SG189830A1 - 4- (5-cyano-pyrazol-1-yl) -piperidine derivatives as gpr 119 modulators - Google Patents
4- (5-cyano-pyrazol-1-yl) -piperidine derivatives as gpr 119 modulators Download PDFInfo
- Publication number
- SG189830A1 SG189830A1 SG2013023189A SG2013023189A SG189830A1 SG 189830 A1 SG189830 A1 SG 189830A1 SG 2013023189 A SG2013023189 A SG 2013023189A SG 2013023189 A SG2013023189 A SG 2013023189A SG 189830 A1 SG189830 A1 SG 189830A1
- Authority
- SG
- Singapore
- Prior art keywords
- methyl
- cyano
- carboxylate
- pyrazol
- piperidine
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- C—CHEMISTRY; METALLURGY
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Applications Claiming Priority (2)
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EP (1) | EP2643310A1 (es) |
JP (1) | JP2013543885A (es) |
KR (1) | KR20130083915A (es) |
CN (1) | CN103298801A (es) |
AP (1) | AP2013006809A0 (es) |
AR (1) | AR088121A1 (es) |
AU (1) | AU2011333427A1 (es) |
BR (1) | BR112013011865A2 (es) |
CA (1) | CA2814231A1 (es) |
CL (1) | CL2013001054A1 (es) |
CO (1) | CO6801716A2 (es) |
CR (1) | CR20130139A (es) |
CU (1) | CU20130059A7 (es) |
DO (1) | DOP2013000102A (es) |
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TW (1) | TWI433843B (es) |
UY (1) | UY33742A (es) |
WO (1) | WO2012069948A1 (es) |
ZA (1) | ZA201302362B (es) |
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CA2836487A1 (en) | 2011-06-09 | 2012-12-13 | Rhizen Pharmaceuticals Sa | Novel compounds as modulators of gpr-119 |
AU2013290100A1 (en) | 2012-07-11 | 2015-01-29 | Elcelyx Therapeutics, Inc. | Compositions comprising statins, biguanides and further agents for reducing cardiometabolic risk |
JP2017119628A (ja) * | 2014-05-09 | 2017-07-06 | 日産化学工業株式会社 | 置換アゾール化合物及び糖尿病治療薬 |
CN104610151A (zh) * | 2015-02-13 | 2015-05-13 | 佛山市赛维斯医药科技有限公司 | 含酰肼和烷氧苯类结构的化合物、其制备方法及用途 |
CN104892517A (zh) * | 2015-02-13 | 2015-09-09 | 佛山市赛维斯医药科技有限公司 | 酰肼类化合物、其制备方法及用途 |
CN104592120A (zh) * | 2015-02-13 | 2015-05-06 | 佛山市赛维斯医药科技有限公司 | 一种环丙基酰肼和甲氧苯类gpr119激动剂、制备方法及其用途 |
ES2883591T3 (es) | 2016-02-18 | 2021-12-09 | Syngenta Participations Ag | Derivados de pirazol pesticídicamente activos |
CN106631992B (zh) * | 2017-01-05 | 2019-01-18 | 桑迪亚医药技术(上海)有限责任公司 | 一种4-氧-3,4-二氢-2h-吡啶-1-甲酸叔丁酯的合成方法 |
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WO2009014910A2 (en) * | 2007-07-19 | 2009-01-29 | Metabolex, Inc. | N-azacyclic substituted pyrrole, pyrazole, imidazole, triazole and tetrazole derivatives as agonists of the rup3 or gpr119 receptor for the treatment of diabetes and metabolic disorders |
US20090270404A1 (en) * | 2008-03-31 | 2009-10-29 | Metabolex, Inc. | Oxymethylene aryl compounds and uses thereof |
EA020106B1 (ru) * | 2009-06-05 | 2014-08-29 | Пфайзер Инк. | Производные l-(пиперидин-4-ил)пиразола в качестве модуляторов gpr119 |
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- 2011-11-09 MA MA35928A patent/MA34805B1/fr unknown
- 2011-11-09 AU AU2011333427A patent/AU2011333427A1/en not_active Abandoned
- 2011-11-09 MX MX2013004083A patent/MX2013004083A/es unknown
- 2011-11-09 EA EA201370118A patent/EA201370118A1/ru unknown
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- 2011-11-09 CN CN2011800550665A patent/CN103298801A/zh active Pending
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- 2011-11-09 WO PCT/IB2011/054996 patent/WO2012069948A1/en active Application Filing
- 2011-11-09 CA CA2814231A patent/CA2814231A1/en not_active Abandoned
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2013
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BR112013011865A2 (pt) | 2016-08-23 |
CU20130059A7 (es) | 2013-06-28 |
PE20140409A1 (es) | 2014-03-23 |
AR088121A1 (es) | 2014-05-14 |
NI201300044A (es) | 2013-08-01 |
JP2013543885A (ja) | 2013-12-09 |
DOP2013000102A (es) | 2013-07-15 |
GT201300135A (es) | 2015-02-19 |
KR20130083915A (ko) | 2013-07-23 |
CL2013001054A1 (es) | 2013-09-27 |
EA201370118A1 (ru) | 2013-12-30 |
TW201300373A (zh) | 2013-01-01 |
CA2814231A1 (en) | 2012-05-31 |
TWI433843B (zh) | 2014-04-11 |
MA34805B1 (fr) | 2014-01-02 |
WO2012069948A1 (en) | 2012-05-31 |
CO6801716A2 (es) | 2013-11-29 |
AP2013006809A0 (en) | 2013-04-30 |
ECSP13012630A (es) | 2013-07-31 |
ZA201302362B (en) | 2014-06-25 |
AU2011333427A1 (en) | 2013-04-11 |
UY33742A (es) | 2012-06-29 |
MX2013004083A (es) | 2013-06-13 |
CN103298801A (zh) | 2013-09-11 |
EP2643310A1 (en) | 2013-10-02 |
CR20130139A (es) | 2013-06-28 |
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