TR201908994T4 - Farmasötik bileşimler. - Google Patents

Farmasötik bileşimler. Download PDF

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Publication number
TR201908994T4
TR201908994T4 TR2019/08994T TR201908994T TR201908994T4 TR 201908994 T4 TR201908994 T4 TR 201908994T4 TR 2019/08994 T TR2019/08994 T TR 2019/08994T TR 201908994 T TR201908994 T TR 201908994T TR 201908994 T4 TR201908994 T4 TR 201908994T4
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Turkey
Prior art keywords
pharmaceutical compositions
formula
drugs
medicine
compounds
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TR2019/08994T
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English (en)
Inventor
paul cook Gary
Thomas Gwozdz Garry
Patrick Laslo Theodore
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Kalvista Pharmaceuticals Ltd
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Publication of TR201908994T4 publication Critical patent/TR201908994T4/tr

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    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
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    • A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
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    • A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183—Amino acids, e.g. glycine, EDTA or aspartame
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0048—Eye, e.g. artificial tears
    • A61K9/0051—Ocular inserts or implants

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Abstract

Buluş, suda az çözünen ilaçların sulu süspansiyon farmasötik bileşimleri, bu bileşimlerin hazırlanması ve tıpta kullanımı, özellikle de oküler hastalıkların tedavisinde kullanımları için işlemler ile ilgili olup, burada adı geçen ilaçlar, formül (I) bileşiklerinden (Formül (I)) seçilmekte, buradaki R1-R9, burada tanımlanmaktadır.
TR2019/08994T 2013-01-09 2014-01-09 Farmasötik bileşimler. TR201908994T4 (tr)

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US201361750568P 2013-01-09 2013-01-09
GB1301895.7A GB2510407A (en) 2013-02-04 2013-02-04 Aqueous suspensions of kallikrein inhibitors for parenteral administration

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CA2897274C (en) 2021-06-29
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GB201301895D0 (en) 2013-03-20
US10478409B2 (en) 2019-11-19
EP2943181B1 (en) 2019-04-10
ES2728967T3 (es) 2019-10-29
US9849100B2 (en) 2017-12-26
PL2943181T3 (pl) 2019-09-30
GB2510407A (en) 2014-08-06
EP2943181A1 (en) 2015-11-18
US20150342910A1 (en) 2015-12-03
WO2014108685A1 (en) 2014-07-17
CA2897274A1 (en) 2014-07-17
JP2016504406A (ja) 2016-02-12

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