SK59695A3 - 5,6-dihydro-4h-imidazo£2',1':2,3| imidazo-£4,5,1-ij| quinoline derivatives and 4,5-dihydroimidazole £1,2-a| pyrolo-£1,2,3-cd| benzimidazole derivatives, method of their preparation and pharmaceutical agents containing them - Google Patents

5,6-dihydro-4h-imidazo£2',1':2,3| imidazo-£4,5,1-ij| quinoline derivatives and 4,5-dihydroimidazole £1,2-a| pyrolo-£1,2,3-cd| benzimidazole derivatives, method of their preparation and pharmaceutical agents containing them Download PDF

Info

Publication number
SK59695A3
SK59695A3 SK596-95A SK59695A SK59695A3 SK 59695 A3 SK59695 A3 SK 59695A3 SK 59695 A SK59695 A SK 59695A SK 59695 A3 SK59695 A3 SK 59695A3
Authority
SK
Slovakia
Prior art keywords
formula
imidazo
group
mixture
dihydro
Prior art date
Application number
SK596-95A
Other languages
English (en)
Slovak (sk)
Inventor
Pascal George
Mireille Sevrin
Michel Peynot
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of SK59695A3 publication Critical patent/SK59695A3/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/16—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/16—Peri-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
SK596-95A 1994-05-10 1995-05-09 5,6-dihydro-4h-imidazo£2',1':2,3| imidazo-£4,5,1-ij| quinoline derivatives and 4,5-dihydroimidazole £1,2-a| pyrolo-£1,2,3-cd| benzimidazole derivatives, method of their preparation and pharmaceutical agents containing them SK59695A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9405715A FR2719843B1 (fr) 1994-05-10 1994-05-10 Dérivés de 5,6-dihydro-4h-imidazo [2',1':2,3] imidazo-[4,5,1-ij] quinoléine et de 4,5-dihydroimidazo [1,2-a] pyrrolo-[1,2,3-cd] benzimidazole, leur préparation et leur application en thérapeutique.

Publications (1)

Publication Number Publication Date
SK59695A3 true SK59695A3 (en) 1995-12-06

Family

ID=9463058

Family Applications (1)

Application Number Title Priority Date Filing Date
SK596-95A SK59695A3 (en) 1994-05-10 1995-05-09 5,6-dihydro-4h-imidazo£2',1':2,3| imidazo-£4,5,1-ij| quinoline derivatives and 4,5-dihydroimidazole £1,2-a| pyrolo-£1,2,3-cd| benzimidazole derivatives, method of their preparation and pharmaceutical agents containing them

Country Status (18)

Country Link
US (1) US5512590A (hu)
EP (1) EP0682025A1 (hu)
JP (1) JPH0853450A (hu)
KR (1) KR950032193A (hu)
CN (1) CN1115761A (hu)
AU (1) AU1793595A (hu)
CA (1) CA2148951A1 (hu)
CZ (1) CZ119495A3 (hu)
FI (1) FI952249A (hu)
FR (1) FR2719843B1 (hu)
HU (1) HUT72666A (hu)
IL (1) IL113672A (hu)
NO (1) NO951811L (hu)
NZ (1) NZ272089A (hu)
PL (1) PL308517A1 (hu)
RU (1) RU95107157A (hu)
SK (1) SK59695A3 (hu)
ZA (1) ZA953750B (hu)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0120345D0 (en) * 2001-08-21 2001-10-17 Merck Sharp & Dohme Therapeutic agents
CA2509561A1 (en) * 2002-12-18 2004-07-15 Mallinckrodt Inc. Synthesis of heteroaryl acetamides
AU2005262622A1 (en) * 2004-06-22 2006-01-19 Mallinckrodt Inc. Synthesis of heteroaryl acetamides from reaction mixtures having reduced water content
CA2604887A1 (en) * 2005-04-07 2006-10-19 Hythiam, Inc. Improved methods of and compositions for the prevention of anxiety, substance abuse, and dependence
AR053902A1 (es) 2005-06-14 2007-05-23 Schering Corp Inhibidores de aspartil proteasa heterociclicos macrociclicos
WO2021067682A1 (en) * 2019-10-03 2021-04-08 Dana-Farber Cancer Institute, Inc. Tricyclic kinase inhibitors and uses thereof
EP4146639A1 (en) 2020-05-06 2023-03-15 Ajax Therapeutics, Inc. 6-heteroaryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors
TW202241889A (zh) 2020-12-23 2022-11-01 美商雅捷可斯治療公司 作為ｊａｋ２抑制劑之６－雜芳基氧基苯并咪唑及氮雜苯并咪唑
WO2023086319A1 (en) 2021-11-09 2023-05-19 Ajax Therapeutics, Inc. 6-he tero aryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3732243A (en) * 1970-06-23 1973-05-08 Sankyo Co 2-(p-bromophenyl)-9-dimethyl-amino-propyl-9h-imidazo(1,2-a)benzimidazole
FR2568879B1 (fr) * 1984-08-07 1986-12-12 Synthelabo Imidazo(1,2-a)quinolines, leur preparation et leur application en therapeutique
FR2593817B1 (fr) * 1986-01-31 1988-04-15 Synthelabo Derives de tetrahydro-5,6,7,8 imidazo(1,2-a)pyridine, leur preparation et leur application en therapeutique
ATE117688T1 (de) * 1989-06-09 1995-02-15 Upjohn Co Heterozyklische amine mit zns-wirksamkeit.
EP0607076A1 (fr) * 1993-01-15 1994-07-20 Synthelabo Dérivés de 9h-imidazo 1,2-a benzimidazole-3-acétamide à activité GABA

Also Published As

Publication number Publication date
RU95107157A (ru) 1997-03-20
IL113672A0 (en) 1995-08-31
CN1115761A (zh) 1996-01-31
KR950032193A (ko) 1995-12-20
PL308517A1 (en) 1995-11-13
ZA953750B (en) 1996-04-02
JPH0853450A (ja) 1996-02-27
EP0682025A1 (fr) 1995-11-15
FR2719843B1 (fr) 1996-06-07
FI952249A (fi) 1995-11-11
NO951811D0 (no) 1995-05-09
IL113672A (en) 1997-11-20
AU1793595A (en) 1995-11-16
FI952249A0 (fi) 1995-05-09
US5512590A (en) 1996-04-30
CZ119495A3 (en) 1995-12-13
FR2719843A1 (fr) 1995-11-17
CA2148951A1 (en) 1995-11-11
HUT72666A (en) 1996-05-28
NO951811L (no) 1995-11-13
NZ272089A (en) 1996-07-26

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