SI2454266T1 - Citratna sol 9e-15-(2-pirolidin-1-il-etoksi)-7,12,25-trioksa-19,21,24-triaza-tetra- ciklo (18.3.1.1(2,5).1(14)18)heksakosa-1(24),2,4,9,14,16,18(26),20,22- nonaena - Google Patents
Citratna sol 9e-15-(2-pirolidin-1-il-etoksi)-7,12,25-trioksa-19,21,24-triaza-tetra- ciklo (18.3.1.1(2,5).1(14)18)heksakosa-1(24),2,4,9,14,16,18(26),20,22- nonaenaInfo
- Publication number
- SI2454266T1 SI2454266T1 SI201030347T SI201030347T SI2454266T1 SI 2454266 T1 SI2454266 T1 SI 2454266T1 SI 201030347 T SI201030347 T SI 201030347T SI 201030347 T SI201030347 T SI 201030347T SI 2454266 T1 SI2454266 T1 SI 2454266T1
- Authority
- SI
- Slovenia
- Prior art keywords
- chexacosa
- nonaene
- trioxa
- triaza
- pyrrolidin
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/18—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US22560909P | 2009-07-15 | 2009-07-15 | |
PCT/SG2010/000265 WO2011008172A1 (en) | 2009-07-15 | 2010-07-14 | 9e-15-(2-pyrrolidin-1-yl-ethoxy)-7,12,25-trioxa-19,21,24-triaza- tetracyclo[18.3.1.1(2,5).1(14)18)]hexacosa-1(24),2,4,9,14,16,18(26),20,22-nonaene citrate salt |
EP10737645.1A EP2454266B1 (en) | 2009-07-15 | 2010-07-14 | 9e-15-(2-pyrrolidin-1-yl-ethoxy)-7,12,25-trioxa-19,21,24-triaza- tetracyclo[18.3.1.1(2,5).1(14)18)]hexacosa-1(24),2,4,9,14,16,18(26),20,22-nonaene citrate salt |
Publications (1)
Publication Number | Publication Date |
---|---|
SI2454266T1 true SI2454266T1 (sl) | 2013-10-30 |
Family
ID=42790728
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SI201030347T SI2454266T1 (sl) | 2009-07-15 | 2010-07-14 | Citratna sol 9e-15-(2-pirolidin-1-il-etoksi)-7,12,25-trioksa-19,21,24-triaza-tetra- ciklo (18.3.1.1(2,5).1(14)18)heksakosa-1(24),2,4,9,14,16,18(26),20,22- nonaena |
Country Status (19)
Country | Link |
---|---|
US (1) | US9062074B2 (sl) |
EP (1) | EP2454266B1 (sl) |
JP (2) | JP6013911B2 (sl) |
CN (1) | CN102762577B (sl) |
AR (2) | AR077483A1 (sl) |
BR (1) | BR112012000750B1 (sl) |
CA (1) | CA2768210C (sl) |
DK (1) | DK2454266T3 (sl) |
ES (1) | ES2429525T3 (sl) |
HK (1) | HK1178159A1 (sl) |
HR (1) | HRP20130941T1 (sl) |
MX (1) | MX2012000680A (sl) |
PL (1) | PL2454266T3 (sl) |
PT (1) | PT2454266E (sl) |
RU (1) | RU2543721C2 (sl) |
SI (1) | SI2454266T1 (sl) |
SM (1) | SMT201300112B (sl) |
TW (1) | TWI537276B (sl) |
WO (1) | WO2011008172A1 (sl) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN113559075A (zh) | 2014-11-17 | 2021-10-29 | 康泰科思特生物制药公司 | 奥那司酮延长释放组合物和方法 |
BR112018005999A2 (pt) | 2015-09-25 | 2019-01-08 | Context Biopharma Inc | métodos para a produção de intermediários de onapristona |
AU2016370499B2 (en) | 2015-12-15 | 2022-06-30 | Context Biopharma Inc. | Amorphous onapristone compositions and methods of making the same |
US20180148471A1 (en) | 2016-11-30 | 2018-05-31 | Arno Therapeutics, Inc. | Methods for onapristone synthesis dehydration and deprotection |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MY110603A (en) * | 1993-05-27 | 1998-08-29 | Novartis Ag | Tetrahydropyran derivatives |
WO2004078682A2 (en) * | 2003-03-05 | 2004-09-16 | Irm Llc | Cyclic compounds and compositions as protein kinase inhibitors |
WO2007058627A1 (en) * | 2005-11-16 | 2007-05-24 | S*Bio Pte Ltd | Oxygen linked pyrimidine derivatives |
-
2010
- 2010-07-14 BR BR112012000750-5A patent/BR112012000750B1/pt active IP Right Grant
- 2010-07-14 CA CA2768210A patent/CA2768210C/en active Active
- 2010-07-14 ES ES10737645T patent/ES2429525T3/es active Active
- 2010-07-14 PL PL10737645T patent/PL2454266T3/pl unknown
- 2010-07-14 JP JP2012520571A patent/JP6013911B2/ja active Active
- 2010-07-14 SI SI201030347T patent/SI2454266T1/sl unknown
- 2010-07-14 DK DK10737645.1T patent/DK2454266T3/da active
- 2010-07-14 MX MX2012000680A patent/MX2012000680A/es active IP Right Grant
- 2010-07-14 US US13/384,139 patent/US9062074B2/en active Active
- 2010-07-14 RU RU2012105044/04A patent/RU2543721C2/ru active
- 2010-07-14 WO PCT/SG2010/000265 patent/WO2011008172A1/en active Application Filing
- 2010-07-14 EP EP10737645.1A patent/EP2454266B1/en active Active
- 2010-07-14 CN CN201080032627.5A patent/CN102762577B/zh active Active
- 2010-07-14 PT PT107376451T patent/PT2454266E/pt unknown
- 2010-07-15 TW TW099123331A patent/TWI537276B/zh active
- 2010-07-15 AR ARP100102594A patent/AR077483A1/es not_active Application Discontinuation
-
2013
- 2013-04-29 HK HK13105191.1A patent/HK1178159A1/xx unknown
- 2013-10-04 SM SM201300112T patent/SMT201300112B/xx unknown
- 2013-10-07 HR HRP20130941AT patent/HRP20130941T1/hr unknown
-
2015
- 2015-05-07 JP JP2015094972A patent/JP2015164941A/ja active Pending
-
2019
- 2019-08-05 AR ARP190102219A patent/AR114987A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
BR112012000750A8 (pt) | 2018-02-06 |
ES2429525T3 (es) | 2013-11-15 |
MX2012000680A (es) | 2012-02-28 |
JP2012533539A (ja) | 2012-12-27 |
PL2454266T3 (pl) | 2014-01-31 |
AR114987A2 (es) | 2020-11-11 |
EP2454266B1 (en) | 2013-07-10 |
BR112012000750B1 (pt) | 2021-05-25 |
US9062074B2 (en) | 2015-06-23 |
CA2768210C (en) | 2017-08-15 |
AR077483A1 (es) | 2011-08-31 |
RU2543721C2 (ru) | 2015-03-10 |
TW201107336A (en) | 2011-03-01 |
TWI537276B (zh) | 2016-06-11 |
CN102762577B (zh) | 2015-01-07 |
WO2011008172A1 (en) | 2011-01-20 |
RU2012105044A (ru) | 2013-08-20 |
DK2454266T3 (da) | 2013-09-08 |
HK1178159A1 (en) | 2013-09-06 |
CA2768210A1 (en) | 2011-01-20 |
BR112012000750A2 (pt) | 2016-08-09 |
CN102762577A (zh) | 2012-10-31 |
US20120196876A1 (en) | 2012-08-02 |
PT2454266E (pt) | 2013-10-10 |
SMT201300112B (it) | 2013-11-08 |
EP2454266A1 (en) | 2012-05-23 |
JP2015164941A (ja) | 2015-09-17 |
JP6013911B2 (ja) | 2016-10-25 |
HRP20130941T1 (hr) | 2013-11-08 |
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