FI952249A - 5,6-dihydro-4H-imidatso/2'1':2,3/imidatso/4,5,1-ij/kinoliini ja 4,5-dihydroimidatso/1,2-a/pyrrolo/1,2,3-cd/-bentsimidatsolijohdannaiset, niiden valmistus ja terapeuttinen käyttö - Google Patents

5,6-dihydro-4H-imidatso/2'1':2,3/imidatso/4,5,1-ij/kinoliini ja 4,5-dihydroimidatso/1,2-a/pyrrolo/1,2,3-cd/-bentsimidatsolijohdannaiset, niiden valmistus ja terapeuttinen käyttö Download PDF

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Publication number
FI952249A
FI952249A FI952249A FI952249A FI952249A FI 952249 A FI952249 A FI 952249A FI 952249 A FI952249 A FI 952249A FI 952249 A FI952249 A FI 952249A FI 952249 A FI952249 A FI 952249A
Authority
FI
Finland
Prior art keywords
imidazo
dihydroimidazo
pyrrolo
quinoline
dihydro
Prior art date
Application number
FI952249A
Other languages
English (en)
Swedish (sv)
Other versions
FI952249A0 (fi
Inventor
Pascal George
Mireille Sevrin
Michel Peynot
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of FI952249A0 publication Critical patent/FI952249A0/fi
Publication of FI952249A publication Critical patent/FI952249A/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/16—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/16—Peri-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI952249A 1994-05-10 1995-05-09 5,6-dihydro-4H-imidatso/2'1':2,3/imidatso/4,5,1-ij/kinoliini ja 4,5-dihydroimidatso/1,2-a/pyrrolo/1,2,3-cd/-bentsimidatsolijohdannaiset, niiden valmistus ja terapeuttinen käyttö FI952249A (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9405715A FR2719843B1 (fr) 1994-05-10 1994-05-10 Dérivés de 5,6-dihydro-4h-imidazo [2',1':2,3] imidazo-[4,5,1-ij] quinoléine et de 4,5-dihydroimidazo [1,2-a] pyrrolo-[1,2,3-cd] benzimidazole, leur préparation et leur application en thérapeutique.

Publications (2)

Publication Number Publication Date
FI952249A0 FI952249A0 (fi) 1995-05-09
FI952249A true FI952249A (fi) 1995-11-11

Family

ID=9463058

Family Applications (1)

Application Number Title Priority Date Filing Date
FI952249A FI952249A (fi) 1994-05-10 1995-05-09 5,6-dihydro-4H-imidatso/2'1':2,3/imidatso/4,5,1-ij/kinoliini ja 4,5-dihydroimidatso/1,2-a/pyrrolo/1,2,3-cd/-bentsimidatsolijohdannaiset, niiden valmistus ja terapeuttinen käyttö

Country Status (18)

Country Link
US (1) US5512590A (fi)
EP (1) EP0682025A1 (fi)
JP (1) JPH0853450A (fi)
KR (1) KR950032193A (fi)
CN (1) CN1115761A (fi)
AU (1) AU1793595A (fi)
CA (1) CA2148951A1 (fi)
CZ (1) CZ119495A3 (fi)
FI (1) FI952249A (fi)
FR (1) FR2719843B1 (fi)
HU (1) HUT72666A (fi)
IL (1) IL113672A (fi)
NO (1) NO951811L (fi)
NZ (1) NZ272089A (fi)
PL (1) PL308517A1 (fi)
RU (1) RU95107157A (fi)
SK (1) SK59695A3 (fi)
ZA (1) ZA953750B (fi)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0120345D0 (en) * 2001-08-21 2001-10-17 Merck Sharp & Dohme Therapeutic agents
AU2003297153B2 (en) * 2002-12-18 2010-06-10 Mallinckrodt Inc. Synthesis of heteroaryl acetamides
CN1972939A (zh) * 2004-06-22 2007-05-30 马林克罗特公司 由具有减少的水含量的反应混合物合成杂芳基乙酰胺
EP1868593A2 (en) * 2005-04-07 2007-12-26 Hythiam, Inc. Improved methods of and compositions for the prevention of anxiety, substance abuse, and dependence
MX2007016185A (es) 2005-06-14 2008-03-07 Schering Corp Inhibidores de aspartil proteasa heterociclicos macrociclicos.
CA3156828A1 (en) * 2019-10-03 2021-04-08 Dana-Farber Cancer Institute, Inc. Tricyclic kinase inhibitors and uses thereof
JP2023525047A (ja) 2020-05-06 2023-06-14 エイジャックス セラピューティクス， インコーポレイテッド Ｊａｋ２阻害薬としての６－ヘテロアリールオキシベンゾイミダゾール及びアザベンゾイミダゾール
CA3234638A1 (en) 2021-11-09 2023-05-19 Ajax Therapeutics, Inc. 6-heteroaryloxy benzimidazoles and azabenzimidazoles as jak2 inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3732243A (en) * 1970-06-23 1973-05-08 Sankyo Co 2-(p-bromophenyl)-9-dimethyl-amino-propyl-9h-imidazo(1,2-a)benzimidazole
FR2568879B1 (fr) * 1984-08-07 1986-12-12 Synthelabo Imidazo(1,2-a)quinolines, leur preparation et leur application en therapeutique
FR2593817B1 (fr) * 1986-01-31 1988-04-15 Synthelabo Derives de tetrahydro-5,6,7,8 imidazo(1,2-a)pyridine, leur preparation et leur application en therapeutique
DE69016430T2 (de) * 1989-06-09 1995-06-01 Upjohn Co Heterozyklische amine mit zns-wirksamkeit.
EP0607076A1 (fr) * 1993-01-15 1994-07-20 Synthelabo Dérivés de 9h-imidazo 1,2-a benzimidazole-3-acétamide à activité GABA

Also Published As

Publication number Publication date
NZ272089A (en) 1996-07-26
IL113672A0 (en) 1995-08-31
RU95107157A (ru) 1997-03-20
KR950032193A (ko) 1995-12-20
EP0682025A1 (fr) 1995-11-15
NO951811L (no) 1995-11-13
FR2719843A1 (fr) 1995-11-17
HUT72666A (en) 1996-05-28
PL308517A1 (en) 1995-11-13
FR2719843B1 (fr) 1996-06-07
CA2148951A1 (en) 1995-11-11
JPH0853450A (ja) 1996-02-27
AU1793595A (en) 1995-11-16
SK59695A3 (en) 1995-12-06
CZ119495A3 (en) 1995-12-13
US5512590A (en) 1996-04-30
FI952249A0 (fi) 1995-05-09
IL113672A (en) 1997-11-20
NO951811D0 (no) 1995-05-09
CN1115761A (zh) 1996-01-31
ZA953750B (en) 1996-04-02

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