 2025-01-29 | 興和株式会社 | 新規ニコチンアミド化合物及びその用途 |
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| NZ582188A (en) * | 2007-07-11 | 2012-03-30 | Pfizer | Pharmaceutical compositions and methods of treating dry eye disorders |
| TWI466885B (zh) * | 2009-07-31 | 2015-01-01 | Japan Tobacco Inc | 含氮螺環化合物及其醫藥用途 |
| JP6427497B2 (ja) * | 2013-10-21 | 2018-11-21 | 日本たばこ産業株式会社 | 眼疾患の治療剤又は予防剤 |
| CA2991020A1 (en) * | 2015-07-07 | 2017-01-12 | Japan Tobacco Inc. | Method for producing 7h-pyrrolo[2, 3-d]pyrimidine derivative and intermediate thereof |
| TWI790218B (zh) | 2016-12-21 | 2023-01-21 | 日商日本煙草產業股份有限公司 | 7Ｈ－吡咯并[2,3－ｄ]嘧啶衍生物的製造方法及其共結晶 |
| EP3559003B1 (en) * | 2016-12-21 | 2022-08-24 | Japan Tobacco Inc. | Crystalline forms of a janus kinase inhibitor |
| CN119367282A (zh) * | 2019-12-27 | 2025-01-28 | 乐敦制药株式会社 | 水性组合物 |
| JP7722931B2 (ja) * | 2019-12-27 | 2025-08-13 | ロート製薬株式会社 | 水性組成物 |
| US20230285564A1 (en) * | 2020-07-30 | 2023-09-14 | Rohto Pharmaceutical Co., Ltd. | Aqueous Composition |
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- 2020-08-06 WO PCT/JP2020/030231 patent/WO2021025129A1/ja not_active Ceased
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| JPWO2021025129A1 (https=) | 2021-02-11 |
| WO2021025129A1 (ja) | 2021-02-11 |
| CN118903144A (zh) | 2024-11-08 |
| CN114173788A (zh) | 2022-03-11 |
| JP7597714B2 (ja) | 2024-12-10 |
| US20220280515A1 (en) | 2022-09-08 |
| EP4011450A4 (en) | 2023-08-09 |
| EP4011450A1 (en) | 2022-06-15 |
| KR20220044288A (ko) | 2022-04-07 |
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