TW200734324A - Therapeutic agents - Google Patents

Therapeutic agents

Info

Publication number
TW200734324A
TW200734324A TW095126223A TW95126223A TW200734324A TW 200734324 A TW200734324 A TW 200734324A TW 095126223 A TW095126223 A TW 095126223A TW 95126223 A TW95126223 A TW 95126223A TW 200734324 A TW200734324 A TW 200734324A
Authority
TW
Taiwan
Prior art keywords
therapeutic agents
compounds
psychiatric
obesity
preparing
Prior art date
Application number
TW095126223A
Other languages
English (en)
Inventor
Lei-Feng Cheng
Maria Jonforsen
Peter Schell
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34897416&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TW200734324(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of TW200734324A publication Critical patent/TW200734324A/zh

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Endocrinology (AREA)
  • Reproductive Health (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
  • Pulmonology (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Rheumatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Psychology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Vascular Medicine (AREA)
  • Otolaryngology (AREA)
  • Addiction (AREA)
  • Nutrition Science (AREA)
TW095126223A 2005-07-19 2006-07-18 Therapeutic agents TW200734324A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0514738.4A GB0514738D0 (en) 2005-07-19 2005-07-19 Therapeutic agents

Publications (1)

Publication Number Publication Date
TW200734324A true TW200734324A (en) 2007-09-16

Family

ID=34897416

Family Applications (1)

Application Number Title Priority Date Filing Date
TW095126223A TW200734324A (en) 2005-07-19 2006-07-18 Therapeutic agents

Country Status (16)

Country Link
US (1) US20080287517A1 (zh)
EP (1) EP1910331A1 (zh)
JP (1) JP2009501771A (zh)
KR (1) KR20080032206A (zh)
CN (1) CN101223159A (zh)
AR (1) AR057461A1 (zh)
AU (1) AU2006271499A1 (zh)
CA (1) CA2615588A1 (zh)
GB (1) GB0514738D0 (zh)
IL (1) IL188388A0 (zh)
MX (1) MX2008000891A (zh)
NO (1) NO20080025L (zh)
TW (1) TW200734324A (zh)
UY (1) UY29678A1 (zh)
WO (1) WO2007010217A1 (zh)
ZA (1) ZA200800327B (zh)

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CN101472896A (zh) * 2006-06-20 2009-07-01 阿斯利康(瑞典)有限公司 治疗药剂
JP2009541283A (ja) * 2006-06-20 2009-11-26 アストラゼネカ アクチボラグ 治療薬
EP1946777A1 (en) * 2007-01-16 2008-07-23 Laboratorios del Dr. Esteve S.A. Substituted pyrazoline for preventing weight gain
ES2341522B1 (es) * 2008-12-18 2011-06-06 Laboratorios Del Dr. Esteve, S.A. Compuestos de pirazolina sustituida en la posicion, 4 preparacion y composiciones farmaceuticas que comprenden los mismos.
US9133128B2 (en) 2011-06-17 2015-09-15 Research Triangle Institute Pyrazole derivatives as cannabinoid receptor 1 antagonists
CN109516955B (zh) * 2017-09-20 2022-07-26 华东师范大学 含氮五元芳香杂环化合物及其制备方法和应用
CN113274391B (zh) * 2021-06-01 2022-07-05 苏州大学 吡唑衍生物在制备p2y6r相关治疗动脉粥样硬化及抗炎药物中的应用
WO2023205180A1 (en) 2022-04-19 2023-10-26 Nurix Therapeutics, Inc. Biomarkers for cbl, and compositions and methods for their use
US20230414598A1 (en) 2022-06-22 2023-12-28 Nurix Therapeutics, Inc. Combination therapies with cbl-b inhibitor compounds and antiemetic agents

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FR2665898B1 (fr) * 1990-08-20 1994-03-11 Sanofi Derives d'amido-3 pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2692575B1 (fr) * 1992-06-23 1995-06-30 Sanofi Elf Nouveaux derives du pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2714057B1 (fr) * 1993-12-17 1996-03-08 Sanofi Elf Nouveaux dérivés du 3-pyrazolecarboxamide, procédé pour leur préparation et compositions pharmaceutiques les contenant.
FR2732967B1 (fr) * 1995-04-11 1997-07-04 Sanofi Sa 1-phenylpyrazole-3-carboxamides substitues, actifs sur la neurotensine, leur preparation, les compositions pharmaceutiques en contenant
TNSN99111A1 (fr) * 1998-06-11 2005-11-10 Pfizer Derives de sulfonylbenzene nouveaux, procede pour leur preparation et compositions pharmaceutiques les contenant.
FR2789079B3 (fr) * 1999-02-01 2001-03-02 Sanofi Synthelabo Derive d'acide pyrazolecarboxylique, sa preparation, les compositions pharmaceutiques en contenant
EP1224173B1 (en) * 1999-10-18 2005-10-12 The University Of Connecticut Pyrazole derivatives as cannabinoid receptor antagonists
US7393842B2 (en) * 2001-08-31 2008-07-01 University Of Connecticut Pyrazole analogs acting on cannabinoid receptors
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KR20080032206A (ko) 2008-04-14
JP2009501771A (ja) 2009-01-22
US20080287517A1 (en) 2008-11-20
CA2615588A1 (en) 2007-01-25
NO20080025L (no) 2008-04-16
IL188388A0 (en) 2008-04-13
AR057461A1 (es) 2007-12-05
EP1910331A1 (en) 2008-04-16
UY29678A1 (es) 2007-02-28
GB0514738D0 (en) 2005-08-24
AU2006271499A1 (en) 2007-01-25
CN101223159A (zh) 2008-07-16

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