SG78188G - Carboxyalkyl dipeptides,processes for their production and pharmaceutical compositions containing them - Google Patents

Carboxyalkyl dipeptides,processes for their production and pharmaceutical compositions containing them

Info

Publication number
SG78188G
SG78188G SG781/88A SG78188A SG78188G SG 78188 G SG78188 G SG 78188G SG 781/88 A SG781/88 A SG 781/88A SG 78188 A SG78188 A SG 78188A SG 78188 G SG78188 G SG 78188G
Authority
SG
Singapore
Prior art keywords
lower alkyl
chem
bridge
hydrogen
alkoxy
Prior art date
Application number
SG781/88A
Other languages
English (en)
Original Assignee
Schering Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26895254&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG78188(G) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Corp filed Critical Schering Corp
Publication of SG78188G publication Critical patent/SG78188G/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Saccharide Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Apparatus For Disinfection Or Sterilisation (AREA)
SG781/88A 1980-10-23 1988-11-21 Carboxyalkyl dipeptides,processes for their production and pharmaceutical compositions containing them SG78188G (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US19988680A 1980-10-23 1980-10-23
US25848481A 1981-04-28 1981-04-28

Publications (1)

Publication Number Publication Date
SG78188G true SG78188G (en) 1989-03-23

Family

ID=26895254

Family Applications (1)

Application Number Title Priority Date Filing Date
SG781/88A SG78188G (en) 1980-10-23 1988-11-21 Carboxyalkyl dipeptides,processes for their production and pharmaceutical compositions containing them

Country Status (28)

Country Link
US (2) US4818749A (ko)
EP (1) EP0050800B2 (ko)
JP (1) JPH01163197A (ko)
KR (1) KR880001843B1 (ko)
AT (1) ATE20469T1 (ko)
AU (1) AU554362B2 (ko)
CA (1) CA1341206C (ko)
CY (1) CY1469A (ko)
DE (2) DE3174844D1 (ko)
DK (1) DK161523C (ko)
ES (1) ES506414A0 (ko)
FI (1) FI83222C (ko)
GR (1) GR75059B (ko)
HK (1) HK36189A (ko)
HU (1) HU193146B (ko)
IE (1) IE53802B1 (ko)
IL (1) IL64085A (ko)
KE (1) KE3845A (ko)
LU (1) LU88621I2 (ko)
MA (1) MA19309A1 (ko)
MY (1) MY8700683A (ko)
NL (1) NL940001I2 (ko)
NO (2) NO164983C (ko)
NZ (1) NZ198702A (ko)
OA (1) OA06929A (ko)
PH (1) PH21916A (ko)
PT (1) PT73861B (ko)
SG (1) SG78188G (ko)

Families Citing this family (144)

* Cited by examiner, † Cited by third party
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GR75059B (ko) 1984-07-13
NO813546L (no) 1982-04-26
HK36189A (en) 1989-05-12
KE3845A (en) 1989-04-07
FI83222C (sv) 1991-06-10
DK161523C (da) 1991-12-23
CA1341206C (en) 2001-03-20
MA19309A1 (fr) 1982-07-01
PT73861A (en) 1981-11-01
OA06929A (fr) 1983-05-31
AU554362B2 (en) 1986-08-21
JPH01163197A (ja) 1989-06-27
PT73861B (en) 1985-11-12
ES8308838A1 (es) 1983-10-01
CY1469A (en) 1989-07-21
EP0050800A1 (en) 1982-05-05
DK161523B (da) 1991-07-15
IE53802B1 (en) 1989-03-01
KR830007519A (ko) 1983-10-21
MY8700683A (en) 1987-12-31
DK462581A (da) 1982-04-24
FI83222B (fi) 1991-02-28
US4831157A (en) 1989-05-16
US4818749A (en) 1989-04-04
IL64085A (en) 1986-12-31
AU7661481A (en) 1982-04-29
EP0050800B2 (en) 1995-06-07
NO164983B (no) 1990-08-27
NZ198702A (en) 1985-08-30
LU88621I2 (fr) 1995-09-01
NO1995008I1 (no) 1995-09-22
NL940001I2 (nl) 1998-03-02
HU193146B (en) 1987-08-28
ATE20469T1 (de) 1986-07-15
IE812475L (en) 1982-04-23
FI813283L (fi) 1982-04-24
NL940001I1 (nl) 1994-03-01
KR880001843B1 (ko) 1988-09-21
DE19575012I2 (de) 2002-01-24
ES506414A0 (es) 1983-10-01
DE3174844D1 (en) 1986-07-24
PH21916A (en) 1988-04-08
EP0050800B1 (en) 1986-06-18
NO164983C (no) 1990-12-05

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