SU799669A3 - Способ получени цефалоспоринов - Google Patents

Способ получени цефалоспоринов Download PDF

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Publication number
SU799669A3
SU799669A3 SU772483403A SU2483403A SU799669A3 SU 799669 A3 SU799669 A3 SU 799669A3 SU 772483403 A SU772483403 A SU 772483403A SU 2483403 A SU2483403 A SU 2483403A SU 799669 A3 SU799669 A3 SU 799669A3
Authority
SU
USSR - Soviet Union
Prior art keywords
compounds
alkyl
hydrogen atom
image
pyrazinyl
Prior art date
Application number
SU772483403A
Other languages
English (en)
Russian (ru)
Inventor
Паламидесси Джорджо
Дзарини Франко
Франчески Джованни
Скиоппокасси Джованна
Аркамоне Федерико
Original Assignee
Фармиталия Карло-Эрба С.П.А. (Фирма)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Фармиталия Карло-Эрба С.П.А. (Фирма) filed Critical Фармиталия Карло-Эрба С.П.А. (Фирма)
Application granted granted Critical
Publication of SU799669A3 publication Critical patent/SU799669A3/ru

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D501/00Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/207-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/247-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/36Methylene radicals, substituted by sulfur atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SU772483403A 1976-05-21 1977-05-20 Способ получени цефалоспоринов SU799669A3 (ru)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB21032/76A GB1579532A (en) 1976-05-21 1976-05-21 Cephalosporins

Publications (1)

Publication Number Publication Date
SU799669A3 true SU799669A3 (ru) 1981-01-23

Family

ID=10156029

Family Applications (1)

Application Number Title Priority Date Filing Date
SU772483403A SU799669A3 (ru) 1976-05-21 1977-05-20 Способ получени цефалоспоринов

Country Status (22)

Country Link
US (1) US4148996A (US07534539-20090519-C00280.png)
JP (1) JPS52142093A (US07534539-20090519-C00280.png)
AT (1) AT355719B (US07534539-20090519-C00280.png)
AU (1) AU509448B2 (US07534539-20090519-C00280.png)
BE (1) BE854845A (US07534539-20090519-C00280.png)
CA (1) CA1102790A (US07534539-20090519-C00280.png)
CH (1) CH639095A5 (US07534539-20090519-C00280.png)
CS (1) CS199676B2 (US07534539-20090519-C00280.png)
DE (1) DE2722666C2 (US07534539-20090519-C00280.png)
DK (1) DK216877A (US07534539-20090519-C00280.png)
FR (1) FR2424922A1 (US07534539-20090519-C00280.png)
GB (1) GB1579532A (US07534539-20090519-C00280.png)
GR (1) GR73013B (US07534539-20090519-C00280.png)
HU (1) HU174072B (US07534539-20090519-C00280.png)
IL (1) IL52123A (US07534539-20090519-C00280.png)
NL (1) NL7705262A (US07534539-20090519-C00280.png)
NO (1) NO771744L (US07534539-20090519-C00280.png)
NZ (1) NZ184110A (US07534539-20090519-C00280.png)
SE (1) SE433851B (US07534539-20090519-C00280.png)
SU (1) SU799669A3 (US07534539-20090519-C00280.png)
YU (1) YU123077A (US07534539-20090519-C00280.png)
ZA (1) ZA772859B (US07534539-20090519-C00280.png)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017004077A1 (en) * 2015-06-29 2017-01-05 Duke University Antimicrobial prochelators to target drug-resistant bacteria and methods of making and using the same

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL38099A (en) * 1970-12-17 1976-01-30 Smith Kline French Lab 3-heterocyclyl thiomethylcephalosporins
US4007173A (en) * 1973-05-07 1977-02-08 Smithkline Corporation α-amino-α-(ureidophenyl)acetamidocephalosporins
DE2359544A1 (de) * 1973-11-29 1975-10-30 Hoechst Ag Cephemderivate und verfahren zu ihrer herstellung
US3960849A (en) * 1974-03-13 1976-06-01 E. R. Squibb & Sons, Inc. Amino-1,2,4-oxadiazolyl-3-acetyl cephalosporins
DE2512284A1 (de) * 1974-03-28 1975-10-09 Fujisawa Pharmaceutical Co Cephalosporansaeurederivate, verfahren zu ihrer herstellung und sie enthaltende pharmazeutische mittel

Also Published As

Publication number Publication date
AU2507177A (en) 1978-11-16
SE7705934L (sv) 1977-11-22
CH639095A5 (de) 1983-10-31
HU174072B (hu) 1979-10-28
US4148996A (en) 1979-04-10
GB1579532A (en) 1980-11-19
DK216877A (da) 1977-11-22
IL52123A (en) 1980-11-30
FR2424922B1 (US07534539-20090519-C00280.png) 1983-07-08
CS199676B2 (en) 1980-07-31
DE2722666A1 (de) 1977-12-01
DE2722666C2 (de) 1982-04-15
ZA772859B (en) 1978-04-26
NL7705262A (nl) 1977-11-23
FR2424922A1 (fr) 1979-11-30
NO771744L (no) 1977-11-22
NZ184110A (en) 1979-08-31
IL52123A0 (en) 1977-07-31
JPS52142093A (en) 1977-11-26
SE433851B (sv) 1984-06-18
YU123077A (en) 1982-10-31
CA1102790A (en) 1981-06-09
GR73013B (US07534539-20090519-C00280.png) 1984-01-25
AT355719B (de) 1980-03-25
ATA348977A (de) 1979-08-15
BE854845A (fr) 1977-11-21
AU509448B2 (en) 1980-05-15

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