TR199901705T2 - Trisiklik karbapenem bilesikleri. - Google Patents

Trisiklik karbapenem bilesikleri.

Info

Publication number
TR199901705T2
TR199901705T2 TR1999/01705T TR9901705T TR199901705T2 TR 199901705 T2 TR199901705 T2 TR 199901705T2 TR 1999/01705 T TR1999/01705 T TR 1999/01705T TR 9901705 T TR9901705 T TR 9901705T TR 199901705 T2 TR199901705 T2 TR 199901705T2
Authority
TR
Turkey
Prior art keywords
icleric
carbapenem
tricyclic
bile
chain
Prior art date
Application number
TR1999/01705T
Other languages
English (en)
Inventor
Rossi Tino
Andreotti Daniele
Tedesco Giovanna
Tarsi Luca
Ratti Emiliangelo
Feriani Aldo
Antonia Pizzi Domenica
Gaviraghi Giovari
Biondi Stefano
Finizia Gabriella
Original Assignee
Glaxo Wellcome Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Wellcome Spa filed Critical Glaxo Wellcome Spa
Publication of TR199901705T2 publication Critical patent/TR199901705T2/tr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D477/00—Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)

Abstract

Antibakteriyel bir etkinlige sahip bir formül (I) bilesigi, tuzlari ve metabolik olarak kararsiz esterleri; burada R istege bagli olarak ikameli aril veya heteroaril grubunu temsil eder; A bir propilen zincirini temsil eder veya A, biri bir oksijen veya kükürt atomu veya NH grubu veya ikameli bir türevi arasindan seçilen ve diger ikisi metilen gruplari olan 3 üyeli bir zincirdir; ayrica bunlarin hazirlanmasi için islemler ve tipta kullanimlari açiklanmaktadir.
TR1999/01705T 1996-11-14 1997-11-12 Trisiklik karbapenem bilesikleri. TR199901705T2 (tr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9623684.9A GB9623684D0 (en) 1996-11-14 1996-11-14 Chemical compounds

Publications (1)

Publication Number Publication Date
TR199901705T2 true TR199901705T2 (tr) 1999-12-21

Family

ID=10802915

Family Applications (1)

Application Number Title Priority Date Filing Date
TR1999/01705T TR199901705T2 (tr) 1996-11-14 1997-11-12 Trisiklik karbapenem bilesikleri.

Country Status (17)

Country Link
EP (1) EP0937078B1 (tr)
JP (1) JP2001503765A (tr)
KR (1) KR20000053258A (tr)
AR (1) AR010585A1 (tr)
AT (1) ATE232532T1 (tr)
AU (1) AU727328B2 (tr)
BR (1) BR9713982A (tr)
CA (1) CA2271732A1 (tr)
DE (1) DE69719054T2 (tr)
ES (1) ES2191207T3 (tr)
GB (1) GB9623684D0 (tr)
HR (1) HRP970611A2 (tr)
PE (1) PE14099A1 (tr)
TR (1) TR199901705T2 (tr)
TW (1) TW438802B (tr)
WO (1) WO1998021210A1 (tr)
ZA (1) ZA9710207B (tr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU744739B2 (en) 1998-02-17 2002-02-28 Nippon Kayaku Kabushiki Kaisha Novel acetamide derivative and use thereof
US7601847B2 (en) 2004-10-26 2009-10-13 Wyeth Preparation and purification of 4-(indazol-3-yl)phenols

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CZ435990A3 (cs) * 1989-09-08 1999-11-17 Glaxo S.P.A. Kyselina 10-(1-hydroxyethyl)-11-oxo-1-azatricyklo/7,2,0,03,8/-undec-2en-2-karboxylová a její deriváty, způsob jejich výroby, použití pro výrobu farmaceutických prostředků a farmaceutické prostředky s jejich obsahem
AU636913B2 (en) * 1989-10-11 1993-05-13 Takeda Chemical Industries Ltd. Tricyclic carbapenem compounds
EP0507313A1 (en) * 1991-04-05 1992-10-07 Takeda Chemical Industries, Ltd. Polycyclic carbapenem compounds, their production and use
JPH06166688A (ja) * 1992-10-02 1994-06-14 Takeda Chem Ind Ltd カルバペネム化合物、その製造法および抗菌組成物
JPH08245628A (ja) * 1995-01-12 1996-09-24 Takeda Chem Ind Ltd カルバペネム化合物、その製造法および剤

Also Published As

Publication number Publication date
HRP970611A2 (en) 1998-10-31
ZA9710207B (en) 1999-05-12
WO1998021210A1 (en) 1998-05-22
GB9623684D0 (en) 1997-01-08
AU5481598A (en) 1998-06-03
DE69719054D1 (de) 2003-03-20
CA2271732A1 (en) 1998-05-22
KR20000053258A (ko) 2000-08-25
AU727328B2 (en) 2000-12-07
ATE232532T1 (de) 2003-02-15
ES2191207T3 (es) 2003-09-01
JP2001503765A (ja) 2001-03-21
PE14099A1 (es) 1999-03-19
DE69719054T2 (de) 2003-11-27
BR9713982A (pt) 2000-05-02
AR010585A1 (es) 2000-06-28
TW438802B (en) 2001-06-07
EP0937078A1 (en) 1999-08-25
EP0937078B1 (en) 2003-02-12

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