SI1305318T1 - Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo (2,1-b) (1,3)benzothiazepines - Google Patents

Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo (2,1-b) (1,3)benzothiazepines

Info

Publication number
SI1305318T1
SI1305318T1 SI200130086T SI200130086T SI1305318T1 SI 1305318 T1 SI1305318 T1 SI 1305318T1 SI 200130086 T SI200130086 T SI 200130086T SI 200130086 T SI200130086 T SI 200130086T SI 1305318 T1 SI1305318 T1 SI 1305318T1
Authority
SI
Slovenia
Prior art keywords
preparation
sub
benzothiazepines
dihydropyrrolo
amino substituted
Prior art date
Application number
SI200130086T
Other languages
English (en)
Slovenian (sl)
Inventor
Patrizia Sigma-Tau Ind.Pharm.Riunite Spa MINETTI
D Sigma-Tau Ind.Pharma.Riunite S.p.A MASTROIANNI
Original Assignee
Sigma-Tau
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sigma-Tau filed Critical Sigma-Tau
Publication of SI1305318T1 publication Critical patent/SI1305318T1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • General Health & Medical Sciences (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
SI200130086T 2000-08-01 2001-07-20 Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo (2,1-b) (1,3)benzothiazepines SI1305318T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT2000RM000434A IT1317886B1 (it) 2000-08-01 2000-08-01 Procedimento per la preparazione di 9,10-diidro-pirrolo (2,1-b)(1,3)benzotiazepine 9-ammino sostituite.
PCT/IT2001/000391 WO2002010174A1 (en) 2000-08-01 2001-07-20 Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo [2,1-b][1,3]benzotiazepines

Publications (1)

Publication Number Publication Date
SI1305318T1 true SI1305318T1 (en) 2004-08-31

Family

ID=11454867

Family Applications (1)

Application Number Title Priority Date Filing Date
SI200130086T SI1305318T1 (en) 2000-08-01 2001-07-20 Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo (2,1-b) (1,3)benzothiazepines

Country Status (22)

Country Link
US (1) US7078521B2 (cs)
EP (1) EP1305318B1 (cs)
JP (1) JP2004505089A (cs)
KR (1) KR100801269B1 (cs)
CN (1) CN100354281C (cs)
AT (1) ATE261977T1 (cs)
AU (2) AU7768701A (cs)
BR (1) BR0112974A (cs)
CA (1) CA2415050C (cs)
CZ (1) CZ294502B6 (cs)
DE (1) DE60102385T2 (cs)
DK (1) DK1305318T3 (cs)
ES (1) ES2215922T3 (cs)
HU (2) HUP0301647A3 (cs)
IT (1) IT1317886B1 (cs)
MX (1) MXPA03000917A (cs)
PL (1) PL202400B1 (cs)
PT (1) PT1305318E (cs)
SI (1) SI1305318T1 (cs)
SK (1) SK287190B6 (cs)
TR (1) TR200400821T4 (cs)
WO (1) WO2002010174A1 (cs)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1301965B1 (it) * 1998-07-28 2000-07-20 Sigma Tau Ind Farmaceuti Pirrolo (2,1-b)(1,3) benzotiazepine con attivita' antipsicoticaatipica.

Also Published As

Publication number Publication date
ITRM20000434A0 (it) 2000-08-01
DE60102385T2 (de) 2005-02-17
PL202400B1 (pl) 2009-06-30
PT1305318E (pt) 2004-08-31
ITRM20000434A1 (it) 2002-02-01
HUP0301647A3 (en) 2009-08-28
CZ200311A3 (cs) 2003-05-14
CN100354281C (zh) 2007-12-12
HUP0301647A2 (hu) 2003-11-28
ATE261977T1 (de) 2004-04-15
CZ294502B6 (cs) 2005-01-12
DE60102385D1 (de) 2004-04-22
KR20030013525A (ko) 2003-02-14
SK1262003A3 (en) 2004-03-02
AU2001277687B2 (en) 2006-10-05
CA2415050A1 (en) 2002-02-07
US7078521B2 (en) 2006-07-18
DK1305318T3 (da) 2004-07-26
BR0112974A (pt) 2003-07-08
WO2002010174A1 (en) 2002-02-07
US20030181437A1 (en) 2003-09-25
EP1305318B1 (en) 2004-03-17
HUP0301648A2 (hu) 2003-08-28
PL365009A1 (en) 2004-12-27
IT1317886B1 (it) 2003-07-15
MXPA03000917A (es) 2003-09-05
JP2004505089A (ja) 2004-02-19
ES2215922T3 (es) 2004-10-16
HUP0301648A3 (en) 2004-06-28
CN1443188A (zh) 2003-09-17
TR200400821T4 (tr) 2004-07-21
AU7768701A (en) 2002-02-13
KR100801269B1 (ko) 2008-02-04
EP1305318A1 (en) 2003-05-02
CA2415050C (en) 2009-10-27
SK287190B6 (sk) 2010-02-08
HK1059775A1 (en) 2004-07-16

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