SG136958A1 - Antagonistic analogs of gh-rh (2003) - Google Patents

Antagonistic analogs of gh-rh (2003)

Info

Publication number
SG136958A1
SG136958A1 SG200716961-8A SG2007169618A SG136958A1 SG 136958 A1 SG136958 A1 SG 136958A1 SG 2007169618 A SG2007169618 A SG 2007169618A SG 136958 A1 SG136958 A1 SG 136958A1
Authority
SG
Singapore
Prior art keywords
antagonistic analogs
antagonistic
analogs
Prior art date
Application number
SG200716961-8A
Other languages
English (en)
Inventor
Andrew V Schally
Jozsef Varga
Marta Zarandi
Ren Zhi Cai
Original Assignee
Univ Tulane
Us Health
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Univ Tulane, Us Health filed Critical Univ Tulane
Publication of SG136958A1 publication Critical patent/SG136958A1/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/60—Growth hormone-releasing factor [GH-RF], i.e. somatoliberin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/06—Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Endocrinology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biophysics (AREA)
  • Toxicology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Zoology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Diabetes (AREA)
  • Analytical Chemistry (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
SG200716961-8A 2003-08-05 2004-07-26 Antagonistic analogs of gh-rh (2003) SG136958A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US49270603P 2003-08-05 2003-08-05

Publications (1)

Publication Number Publication Date
SG136958A1 true SG136958A1 (en) 2007-11-29

Family

ID=34193144

Family Applications (1)

Application Number Title Priority Date Filing Date
SG200716961-8A SG136958A1 (en) 2003-08-05 2004-07-26 Antagonistic analogs of gh-rh (2003)

Country Status (19)

Country Link
US (1) US7452865B2 (no)
EP (1) EP1651662A4 (no)
JP (1) JP2007526900A (no)
KR (1) KR20060088875A (no)
CN (1) CN1871020A (no)
AR (1) AR049149A1 (no)
AU (1) AU2004265280A1 (no)
BR (1) BRPI0413257A (no)
CA (1) CA2534436A1 (no)
IL (1) IL173201A0 (no)
MX (1) MXPA06001369A (no)
NO (1) NO20061060L (no)
PL (1) PL380437A1 (no)
RS (1) RS20060086A (no)
RU (1) RU2335506C2 (no)
SG (1) SG136958A1 (no)
TW (1) TW200517400A (no)
WO (1) WO2005016953A2 (no)
ZA (1) ZA200600966B (no)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009108364A2 (en) * 2008-02-27 2009-09-03 Ipsen Pharma S.A.S. Antagonistic analogues of ghrh
US8691942B2 (en) 2008-03-28 2014-04-08 University Of Miami N- and C- terminal substituted antagonistic analogs of GH-RH
BRPI0910873A2 (pt) * 2008-03-28 2015-10-06 Us Of America Represented By The Dept Of Veterans Affairs análogos antagonistas de gh-rh substituídos nos terminais n e c
KR101731655B1 (ko) * 2008-06-12 2017-05-11 입센 바이오이노베이션 리미티드 암 억제 방법
EP3590956A1 (en) * 2008-06-12 2020-01-08 Ipsen Bioinnovation Limited Suppression of neuroendocrine diseases
US8796216B2 (en) 2008-06-12 2014-08-05 Syntaxin Limited Suppression of neuroendocrine diseases
US8227421B2 (en) * 2009-09-17 2012-07-24 University Of Miami Fluorinated GHRH antagonists
US8980249B2 (en) 2010-06-03 2015-03-17 University Of Miami Agonists of growth hormone releasing hormone as effectors for survival and proliferation of pancreatic islets
BR112013027150A2 (pt) 2011-04-21 2017-06-06 Theratechnologies Inc thera
US9079974B2 (en) * 2011-12-21 2015-07-14 The University Of Miami GH-RH analogs with potent agonistic effects
EP2866894A4 (en) * 2012-06-27 2016-03-16 Univ Miami COMPOSITION AND METHOD FOR THE TREATMENT OF MORBUS ALZHEIMER
WO2014100809A2 (en) 2012-12-21 2014-06-26 University Of Miami Ghrh agonists for the treatment of ischemic disorders
WO2014100816A2 (en) 2012-12-21 2014-06-26 University Of Miami Ghrh agonists for islet cell transplantation and function and the treatment of diabetes
EP3920961A4 (en) 2019-02-08 2022-12-14 United States Government as represented by the Department of Veterans Affairs GROWTH HORMONE RELEASING HORMONE ANTAGONISTS AND THEIR USES
WO2021222129A1 (en) 2020-04-27 2021-11-04 The University Of Miami Method of treating an inflammatory disorder
CN114195881B (zh) * 2021-12-16 2022-09-16 浙江湃肽生物股份有限公司 一种制备醋酸舍莫瑞林的方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5942489A (en) * 1996-05-03 1999-08-24 The Administrators Of The Tulane Educational Fund HGH-RH(1-29)NH2 analogues having antagonistic activity
US6057422A (en) * 1998-11-25 2000-05-02 The Administrators Of The Tulane Educational Fund Antagonistic analogs of GH-RH inhibiting IGF-I and -II

Also Published As

Publication number Publication date
US7452865B2 (en) 2008-11-18
RU2006106701A (ru) 2007-09-20
TW200517400A (en) 2005-06-01
MXPA06001369A (es) 2007-02-19
CA2534436A1 (en) 2005-02-24
WO2005016953A2 (en) 2005-02-24
ZA200600966B (en) 2007-05-30
KR20060088875A (ko) 2006-08-07
US20070042950A1 (en) 2007-02-22
NO20061060L (no) 2006-05-03
IL173201A0 (en) 2006-06-11
CN1871020A (zh) 2006-11-29
PL380437A1 (pl) 2007-01-22
EP1651662A2 (en) 2006-05-03
RS20060086A (en) 2008-08-07
AR049149A1 (es) 2006-07-05
BRPI0413257A (pt) 2006-10-03
AU2004265280A1 (en) 2005-02-24
RU2335506C2 (ru) 2008-10-10
WO2005016953A3 (en) 2006-02-09
EP1651662A4 (en) 2009-07-01
JP2007526900A (ja) 2007-09-20

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