SK19062001A3 - Spôsob prípravy (-)-(1S,4R) N-chráneného 4-amino-2-cyklopentén-1-karboxylát esterov - Google Patents

Spôsob prípravy (-)-(1S,4R) N-chráneného 4-amino-2-cyklopentén-1-karboxylát esterov Download PDF

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Publication number
SK19062001A3
SK19062001A3 SK1906-2001A SK19062001A SK19062001A3 SK 19062001 A3 SK19062001 A3 SK 19062001A3 SK 19062001 A SK19062001 A SK 19062001A SK 19062001 A3 SK19062001 A3 SK 19062001A3
Authority
SK
Slovakia
Prior art keywords
formula
compound
tertiary amine
tartaric acid
methyl
Prior art date
Application number
SK1906-2001A
Other languages
English (en)
Slovak (sk)
Inventor
Max Rey
Gregor Welti
Cynthia Maryanoff
Original Assignee
Biocryst Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biocryst Pharmaceuticals, Inc. filed Critical Biocryst Pharmaceuticals, Inc.
Publication of SK19062001A3 publication Critical patent/SK19062001A3/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C269/00—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
    • C07C269/04—Preparation of derivatives of carbamic acid, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups from amines with formation of carbamate groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/46—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • C07C229/48—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton with amino groups and carboxyl groups bound to carbon atoms of the same non-condensed ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/10—Systems containing only non-condensed rings with a five-membered ring the ring being unsaturated
SK1906-2001A 1999-06-28 2000-06-09 Spôsob prípravy (-)-(1S,4R) N-chráneného 4-amino-2-cyklopentén-1-karboxylát esterov SK19062001A3 (sk)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14129299P 1999-06-28 1999-06-28
PCT/US2000/015969 WO2001001569A2 (en) 1999-06-28 2000-06-09 Process for preparing (-)-(1s,4r) n-protected 4-amino-2-cyclopentene-1-carboxylate esters

Publications (1)

Publication Number Publication Date
SK19062001A3 true SK19062001A3 (sk) 2003-03-04

Family

ID=22495050

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1906-2001A SK19062001A3 (sk) 1999-06-28 2000-06-09 Spôsob prípravy (-)-(1S,4R) N-chráneného 4-amino-2-cyklopentén-1-karboxylát esterov

Country Status (16)

Country Link
US (1) US6495711B2 (ja)
EP (1) EP1206443A2 (ja)
JP (1) JP4532801B2 (ja)
KR (1) KR20020013937A (ja)
CN (1) CN1358170A (ja)
AR (1) AR024493A1 (ja)
AU (1) AU5479700A (ja)
BR (1) BR0011767A (ja)
CA (1) CA2377801A1 (ja)
CZ (1) CZ20014656A3 (ja)
HU (1) HUP0201873A3 (ja)
IL (1) IL147243A0 (ja)
NO (1) NO20016390L (ja)
PL (1) PL352675A1 (ja)
SK (1) SK19062001A3 (ja)
WO (1) WO2001001569A2 (ja)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101538228B (zh) * 2008-03-21 2012-05-30 北京普世康医药技术有限公司 抗流感和禽流感病毒药物化合物帕拉米韦的合成方法
CN102863359B (zh) * 2012-05-16 2014-05-07 常州制药厂有限公司 一种抗流感药物的合成方法
WO2016067182A2 (en) * 2014-10-27 2016-05-06 Granules India Limited Process for the preparation of amino alcohol derivatives or salts thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8815265D0 (en) 1988-06-27 1988-08-03 Wellcome Found Therapeutic nucleosides
DK0424064T3 (da) 1989-10-16 1995-06-26 Chiroscience Ltd Chirale azabicycloheptanoner og fremgangsmåde til fremstilling deraf
JPH06116217A (ja) * 1992-10-02 1994-04-26 Kuraray Co Ltd （±）−シス−４−アミノシクロペント−２−エンカルボン酸誘導体の光学分割法
US5399580A (en) * 1993-03-08 1995-03-21 Burroughs Wellcome Co. Therapeutic nucleosides-uses
US6410594B1 (en) 1996-06-14 2002-06-25 Biocryst Pharmaceuticals, Inc. Substituted cyclopentane compounds useful as neuraminidase inhibitors
GB9625455D0 (en) * 1996-12-07 1997-01-22 Glaxo Group Ltd Process for resolving mixtures of carbocyclic steroisomers
ZA9811595B (en) * 1997-12-17 2000-06-19 Biocryst Pharm Inc Substituted cyclopentane and cyclopentene compounds useful as neuraminidase inhibitors.

Also Published As

Publication number Publication date
HUP0201873A2 (en) 2002-10-28
JP2003503368A (ja) 2003-01-28
NO20016390D0 (no) 2001-12-27
US6495711B2 (en) 2002-12-17
AU5479700A (en) 2001-01-31
KR20020013937A (ko) 2002-02-21
EP1206443A2 (en) 2002-05-22
IL147243A0 (en) 2002-08-14
PL352675A1 (en) 2003-09-08
AR024493A1 (es) 2002-10-02
NO20016390L (no) 2002-02-19
WO2001001569A2 (en) 2001-01-04
JP4532801B2 (ja) 2010-08-25
CN1358170A (zh) 2002-07-10
WO2001001569A3 (en) 2001-05-03
HUP0201873A3 (en) 2003-03-28
CA2377801A1 (en) 2001-01-04
BR0011767A (pt) 2002-04-23
CZ20014656A3 (cs) 2002-11-13
US20020052524A1 (en) 2002-05-02

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