SK125693A3 - Cephalosporin derivatives - Google Patents

Cephalosporin derivatives Download PDF

Info

Publication number
SK125693A3
SK125693A3 SK1256-93A SK125693A SK125693A3 SK 125693 A3 SK125693 A3 SK 125693A3 SK 125693 A SK125693 A SK 125693A SK 125693 A3 SK125693 A3 SK 125693A3
Authority
SK
Slovakia
Prior art keywords
formula
compound
pharmaceutically acceptable
esters
salts
Prior art date
Application number
SK1256-93A
Other languages
English (en)
Slovak (sk)
Inventor
Scott L Dax
Dennis D Keith
Pamela L Rossman
Chung-Chen Wei
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of SK125693A3 publication Critical patent/SK125693A3/sk

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
    • C07D501/26—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
    • C07D501/34—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by carboxylic acids containing hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SK1256-93A 1992-11-12 1993-11-10 Cephalosporin derivatives SK125693A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US97625092A 1992-11-12 1992-11-12
US97624892A 1992-11-12 1992-11-12

Publications (1)

Publication Number Publication Date
SK125693A3 true SK125693A3 (en) 1994-09-07

Family

ID=27130586

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1256-93A SK125693A3 (en) 1992-11-12 1993-11-10 Cephalosporin derivatives

Country Status (19)

Country Link
EP (1) EP0597303A2 (no)
JP (1) JPH06199868A (no)
KR (1) KR940011470A (no)
CN (1) CN1141922A (no)
AU (1) AU5051793A (no)
BG (1) BG98208A (no)
BR (1) BR9304699A (no)
CA (1) CA2108609A1 (no)
CZ (1) CZ239893A3 (no)
FI (1) FI935025A (no)
HU (1) HUT65717A (no)
IS (1) IS4093A (no)
LV (1) LV10277A (no)
MX (1) MX9306985A (no)
NO (1) NO934078D0 (no)
PL (1) PL301024A1 (no)
SI (1) SI9300555A (no)
SK (1) SK125693A3 (no)
UY (1) UY23672A1 (no)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HUT49889A (en) * 1988-03-31 1989-11-28 Hoffmann La Roche Process for producing acyl derivatives
EP0366189A3 (en) * 1988-10-24 1992-01-02 Norwich Eaton Pharmaceuticals, Inc. Novel antimicrobial lactam-quinolones

Also Published As

Publication number Publication date
PL301024A1 (en) 1994-05-16
CA2108609A1 (en) 1994-05-13
NO934078L (no) 1994-05-13
BR9304699A (pt) 1994-06-14
FI935025A0 (fi) 1993-11-12
CZ239893A3 (en) 1994-06-15
HUT65717A (en) 1994-07-28
AU5051793A (en) 1994-05-26
LV10277A (lv) 1994-10-20
CN1141922A (zh) 1997-02-05
KR940011470A (ko) 1994-06-21
JPH06199868A (ja) 1994-07-19
FI935025A (fi) 1994-05-13
BG98208A (en) 1994-05-27
MX9306985A (es) 1995-01-31
EP0597303A3 (no) 1994-08-03
NO934078D0 (no) 1993-11-11
IS4093A (is) 1994-05-13
SI9300555A (en) 1994-06-30
EP0597303A2 (en) 1994-05-18
UY23672A1 (es) 1994-05-06

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