SG11201508924XA - Pd-CATALYZED COUPLING OF PYRAZOLE AMIDES - Google Patents

Pd-CATALYZED COUPLING OF PYRAZOLE AMIDES

Info

Publication number
SG11201508924XA
SG11201508924XA SG11201508924XA SG11201508924XA SG11201508924XA SG 11201508924X A SG11201508924X A SG 11201508924XA SG 11201508924X A SG11201508924X A SG 11201508924XA SG 11201508924X A SG11201508924X A SG 11201508924XA SG 11201508924X A SG11201508924X A SG 11201508924XA
Authority
SG
Singapore
Prior art keywords
catalyzed coupling
pyrazole amides
pyrazole
amides
catalyzed
Prior art date
Application number
SG11201508924XA
Other languages
English (en)
Inventor
Serena Maria Fantasia
Kurt Puentener
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of SG11201508924XA publication Critical patent/SG11201508924XA/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Engineering & Computer Science (AREA)
  • Materials Engineering (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
SG11201508924XA 2013-04-30 2014-04-28 Pd-CATALYZED COUPLING OF PYRAZOLE AMIDES SG11201508924XA (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP13166027 2013-04-30
PCT/EP2014/058549 WO2014177493A1 (fr) 2013-04-30 2014-04-28 Couplage de pyrazole-amides catalysé par pd

Publications (1)

Publication Number Publication Date
SG11201508924XA true SG11201508924XA (en) 2015-11-27

Family

ID=48190360

Family Applications (1)

Application Number Title Priority Date Filing Date
SG11201508924XA SG11201508924XA (en) 2013-04-30 2014-04-28 Pd-CATALYZED COUPLING OF PYRAZOLE AMIDES

Country Status (21)

Country Link
US (1) US9505759B2 (fr)
EP (1) EP2991984B1 (fr)
JP (1) JP2016520047A (fr)
KR (1) KR20160002839A (fr)
CN (1) CN105164126B (fr)
AR (1) AR096118A1 (fr)
AU (1) AU2014261512B2 (fr)
BR (1) BR112015026132A2 (fr)
CA (1) CA2909477A1 (fr)
DK (1) DK2991984T3 (fr)
ES (1) ES2622754T3 (fr)
HK (1) HK1213557A1 (fr)
HU (1) HUE032407T2 (fr)
IL (1) IL242032B (fr)
MX (1) MX2015014729A (fr)
MY (1) MY169128A (fr)
PL (1) PL2991984T3 (fr)
RU (1) RU2663834C2 (fr)
SG (1) SG11201508924XA (fr)
SI (1) SI2991984T1 (fr)
WO (1) WO2014177493A1 (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP6568855B2 (ja) 2014-07-30 2019-08-28 持田製薬株式会社 ピラゾール誘導体の製造方法
WO2016017719A1 (fr) * 2014-07-30 2016-02-04 持田製薬株式会社 Procédé de fabrication d'un dérivé de pyrazole
WO2020021024A1 (fr) * 2018-07-26 2020-01-30 Phenex Pharmaceuticals Ag Composés bicycliques substitués en tant que modulateurs du récepteur d'hydrocarbures aryle (ahr)
CA3180793A1 (fr) 2020-06-05 2021-12-09 George GARIBALDI Utilisation d'un inhibiteur de phosphodiesterase 10 pour le traitement du syndrome de tourette
WO2023164178A2 (fr) * 2022-02-25 2023-08-31 Journey Colab Corp. Procédés de préparation de mescaline

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SE0102808D0 (sv) * 2001-08-22 2001-08-22 Astrazeneca Ab New compounds
MY147647A (en) * 2005-03-21 2012-12-31 S Bio Pte Ltd Imidazo [1,2-a] pyridine derivatives : preparation and pharmaceutical applications
WO2011036127A1 (fr) * 2009-09-24 2011-03-31 F. Hoffmann-La Roche Ag Dérivés d'imidazopyridine ou d'imidazopyrimidine en tant qu'inhibiteurs de phosphodiestérase 10a
US8349824B2 (en) 2010-12-07 2013-01-08 Hoffmann-La Roche Inc. Triazolopyridine compounds
KR101778354B1 (ko) * 2011-08-18 2017-09-13 니뽄 신야쿠 가부시키가이샤 헤테로환 유도체 및 의약
WO2013041472A1 (fr) * 2011-09-19 2013-03-28 F. Hoffmann-La Roche Ag Composés triazolopyridines en tant qu'inhibiteurs de pde10a

Also Published As

Publication number Publication date
AR096118A1 (es) 2015-12-09
AU2014261512B2 (en) 2017-10-05
KR20160002839A (ko) 2016-01-08
DK2991984T3 (en) 2017-05-08
CA2909477A1 (fr) 2014-11-06
RU2663834C2 (ru) 2018-08-10
CN105164126A (zh) 2015-12-16
BR112015026132A2 (pt) 2017-07-25
HUE032407T2 (en) 2017-09-28
MX2015014729A (es) 2016-03-07
EP2991984A1 (fr) 2016-03-09
ES2622754T3 (es) 2017-07-07
AU2014261512A1 (en) 2015-10-15
US9505759B2 (en) 2016-11-29
RU2015145721A (ru) 2017-06-07
WO2014177493A1 (fr) 2014-11-06
CN105164126B (zh) 2017-05-31
PL2991984T3 (pl) 2017-07-31
US20160046628A1 (en) 2016-02-18
IL242032B (en) 2018-06-28
HK1213557A1 (zh) 2016-07-08
MY169128A (en) 2019-02-18
JP2016520047A (ja) 2016-07-11
SI2991984T1 (sl) 2017-05-31
EP2991984B1 (fr) 2017-03-08

Similar Documents

Publication Publication Date Title
HK1223097A1 (zh) 雜芳基取代的吡唑
HK1223098A1 (zh) 雜芳基取代的吡唑
HK1221224A1 (zh) 依洛昔巴特的結晶修飾物
ZA201505397B (en) Novel pyrazole derivative
SG11201507156UA (en) Electrochemical coupling of anilines
HK1222852A1 (zh) 二氨基雜芳基取代的吡唑
EP2960536A4 (fr) Accouplement
HK1218757A1 (zh) 用作卵泡刺激素受體調節劑的吡唑化合物及其用途
HRP20181710T1 (hr) Uporaba derivata benzimidazol-prolina
GB2522768B (en) Coupling
ZA201508015B (en) Solid forms of fungicidal pyrazoles
GB2522767B (en) Coupling
GB2519790B (en) Configuration of network devices
HK1213557A1 (zh) 吡唑酰胺的 -催化偶聯
AU352098S (en) Coupling
GB2539112B (en) Chlorination of sucrose-6-esters
HRP20180644T1 (hr) Derivat pirazola
GB2515540B (en) Coupling
ZA201402420B (en) Tow-hitch coupling
GB201322366D0 (en) Chlorination of sucrose-6-esters
GB201314779D0 (en) Chlorination of sucrose-6-esters