SG10201604731SA - Compounds, compositions and methods useful for cholesterol mobilisation - Google Patents

Compounds, compositions and methods useful for cholesterol mobilisation

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Publication number
SG10201604731SA
SG10201604731SA SG10201604731SA SG10201604731SA SG10201604731SA SG 10201604731S A SG10201604731S A SG 10201604731SA SG 10201604731S A SG10201604731S A SG 10201604731SA SG 10201604731S A SG10201604731S A SG 10201604731SA SG 10201604731S A SG10201604731S A SG 10201604731SA
Authority
SG
Singapore
Prior art keywords
compositions
compounds
methods useful
mobilisation
cholesterol
Prior art date
Application number
SG10201604731SA
Other languages
English (en)
Inventor
Daniela Carmen Oniciu
Jean-Louis Henri Dasseux
Ronald Barbaras
Valery Kochubey
Dmitry Kovalsky
Oleg Gennadievich Rodin
Otto Geoffroy
Anna Rzepiela
Original Assignee
Cerenis Therapeutics Holding Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cerenis Therapeutics Holding Sa filed Critical Cerenis Therapeutics Holding Sa
Publication of SG10201604731SA publication Critical patent/SG10201604731SA/en

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    • A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
    • A61K31/5375—1,4-Oxazines, e.g. morpholine
    • A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
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