TW201406403A - 用於治療外科手術疼痛之麻醉乳液調配物 - Google Patents
用於治療外科手術疼痛之麻醉乳液調配物 Download PDFInfo
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- TW201406403A TW201406403A TW102123473A TW102123473A TW201406403A TW 201406403 A TW201406403 A TW 201406403A TW 102123473 A TW102123473 A TW 102123473A TW 102123473 A TW102123473 A TW 102123473A TW 201406403 A TW201406403 A TW 201406403A
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- fentanyl
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- pain
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4468—Non condensed piperidines, e.g. piperocaine having a nitrogen directly attached in position 4, e.g. clebopride, fentanyl
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- A—HUMAN NECESSITIES
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- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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- A—HUMAN NECESSITIES
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- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
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- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/24—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing atoms other than carbon, hydrogen, oxygen, halogen, nitrogen or sulfur, e.g. cyclomethicone or phospholipids
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pain & Pain Management (AREA)
- Dispersion Chemistry (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Dermatology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Rheumatology (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US5357108P | 2008-05-15 | 2008-05-15 | |
| US12/424,382 US20090286832A1 (en) | 2008-05-15 | 2009-04-15 | Narcotic emulsion formulations for treatment of surgical pain |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TW201406403A true TW201406403A (zh) | 2014-02-16 |
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| TW102123473A TW201406403A (zh) | 2008-05-15 | 2009-05-14 | 用於治療外科手術疼痛之麻醉乳液調配物 |
| TW098115948A TWI413531B (zh) | 2008-05-15 | 2009-05-14 | 用於治療外科手術疼痛之麻醉乳液調配物 |
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| Application Number | Title | Priority Date | Filing Date |
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| TW098115948A TWI413531B (zh) | 2008-05-15 | 2009-05-14 | 用於治療外科手術疼痛之麻醉乳液調配物 |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US20090286832A1 (enExample) |
| EP (1) | EP2276440A4 (enExample) |
| JP (2) | JP5689053B2 (enExample) |
| KR (1) | KR101361479B1 (enExample) |
| CN (1) | CN101938963A (enExample) |
| AR (1) | AR071779A1 (enExample) |
| AU (1) | AU2009246713B2 (enExample) |
| BR (1) | BRPI0907224A2 (enExample) |
| CA (1) | CA2710546A1 (enExample) |
| EA (1) | EA201000991A1 (enExample) |
| IL (1) | IL209145A0 (enExample) |
| MX (1) | MX2010007698A (enExample) |
| NZ (1) | NZ586461A (enExample) |
| TW (2) | TW201406403A (enExample) |
| WO (1) | WO2009140059A2 (enExample) |
| ZA (1) | ZA201004392B (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20090286832A1 (en) * | 2008-05-15 | 2009-11-19 | Kiichiro Nabeta | Narcotic emulsion formulations for treatment of surgical pain |
| MX2011007885A (es) * | 2009-02-26 | 2011-12-08 | Techno Guard Co Ltd | Formulaciones de emulsion de narcoticos para tratamiento de dolor por cancer. |
| JP6081240B2 (ja) * | 2013-03-13 | 2017-02-15 | テルモ株式会社 | レミフェンタニル注射液剤 |
| WO2016038734A1 (ja) | 2014-09-12 | 2016-03-17 | テルモ株式会社 | レミフェンタニル注射液剤 |
| US20230248719A1 (en) * | 2020-06-08 | 2023-08-10 | Harm Reduction Therapeutics, Inc. | Sterilized formulations |
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| JPH0647533B2 (ja) * | 1984-08-10 | 1994-06-22 | 裕 水島 | ４−ビフエニリル酢酸系化合物含有脂肪乳剤 |
| US4816247A (en) * | 1985-09-11 | 1989-03-28 | American Cyanamid Company | Emulsion compositions for administration of sparingly water soluble ionizable hydrophobic drugs |
| EP0770387B1 (en) * | 1995-10-28 | 1999-08-11 | B. Braun Melsungen Ag | Pharmaceutical composition containing a local anesthetic and/or centrally acting analgesic |
| GB9721746D0 (en) | 1997-10-15 | 1997-12-10 | Panos Therapeutics Limited | Compositions |
| US6835194B2 (en) * | 1999-03-18 | 2004-12-28 | Durect Corporation | Implantable devices and methods for treatment of pain by delivery of fentanyl and fentanyl congeners |
| US6541021B1 (en) * | 1999-03-18 | 2003-04-01 | Durect Corporation | Devices and methods for pain management |
| US6455525B1 (en) * | 1999-11-04 | 2002-09-24 | Cephalon, Inc. | Heterocyclic substituted pyrazolones |
| US7211596B2 (en) * | 2001-05-11 | 2007-05-01 | Mitsubishi Pharma Corporation | Stable high-concentration injection containing pyrazolone derivative |
| IL162862A0 (en) * | 2002-01-25 | 2005-11-20 | Theravance Inc | Short-acting sedative hypnotic agents for anesthesia and sedation |
| JP2004043479A (ja) * | 2002-07-11 | 2004-02-12 | Taiho Yakuhin Kogyo Kk | 経鼻吸収用組成物 |
| UA80447C2 (en) * | 2002-10-08 | 2007-09-25 | Methods for treating pain by administering nerve growth factor antagonist and opioid analgesic | |
| PT1556083E (pt) * | 2002-10-08 | 2011-03-17 | Rinat Neuroscience Corp | Métodos para tratar a dor pós-cirúrgica pela administração de um anticorpo contra o factor de crescimento nervoso e composições que contêm o mesmo |
| US7648982B2 (en) * | 2003-02-28 | 2010-01-19 | Ym Biosciences Inc. | Opioid delivery system |
| JP2004275852A (ja) * | 2003-03-14 | 2004-10-07 | Mitsubishi Heavy Ind Ltd | 排煙脱硝触媒及びその製造方法 |
| WO2005112926A1 (en) * | 2004-05-17 | 2005-12-01 | Pharmacofore, Inc. | Compositions and methods for treating or preventing pain |
| DE102004025357B4 (de) * | 2004-05-19 | 2007-03-29 | Beiersdorf Ag | Emulsionskonzentrat mit wasserlöslichen und öllöslichen Polymeren und kosmetische Zubereitung enthaltend Emulsionskonzentrat sowie ein Verfahren zu dessen Herstellung und dessen Verwendung |
| US7871632B2 (en) * | 2004-07-12 | 2011-01-18 | Adventrx Pharmaceuticals, Inc. | Compositions for delivering highly water soluble drugs |
| US20060189682A1 (en) * | 2005-02-02 | 2006-08-24 | Payne Joseph E | Water soluble prodrugs of COX-2 inhibitors |
| US20080128314A1 (en) * | 2005-03-14 | 2008-06-05 | Koichi Takeda | Pharmaceutical Composition Containing Hardly Water Soluble Medicament |
| CN101166515A (zh) * | 2005-04-22 | 2008-04-23 | 美国诺华卡迪亚公司 | 用于非水溶性药物成分静脉注射的乳剂的生产 |
| US8158152B2 (en) * | 2005-11-18 | 2012-04-17 | Scidose Llc | Lyophilization process and products obtained thereby |
| US8252328B2 (en) * | 2006-01-06 | 2012-08-28 | Acelrx Pharmaceuticals, Inc. | Bioadhesive drug formulations for oral transmucosal delivery |
| US8486972B2 (en) * | 2006-01-25 | 2013-07-16 | Insys Therapeutics, Inc. | Sublingual fentanyl spray |
| US20090286832A1 (en) * | 2008-05-15 | 2009-11-19 | Kiichiro Nabeta | Narcotic emulsion formulations for treatment of surgical pain |
| MX2011007885A (es) * | 2009-02-26 | 2011-12-08 | Techno Guard Co Ltd | Formulaciones de emulsion de narcoticos para tratamiento de dolor por cancer. |
-
2009
- 2009-04-15 US US12/424,382 patent/US20090286832A1/en not_active Abandoned
- 2009-04-28 KR KR1020107015502A patent/KR101361479B1/ko not_active Expired - Fee Related
- 2009-04-28 WO PCT/US2009/041991 patent/WO2009140059A2/en not_active Ceased
- 2009-04-28 AU AU2009246713A patent/AU2009246713B2/en not_active Ceased
- 2009-04-28 MX MX2010007698A patent/MX2010007698A/es not_active Application Discontinuation
- 2009-04-28 CA CA2710546A patent/CA2710546A1/en not_active Abandoned
- 2009-04-28 NZ NZ586461A patent/NZ586461A/en not_active IP Right Cessation
- 2009-04-28 BR BRPI0907224-1A patent/BRPI0907224A2/pt not_active IP Right Cessation
- 2009-04-28 CN CN2009801021888A patent/CN101938963A/zh active Pending
- 2009-04-28 EA EA201000991A patent/EA201000991A1/ru unknown
- 2009-04-28 JP JP2011509539A patent/JP5689053B2/ja not_active Expired - Fee Related
- 2009-04-28 EP EP09747145A patent/EP2276440A4/en not_active Withdrawn
- 2009-05-13 AR ARP090101725A patent/AR071779A1/es not_active Application Discontinuation
- 2009-05-14 TW TW102123473A patent/TW201406403A/zh unknown
- 2009-05-14 TW TW098115948A patent/TWI413531B/zh not_active IP Right Cessation
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2010
- 2010-06-22 ZA ZA2010/04392A patent/ZA201004392B/en unknown
- 2010-11-04 IL IL209145A patent/IL209145A0/en unknown
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2014
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| ZA201004392B (en) | 2011-06-29 |
| BRPI0907224A2 (pt) | 2019-02-26 |
| NZ586461A (en) | 2012-07-27 |
| TW201006508A (en) | 2010-02-16 |
| EA201000991A1 (ru) | 2011-06-30 |
| US20090286832A1 (en) | 2009-11-19 |
| JP2011520883A (ja) | 2011-07-21 |
| KR101361479B1 (ko) | 2014-02-12 |
| KR20100126270A (ko) | 2010-12-01 |
| CA2710546A1 (en) | 2009-11-19 |
| EP2276440A2 (en) | 2011-01-26 |
| JP5889364B2 (ja) | 2016-03-22 |
| WO2009140059A3 (en) | 2010-01-07 |
| MX2010007698A (es) | 2010-11-22 |
| TWI413531B (zh) | 2013-11-01 |
| WO2009140059A2 (en) | 2009-11-19 |
| JP2014205681A (ja) | 2014-10-30 |
| IL209145A0 (en) | 2011-01-31 |
| JP5689053B2 (ja) | 2015-03-25 |
| AU2009246713B2 (en) | 2012-10-25 |
| EP2276440A4 (en) | 2011-06-29 |
| CN101938963A (zh) | 2011-01-05 |
| AU2009246713A1 (en) | 2009-11-19 |
| AR071779A1 (es) | 2010-07-14 |
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