SG11202011544UA - Vmat2 inhibitor compounds, compositions, and methods relating thereto - Google Patents

Vmat2 inhibitor compounds, compositions, and methods relating thereto

Info

Publication number
SG11202011544UA
SG11202011544UA SG11202011544UA SG11202011544UA SG11202011544UA SG 11202011544U A SG11202011544U A SG 11202011544UA SG 11202011544U A SG11202011544U A SG 11202011544UA SG 11202011544U A SG11202011544U A SG 11202011544UA SG 11202011544U A SG11202011544U A SG 11202011544UA
Authority
SG
Singapore
Prior art keywords
compositions
inhibitor compounds
methods relating
vmat2 inhibitor
vmat2
Prior art date
Application number
SG11202011544UA
Other languages
English (en)
Inventor
Christopher F O'brien
Nicole Harriott
Original Assignee
Neurocrine Biosciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Neurocrine Biosciences Inc filed Critical Neurocrine Biosciences Inc
Publication of SG11202011544UA publication Critical patent/SG11202011544UA/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Neurosurgery (AREA)
  • General Chemical & Material Sciences (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
SG11202011544UA 2018-06-14 2019-06-13 Vmat2 inhibitor compounds, compositions, and methods relating thereto SG11202011544UA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201862684935P 2018-06-14 2018-06-14
PCT/US2019/037046 WO2019241555A1 (en) 2018-06-14 2019-06-13 Vmat2 inhibitor compounds, compositions, and methods relating thereto

Publications (1)

Publication Number Publication Date
SG11202011544UA true SG11202011544UA (en) 2020-12-30

Family

ID=67263041

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11202011544UA SG11202011544UA (en) 2018-06-14 2019-06-13 Vmat2 inhibitor compounds, compositions, and methods relating thereto

Country Status (16)

Country Link
EP (2) EP4691560A3 (https=)
JP (2) JP2021528386A (https=)
KR (1) KR20210021006A (https=)
CN (1) CN112638387A (https=)
AU (1) AU2019287524A1 (https=)
BR (1) BR112020024018A2 (https=)
CA (1) CA3100694A1 (https=)
EA (1) EA202092750A1 (https=)
IL (1) IL278758A (https=)
JO (1) JOP20200298A1 (https=)
MA (1) MA52896A (https=)
MX (1) MX2020013004A (https=)
PH (1) PH12020552088A1 (https=)
SG (1) SG11202011544UA (https=)
TW (1) TW202011963A (https=)
WO (1) WO2019241555A1 (https=)

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ES3024958T3 (en) 2017-09-21 2025-06-05 Neurocrine Biosciences Inc High dosage valbenazine formulation and compositions, methods, and kits related thereto
KR20250070134A (ko) 2017-10-10 2025-05-20 뉴로크린 바이오사이언시즈 인코퍼레이티드 특정 vmat2 억제제의 투여 방법
JP2021502959A (ja) 2017-10-10 2021-02-04 ニューロクライン バイオサイエンシーズ，インコーポレイテッド 特定のｖｍａｔ２インヒビターを投与するための方法
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US20250000805A1 (en) * 2021-10-29 2025-01-02 Neurocrine Biosciences, Inc. Valbenazine compositions

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Also Published As

Publication number Publication date
JP2024114905A (ja) 2024-08-23
EP4691560A2 (en) 2026-02-11
MX2020013004A (es) 2021-02-17
EA202092750A1 (ru) 2021-05-13
TW202011963A (zh) 2020-04-01
CA3100694A1 (en) 2019-12-19
JOP20200298A1 (ar) 2020-11-22
IL278758A (en) 2021-01-31
MA52896A (fr) 2021-04-21
AU2019287524A1 (en) 2020-12-24
CN112638387A (zh) 2021-04-09
EP4691560A3 (en) 2026-04-15
BR112020024018A2 (pt) 2021-02-23
KR20210021006A (ko) 2021-02-24
EP3806856A1 (en) 2021-04-21
JP2021528386A (ja) 2021-10-21
WO2019241555A1 (en) 2019-12-19
PH12020552088A1 (en) 2021-08-02

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