CA2710546A1 - Narcotic emulsion formulations for treatment of surgical pain - Google Patents
Narcotic emulsion formulations for treatment of surgical pain Download PDFInfo
- Publication number
- CA2710546A1 CA2710546A1 CA2710546A CA2710546A CA2710546A1 CA 2710546 A1 CA2710546 A1 CA 2710546A1 CA 2710546 A CA2710546 A CA 2710546A CA 2710546 A CA2710546 A CA 2710546A CA 2710546 A1 CA2710546 A1 CA 2710546A1
- Authority
- CA
- Canada
- Prior art keywords
- emulsion
- fentanyl
- emulsion formulation
- pain
- formulation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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Classifications
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4468—Non condensed piperidines, e.g. piperocaine having a nitrogen directly attached in position 4, e.g. clebopride, fentanyl
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- A61K9/0012—Galenical forms characterised by the site of application
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- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
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- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
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- A61K47/24—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing atoms other than carbon, hydrogen, oxygen, halogen, nitrogen or sulfur, e.g. cyclomethicone or phospholipids
Landscapes
- Health & Medical Sciences (AREA)
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- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
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- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US5357108P | 2008-05-15 | 2008-05-15 | |
| US61/053,571 | 2008-05-15 | ||
| US12/424,382 | 2009-04-15 | ||
| US12/424,382 US20090286832A1 (en) | 2008-05-15 | 2009-04-15 | Narcotic emulsion formulations for treatment of surgical pain |
| PCT/US2009/041991 WO2009140059A2 (en) | 2008-05-15 | 2009-04-28 | Narcotic emulsion formulations for treatment of surgical pain |
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| CA2710546A1 true CA2710546A1 (en) | 2009-11-19 |
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| CA2710546A Abandoned CA2710546A1 (en) | 2008-05-15 | 2009-04-28 | Narcotic emulsion formulations for treatment of surgical pain |
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| EP (1) | EP2276440A4 (enExample) |
| JP (2) | JP5689053B2 (enExample) |
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| AR (1) | AR071779A1 (enExample) |
| AU (1) | AU2009246713B2 (enExample) |
| BR (1) | BRPI0907224A2 (enExample) |
| CA (1) | CA2710546A1 (enExample) |
| EA (1) | EA201000991A1 (enExample) |
| IL (1) | IL209145A0 (enExample) |
| MX (1) | MX2010007698A (enExample) |
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| TW (2) | TWI413531B (enExample) |
| WO (1) | WO2009140059A2 (enExample) |
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| US20090286832A1 (en) * | 2008-05-15 | 2009-11-19 | Kiichiro Nabeta | Narcotic emulsion formulations for treatment of surgical pain |
| KR101564058B1 (ko) * | 2009-02-26 | 2015-10-29 | 테이코쿠 팔마 유에스에이, 인코포레이티드 | 암 통증 치료용 마취 유상액 제제 |
| JP6081240B2 (ja) * | 2013-03-13 | 2017-02-15 | テルモ株式会社 | レミフェンタニル注射液剤 |
| EP3192509B1 (en) | 2014-09-12 | 2021-03-31 | Terumo Kabushiki Kaisha | Remifentanil injection |
| WO2021252449A1 (en) * | 2020-06-08 | 2021-12-16 | Harm Reduction Therapeutics, Inc. | Sterilized formulations |
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| US4816247A (en) * | 1985-09-11 | 1989-03-28 | American Cyanamid Company | Emulsion compositions for administration of sparingly water soluble ionizable hydrophobic drugs |
| ATE183092T1 (de) * | 1995-10-28 | 1999-08-15 | Braun Melsungen Ag | Lokalanästhetika und/oder zentralanalgetika enthaltende pharmazeutische zusammensetzungen |
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| US6541021B1 (en) * | 1999-03-18 | 2003-04-01 | Durect Corporation | Devices and methods for pain management |
| US6835194B2 (en) * | 1999-03-18 | 2004-12-28 | Durect Corporation | Implantable devices and methods for treatment of pain by delivery of fentanyl and fentanyl congeners |
| US6455525B1 (en) * | 1999-11-04 | 2002-09-24 | Cephalon, Inc. | Heterocyclic substituted pyrazolones |
| CA2446837C (en) * | 2001-05-11 | 2012-01-03 | Mitsubishi Pharma Corporation | Stable high-concentration injection containing pyrazolone derivative |
| RU2315037C2 (ru) * | 2002-01-25 | 2008-01-20 | Тереванс, Инк. | Замещенные эфиры фенилуксусной кислоты в качестве короткодействующих седативных снотворных агентов для кратковременной анестезии и создания седативного эффекта, промежуточное соединение, фармацевтическая композиция и применение |
| JP2004043479A (ja) * | 2002-07-11 | 2004-02-12 | Taiho Yakuhin Kogyo Kk | 経鼻吸収用組成物 |
| UA80447C2 (en) * | 2002-10-08 | 2007-09-25 | Methods for treating pain by administering nerve growth factor antagonist and opioid analgesic | |
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| KR101564058B1 (ko) * | 2009-02-26 | 2015-10-29 | 테이코쿠 팔마 유에스에이, 인코포레이티드 | 암 통증 치료용 마취 유상액 제제 |
-
2009
- 2009-04-15 US US12/424,382 patent/US20090286832A1/en not_active Abandoned
- 2009-04-28 CN CN2009801021888A patent/CN101938963A/zh active Pending
- 2009-04-28 BR BRPI0907224-1A patent/BRPI0907224A2/pt not_active IP Right Cessation
- 2009-04-28 NZ NZ586461A patent/NZ586461A/en not_active IP Right Cessation
- 2009-04-28 EA EA201000991A patent/EA201000991A1/ru unknown
- 2009-04-28 WO PCT/US2009/041991 patent/WO2009140059A2/en not_active Ceased
- 2009-04-28 CA CA2710546A patent/CA2710546A1/en not_active Abandoned
- 2009-04-28 JP JP2011509539A patent/JP5689053B2/ja not_active Expired - Fee Related
- 2009-04-28 AU AU2009246713A patent/AU2009246713B2/en not_active Ceased
- 2009-04-28 KR KR1020107015502A patent/KR101361479B1/ko not_active Expired - Fee Related
- 2009-04-28 MX MX2010007698A patent/MX2010007698A/es not_active Application Discontinuation
- 2009-04-28 EP EP09747145A patent/EP2276440A4/en not_active Withdrawn
- 2009-05-13 AR ARP090101725A patent/AR071779A1/es not_active Application Discontinuation
- 2009-05-14 TW TW098115948A patent/TWI413531B/zh not_active IP Right Cessation
- 2009-05-14 TW TW102123473A patent/TW201406403A/zh unknown
-
2010
- 2010-06-22 ZA ZA2010/04392A patent/ZA201004392B/en unknown
- 2010-11-04 IL IL209145A patent/IL209145A0/en unknown
-
2014
- 2014-05-23 JP JP2014107385A patent/JP5889364B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| EA201000991A1 (ru) | 2011-06-30 |
| AR071779A1 (es) | 2010-07-14 |
| CN101938963A (zh) | 2011-01-05 |
| US20090286832A1 (en) | 2009-11-19 |
| TW201406403A (zh) | 2014-02-16 |
| WO2009140059A2 (en) | 2009-11-19 |
| IL209145A0 (en) | 2011-01-31 |
| JP5889364B2 (ja) | 2016-03-22 |
| AU2009246713A1 (en) | 2009-11-19 |
| NZ586461A (en) | 2012-07-27 |
| BRPI0907224A2 (pt) | 2019-02-26 |
| KR101361479B1 (ko) | 2014-02-12 |
| JP2011520883A (ja) | 2011-07-21 |
| JP5689053B2 (ja) | 2015-03-25 |
| WO2009140059A3 (en) | 2010-01-07 |
| TWI413531B (zh) | 2013-11-01 |
| JP2014205681A (ja) | 2014-10-30 |
| TW201006508A (en) | 2010-02-16 |
| ZA201004392B (en) | 2011-06-29 |
| EP2276440A2 (en) | 2011-01-26 |
| EP2276440A4 (en) | 2011-06-29 |
| AU2009246713B2 (en) | 2012-10-25 |
| MX2010007698A (es) | 2010-11-22 |
| KR20100126270A (ko) | 2010-12-01 |
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