TR200201141T2 - 2-Amino-3,4-dihidro-kinazolinlerin bir ilacın üretiminde kullanımı - Google Patents
2-Amino-3,4-dihidro-kinazolinlerin bir ilacın üretiminde kullanımıInfo
- Publication number
- TR200201141T2 TR200201141T2 TR2002/01141T TR200201141T TR200201141T2 TR 200201141 T2 TR200201141 T2 TR 200201141T2 TR 2002/01141 T TR2002/01141 T TR 2002/01141T TR 200201141 T TR200201141 T TR 200201141T TR 200201141 T2 TR200201141 T2 TR 200201141T2
- Authority
- TR
- Turkey
- Prior art keywords
- dihydro
- drug
- amino
- production
- quinazolines
- Prior art date
Links
- GQRRWNLARRRPRY-UHFFFAOYSA-N 1,4-dihydroquinazolin-2-amine Chemical class C1=CC=C2CNC(N)=NC2=C1 GQRRWNLARRRPRY-UHFFFAOYSA-N 0.000 title abstract 2
- 239000003814 drug Substances 0.000 title abstract 2
- 229940079593 drug Drugs 0.000 title abstract 2
- 230000000302 ischemic effect Effects 0.000 abstract 1
- 238000011321 prophylaxis Methods 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 238000011282 treatment Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/517—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P41/00—Drugs used in surgical methods, e.g. surgery adjuvants for preventing adhesion or for vitreum substitution
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Obesity (AREA)
- Urology & Nephrology (AREA)
- Vascular Medicine (AREA)
- Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Formül I' e göre olan 2-amino-3,4-dihidro-kinazolin' in ve bunlarin farmakolojik tahammül edilebilir tuzlarinin isemik durumlarin tedavi edilmesi ve profilaksina yönelik bir ilacin üretimi için kullanimi tarif edilmektedir. R1, R2 ve R3 istemlerde belirtilen anlamlara sahiptirler. FORMÜL(I)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19951702A DE19951702A1 (de) | 1999-10-27 | 1999-10-27 | Verwendung von 2-Amino-3,4-dihydro-chinazolinen zur Herstellung eines Medikaments zur Behandlung oder Prophylaxe von durch ischämischen Zuständen bewirkten Krankheiten |
Publications (1)
Publication Number | Publication Date |
---|---|
TR200201141T2 true TR200201141T2 (tr) | 2002-11-21 |
Family
ID=7927021
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR2002/01141T TR200201141T2 (tr) | 1999-10-27 | 2000-10-14 | 2-Amino-3,4-dihidro-kinazolinlerin bir ilacın üretiminde kullanımı |
Country Status (28)
Country | Link |
---|---|
US (1) | US6331546B1 (tr) |
EP (1) | EP1244454B1 (tr) |
JP (1) | JP2003512420A (tr) |
KR (1) | KR20020041831A (tr) |
CN (1) | CN1181822C (tr) |
AR (1) | AR026242A1 (tr) |
AT (1) | ATE324111T1 (tr) |
AU (1) | AU7664800A (tr) |
BR (1) | BR0014985A (tr) |
CA (1) | CA2388965A1 (tr) |
CZ (1) | CZ20021414A3 (tr) |
DE (2) | DE19951702A1 (tr) |
EE (1) | EE200200215A (tr) |
HK (1) | HK1050480A1 (tr) |
HR (1) | HRP20020363A2 (tr) |
HU (1) | HUP0203774A3 (tr) |
IL (1) | IL149160A0 (tr) |
MX (1) | MXPA02004035A (tr) |
NO (1) | NO20021710L (tr) |
NZ (1) | NZ518588A (tr) |
PL (1) | PL356399A1 (tr) |
RU (1) | RU2002113667A (tr) |
SK (1) | SK5582002A3 (tr) |
TR (1) | TR200201141T2 (tr) |
TW (1) | TWI227135B (tr) |
WO (1) | WO2001030328A2 (tr) |
YU (1) | YU30602A (tr) |
ZA (1) | ZA200204057B (tr) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE69927987T2 (de) * | 1998-08-13 | 2006-11-09 | Hadasit Medical Research Services & Development Co. Ltd. | Hemmung von mit gewebetrauma verbundenen pathogenen prozessen |
WO2003048129A1 (de) * | 2001-12-05 | 2003-06-12 | Aventis Pharma Deutschland Gmbh | Substituierte 4-phenyltetrahydroisochinoline, verfahren zu ihrer herstellung, ihre verwendung als medikament, sowie sie enthaltendes medikament |
DE10163914A1 (de) * | 2001-12-22 | 2003-07-03 | Aventis Pharma Gmbh | Substituierte 4-Phenyltetrahydroisochinolinium-Salze, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament, sowie sie enthaltendes Medikament |
DE10312963A1 (de) * | 2003-03-24 | 2004-10-07 | Aventis Pharma Deutschland Gmbh | Substituierte 4-Phenyltetrahydroisochinoline, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament, sowie sie enthaltendes Medikament |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3560601A (en) | 1968-11-25 | 1971-02-02 | Ford Motor Co | Process for manufacturing porous thermoplastic sheet material |
IL102764A0 (en) * | 1991-08-16 | 1993-01-31 | Merck & Co Inc | Quinazoline derivatives,and pharmaceutical compositions containing them |
WO1994007498A1 (en) * | 1992-10-07 | 1994-04-14 | Sumitomo Pharmaceuticals Company, Limited | Pharmaceutical composition for inhibiting tumor necrosis factor production |
DE19713427A1 (de) * | 1997-04-01 | 1998-10-08 | Hoechst Ag | Ortho-substituierte Benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
-
1999
- 1999-10-27 DE DE19951702A patent/DE19951702A1/de not_active Withdrawn
-
2000
- 2000-10-14 CN CNB008148872A patent/CN1181822C/zh not_active Expired - Fee Related
- 2000-10-14 NZ NZ518588A patent/NZ518588A/en unknown
- 2000-10-14 TR TR2002/01141T patent/TR200201141T2/tr unknown
- 2000-10-14 AT AT00966165T patent/ATE324111T1/de not_active IP Right Cessation
- 2000-10-14 EE EEP200200215A patent/EE200200215A/xx unknown
- 2000-10-14 KR KR1020027005359A patent/KR20020041831A/ko not_active Application Discontinuation
- 2000-10-14 RU RU2002113667/15A patent/RU2002113667A/ru not_active Application Discontinuation
- 2000-10-14 MX MXPA02004035A patent/MXPA02004035A/es active IP Right Grant
- 2000-10-14 IL IL14916000A patent/IL149160A0/xx unknown
- 2000-10-14 DE DE50012667T patent/DE50012667D1/de not_active Expired - Lifetime
- 2000-10-14 HU HU0203774A patent/HUP0203774A3/hu unknown
- 2000-10-14 BR BR0014985-3A patent/BR0014985A/pt not_active IP Right Cessation
- 2000-10-14 JP JP2001532748A patent/JP2003512420A/ja not_active Abandoned
- 2000-10-14 PL PL00356399A patent/PL356399A1/xx unknown
- 2000-10-14 AU AU76648/00A patent/AU7664800A/en not_active Abandoned
- 2000-10-14 WO PCT/EP2000/010127 patent/WO2001030328A2/de active IP Right Grant
- 2000-10-14 YU YU30602A patent/YU30602A/sh unknown
- 2000-10-14 EP EP00966165A patent/EP1244454B1/de not_active Expired - Lifetime
- 2000-10-14 SK SK558-2002A patent/SK5582002A3/sk unknown
- 2000-10-14 CZ CZ20021414A patent/CZ20021414A3/cs unknown
- 2000-10-14 CA CA002388965A patent/CA2388965A1/en not_active Abandoned
- 2000-10-24 TW TW089122279A patent/TWI227135B/zh not_active IP Right Cessation
- 2000-10-25 AR ARP000105620A patent/AR026242A1/es unknown
- 2000-10-26 US US09/696,233 patent/US6331546B1/en not_active Expired - Fee Related
-
2002
- 2002-04-11 NO NO20021710A patent/NO20021710L/no not_active Application Discontinuation
- 2002-04-25 HR HR20020363A patent/HRP20020363A2/hr not_active Application Discontinuation
- 2002-05-22 ZA ZA200204057A patent/ZA200204057B/en unknown
-
2003
- 2003-04-10 HK HK03102619A patent/HK1050480A1/xx not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
KR20020041831A (ko) | 2002-06-03 |
WO2001030328A3 (de) | 2002-06-20 |
HRP20020363A2 (en) | 2004-02-29 |
WO2001030328A2 (de) | 2001-05-03 |
IL149160A0 (en) | 2002-11-10 |
CA2388965A1 (en) | 2001-05-03 |
CZ20021414A3 (cs) | 2002-07-17 |
EP1244454A2 (de) | 2002-10-02 |
PL356399A1 (en) | 2004-06-28 |
AU7664800A (en) | 2001-05-08 |
EE200200215A (et) | 2003-06-16 |
ZA200204057B (en) | 2003-02-26 |
NZ518588A (en) | 2004-06-25 |
HK1050480A1 (en) | 2003-06-27 |
AR026242A1 (es) | 2003-02-05 |
NO20021710D0 (no) | 2002-04-11 |
SK5582002A3 (en) | 2002-08-06 |
JP2003512420A (ja) | 2003-04-02 |
EP1244454B1 (de) | 2006-04-26 |
RU2002113667A (ru) | 2004-01-10 |
ATE324111T1 (de) | 2006-05-15 |
NO20021710L (no) | 2002-04-11 |
MXPA02004035A (es) | 2002-10-11 |
HUP0203774A2 (en) | 2003-05-28 |
CN1384747A (zh) | 2002-12-11 |
BR0014985A (pt) | 2003-07-22 |
CN1181822C (zh) | 2004-12-29 |
DE50012667D1 (de) | 2006-06-01 |
HUP0203774A3 (en) | 2003-07-28 |
TWI227135B (en) | 2005-02-01 |
DE19951702A1 (de) | 2001-05-03 |
US6331546B1 (en) | 2001-12-18 |
YU30602A (sh) | 2004-12-31 |
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