TNSN07005A1 - Analogues tetrapeptidiques - Google Patents

Analogues tetrapeptidiques

Info

Publication number
TNSN07005A1
TNSN07005A1 TNP2007000005A TNSN07005A TNSN07005A1 TN SN07005 A1 TNSN07005 A1 TN SN07005A1 TN P2007000005 A TNP2007000005 A TN P2007000005A TN SN07005 A TNSN07005 A TN SN07005A TN SN07005 A1 TNSN07005 A1 TN SN07005A1
Authority
TN
Tunisia
Prior art keywords
tetrapeptitiic
analogs
cancer
compositions
compounds
Prior art date
Application number
TNP2007000005A
Other languages
English (en)
Inventor
Bin Chao
Thomas L Deckwerth
Paul S Furth
Steven D Linton
Alfred P Spada
Brett R Ullman
Michael I Weinhouse
Original Assignee
Idun Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Idun Pharmaceuticals Inc filed Critical Idun Pharmaceuticals Inc
Publication of TNSN07005A1 publication Critical patent/TNSN07005A1/fr

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    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
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    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
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    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
    • C07K5/0806—Tripeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1002—Tetrapeptides with the first amino acid being neutral
    • C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
    • C07K5/1008—Tetrapeptides with the first amino acid being neutral and aliphatic the side chain containing 0 or 1 carbon atoms, i.e. Gly, Ala
    • C—CHEMISTRY; METALLURGY
    • C09—DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09B—ORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES, e.g. PIGMENTS; MORDANTS; LAKES
    • C09B57/00—Other synthetic dyes of known constitution
    • C—CHEMISTRY; METALLURGY
    • C09—DYES; PAINTS; POLISHES; NATURAL RESINS; ADHESIVES; COMPOSITIONS NOT OTHERWISE PROVIDED FOR; APPLICATIONS OF MATERIALS NOT OTHERWISE PROVIDED FOR
    • C09B—ORGANIC DYES OR CLOSELY-RELATED COMPOUNDS FOR PRODUCING DYES, e.g. PIGMENTS; MORDANTS; LAKES
    • C09B57/00—Other synthetic dyes of known constitution
    • C09B57/14—Benzoxanthene dyes; Benzothioxanthene dyes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Abstract

DES COMPOSES, COMPOSITIONS ET METHODES POUR LE TRAITEMENT DE MALADIES HYPERPROLIFERATIVES, TELLES QUE LE CANCER, SONT PROPOSES
TNP2007000005A 2004-07-12 2007-01-11 Analogues tetrapeptidiques TNSN07005A1 (fr)

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US58747104P 2004-07-12 2004-07-12
US68387505P 2005-05-23 2005-05-23
PCT/US2005/024700 WO2006017295A2 (fr) 2004-07-12 2005-07-12 Analogues de tetrapeptide

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KR (1) KR20070043831A (fr)
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CA (1) CA2573644A1 (fr)
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IL (1) IL180677A0 (fr)
MA (1) MA28841B1 (fr)
MX (1) MX2007000490A (fr)
NO (1) NO20070782L (fr)
TN (1) TNSN07005A1 (fr)
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EA200700225A1 (ru) 2008-02-28
IL180677A0 (en) 2008-04-13
EP1773348A4 (fr) 2009-05-20
MX2007000490A (es) 2007-06-11
CR8919A (es) 2007-08-31
NO20070782L (no) 2007-04-02
BRPI0513310A (pt) 2008-05-06
MA28841B1 (fr) 2007-09-03
WO2006017295A3 (fr) 2007-07-12
EP2457895A1 (fr) 2012-05-30
AU2005271831A1 (en) 2006-02-16
WO2006017295A2 (fr) 2006-02-16
ZA200700357B (en) 2008-11-26
CA2573644A1 (fr) 2006-02-16
EP2457896A1 (fr) 2012-05-30
KR20070043831A (ko) 2007-04-25
GB0700629D0 (en) 2007-02-21
US20100190688A1 (en) 2010-07-29
JP2011102312A (ja) 2011-05-26
EP1773348A2 (fr) 2007-04-18
JP2008505976A (ja) 2008-02-28
GB2430935A (en) 2007-04-11

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